JP2005524648A5 - - Google Patents
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- Publication number
- JP2005524648A5 JP2005524648A5 JP2003570793A JP2003570793A JP2005524648A5 JP 2005524648 A5 JP2005524648 A5 JP 2005524648A5 JP 2003570793 A JP2003570793 A JP 2003570793A JP 2003570793 A JP2003570793 A JP 2003570793A JP 2005524648 A5 JP2005524648 A5 JP 2005524648A5
- Authority
- JP
- Japan
- Prior art keywords
- carrier peptide
- composition according
- amino acids
- peptide comprises
- opioid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000000203 mixture Substances 0.000 claims 10
- 108090000765 processed proteins & peptides Proteins 0.000 claims 10
- 150000001413 amino acids Chemical class 0.000 claims 8
- 239000008194 pharmaceutical composition Substances 0.000 claims 5
- 239000003814 drug Substances 0.000 claims 2
- 238000004519 manufacturing process Methods 0.000 claims 2
- BRUQQQPBMZOVGD-XFKAJCMBSA-N Oxycodone Chemical group O=C([C@@H]1O2)CC[C@@]3(O)[C@H]4CC5=CC=C(OC)C2=C5[C@@]13CCN4C BRUQQQPBMZOVGD-XFKAJCMBSA-N 0.000 claims 1
- 125000003275 alpha amino acid group Chemical group 0.000 claims 1
- XYYVYLMBEZUESM-UHFFFAOYSA-N dihydrocodeine Natural products C1C(N(CCC234)C)C2C=CC(=O)C3OC2=C4C1=CC=C2OC XYYVYLMBEZUESM-UHFFFAOYSA-N 0.000 claims 1
- 230000002743 euphoric effect Effects 0.000 claims 1
- LLPOLZWFYMWNKH-CMKMFDCUSA-N hydrocodone Chemical group C([C@H]1[C@H](N(CC[C@@]112)C)C3)CC(=O)[C@@H]1OC1=C2C3=CC=C1OC LLPOLZWFYMWNKH-CMKMFDCUSA-N 0.000 claims 1
- 229960000240 hydrocodone Drugs 0.000 claims 1
- OROGSEYTTFOCAN-UHFFFAOYSA-N hydrocodone Natural products C1C(N(CCC234)C)C2C=CC(O)C3OC2=C4C1=CC=C2OC OROGSEYTTFOCAN-UHFFFAOYSA-N 0.000 claims 1
- 229960002085 oxycodone Drugs 0.000 claims 1
- 230000001225 therapeutic effect Effects 0.000 claims 1
- LLPOLZWFYMWNKH-UHFFFAOYSA-N trans-dihydrocodeinone Natural products C1C(N(CCC234)C)C2CCC(=O)C3OC2=C4C1=CC=C2OC LLPOLZWFYMWNKH-UHFFFAOYSA-N 0.000 claims 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35836802P | 2002-02-22 | 2002-02-22 | |
| US60/358,368 | 2002-02-22 | ||
| US36208202P | 2002-03-07 | 2002-03-07 | |
| US60/362,082 | 2002-03-07 | ||
| PCT/US2003/005525 WO2003072046A2 (en) | 2002-02-22 | 2003-02-24 | Novel sustained release pharmaceutical compounds to prevent abuse of controlled substances |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005524648A JP2005524648A (ja) | 2005-08-18 |
| JP2005524648A5 true JP2005524648A5 (enExample) | 2006-09-07 |
| JP4878732B2 JP4878732B2 (ja) | 2012-02-15 |
Family
ID=27767540
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003570793A Expired - Fee Related JP4878732B2 (ja) | 2002-02-22 | 2003-02-24 | 規制物質の濫用を防ぐための新規な持続放出製薬化合物 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7622441B2 (enExample) |
| EP (2) | EP2319540A1 (enExample) |
| JP (1) | JP4878732B2 (enExample) |
| KR (1) | KR100822498B1 (enExample) |
| AU (2) | AU2003219863C1 (enExample) |
| CA (1) | CA2477004C (enExample) |
| ES (1) | ES2500117T3 (enExample) |
| IL (2) | IL163667A0 (enExample) |
| WO (1) | WO2003072046A2 (enExample) |
Families Citing this family (69)
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-
2003
- 2003-02-24 IL IL16366703A patent/IL163667A0/xx active IP Right Grant
- 2003-02-24 WO PCT/US2003/005525 patent/WO2003072046A2/en not_active Ceased
- 2003-02-24 CA CA2477004A patent/CA2477004C/en not_active Expired - Fee Related
- 2003-02-24 EP EP11151658A patent/EP2319540A1/en not_active Withdrawn
- 2003-02-24 AU AU2003219863A patent/AU2003219863C1/en not_active Ceased
- 2003-02-24 JP JP2003570793A patent/JP4878732B2/ja not_active Expired - Fee Related
- 2003-02-24 KR KR1020047013136A patent/KR100822498B1/ko not_active Expired - Fee Related
- 2003-02-24 ES ES03716144.5T patent/ES2500117T3/es not_active Expired - Lifetime
- 2003-02-24 EP EP03716144.5A patent/EP1531844B1/en not_active Expired - Lifetime
-
2004
- 2004-08-22 IL IL163667A patent/IL163667A/en not_active IP Right Cessation
- 2004-08-23 US US10/923,257 patent/US7622441B2/en not_active Expired - Fee Related
-
2008
- 2008-10-16 AU AU2008229978A patent/AU2008229978B2/en not_active Withdrawn - After Issue
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