JP2005507881A - 乾燥粉末医薬製剤 - Google Patents
乾燥粉末医薬製剤 Download PDFInfo
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- JP2005507881A JP2005507881A JP2003528494A JP2003528494A JP2005507881A JP 2005507881 A JP2005507881 A JP 2005507881A JP 2003528494 A JP2003528494 A JP 2003528494A JP 2003528494 A JP2003528494 A JP 2003528494A JP 2005507881 A JP2005507881 A JP 2005507881A
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- 238000005185 salting out Methods 0.000 description 1
- CDAISMWEOUEBRE-UHFFFAOYSA-N scyllo-inosotol Natural products OC1C(O)C(O)C(O)C(O)C1O CDAISMWEOUEBRE-UHFFFAOYSA-N 0.000 description 1
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Images
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Otolaryngology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
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| US32278301P | 2001-09-17 | 2001-09-17 | |
| PCT/US2002/029267 WO2003024396A2 (en) | 2001-09-17 | 2002-09-16 | Dry powder medicament formulations |
Publications (2)
| Publication Number | Publication Date |
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| JP2005507881A true JP2005507881A (ja) | 2005-03-24 |
| JP2005507881A5 JP2005507881A5 (https=) | 2005-12-22 |
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| JP2003528494A Pending JP2005507881A (ja) | 2001-09-17 | 2002-09-16 | 乾燥粉末医薬製剤 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US8337816B2 (https=) |
| EP (1) | EP1487417A4 (https=) |
| JP (1) | JP2005507881A (https=) |
| AU (1) | AU2002333644A1 (https=) |
| WO (1) | WO2003024396A2 (https=) |
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| JP2016539151A (ja) * | 2013-12-06 | 2016-12-15 | オリオン コーポレーション | 乾燥粉末吸入組成物の製造方法 |
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| US20040191176A1 (en) * | 2003-03-28 | 2004-09-30 | Kaplan Leonard W | Formulations for treatment of pulmonary disorders |
| CA2575957C (en) | 2003-09-02 | 2010-11-30 | Norton Healthcare Ltd. | Process for preparing a medicament |
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| KR20090057477A (ko) | 2001-09-14 | 2009-06-05 | 글락소 그룹 리미티드 | 호흡기 질환 치료용 펜에탄올아민 유도체 |
| US8337816B2 (en) | 2001-09-17 | 2012-12-25 | Glaxo Group Limited | Dry powder medicament formulations |
| US20030129242A1 (en) | 2002-01-04 | 2003-07-10 | Bosch H. William | Sterile filtered nanoparticulate formulations of budesonide and beclomethasone having tyloxapol as a surface stabilizer |
| US6559293B1 (en) * | 2002-02-15 | 2003-05-06 | Transform Pharmaceuticals, Inc. | Topiramate sodium trihydrate |
| GB0204719D0 (en) | 2002-02-28 | 2002-04-17 | Glaxo Group Ltd | Medicinal compounds |
| GB0208608D0 (en) | 2002-04-13 | 2002-05-22 | Glaxo Group Ltd | Composition |
| GB0208609D0 (en) | 2002-04-13 | 2002-05-22 | Glaxo Group Ltd | Compositions |
| JP2005523920A (ja) | 2002-04-25 | 2005-08-11 | グラクソ グループ リミテッド | フェネタノールアミン誘導体 |
| GB0217225D0 (en) | 2002-07-25 | 2002-09-04 | Glaxo Group Ltd | Medicinal compounds |
| GB0220730D0 (en) | 2002-09-06 | 2002-10-16 | Glaxo Group Ltd | Medicinal compounds |
| EP1554264B1 (en) | 2002-10-22 | 2007-08-08 | Glaxo Group Limited | Medicinal arylethanolamine compounds |
| GB0225030D0 (en) | 2002-10-28 | 2002-12-04 | Glaxo Group Ltd | Medicinal compounds |
| EP1556342B1 (en) | 2002-10-28 | 2008-03-26 | Glaxo Group Limited | Phenethanolamine derivative for the treatment of respiratory diseases |
| GB0225540D0 (en) | 2002-11-01 | 2002-12-11 | Glaxo Group Ltd | Medicinal compounds |
| GB0225535D0 (en) | 2002-11-01 | 2002-12-11 | Glaxo Group Ltd | Medicinal compounds |
| EP1646370A1 (en) | 2003-07-11 | 2006-04-19 | Glaxo Group Limited | Pharmaceutical formulations |
| GB0316341D0 (en) | 2003-07-11 | 2003-08-13 | Glaxo Group Ltd | Pharmaceutical formulations |
| EP1643973A1 (en) | 2003-07-11 | 2006-04-12 | Glaxo Group Limited | Pharmaceutical formulations comprising magnesium stearate |
-
2002
- 2002-09-16 US US10/489,491 patent/US8337816B2/en active Active
- 2002-09-16 EP EP02798971A patent/EP1487417A4/en not_active Withdrawn
- 2002-09-16 JP JP2003528494A patent/JP2005507881A/ja active Pending
- 2002-09-16 AU AU2002333644A patent/AU2002333644A1/en not_active Abandoned
- 2002-09-16 WO PCT/US2002/029267 patent/WO2003024396A2/en not_active Ceased
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2011019970A (ja) * | 2003-04-14 | 2011-02-03 | Vectura Group Plc | 投与効率を向上させるデバイス及び製薬組成 |
| JP2010509287A (ja) * | 2006-11-10 | 2010-03-25 | ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | 粉末を混合する方法 |
| JP2010533697A (ja) * | 2007-07-19 | 2010-10-28 | ノートン・ヘルスケアー リミテッド | ドライパウダー薬剤 |
| JP2016539151A (ja) * | 2013-12-06 | 2016-12-15 | オリオン コーポレーション | 乾燥粉末吸入組成物の製造方法 |
| JP2020510002A (ja) * | 2017-03-07 | 2020-04-02 | フィリップ・モーリス・プロダクツ・ソシエテ・アノニム | 吸入可能なニコチン製剤、およびその作製および使用方法 |
| KR20210002542A (ko) * | 2018-04-16 | 2021-01-08 | 줄리아 세티 | 갑상선 호르몬을 포함하는 흡입용 약학 건조 파우더 조성물(a pharmaceutical dry powder composition for inhalation comprising a thyroid hormone) |
| JP2021520397A (ja) * | 2018-04-16 | 2021-08-19 | ツェティ，ユリア | 甲状腺ホルモンを含む吸入用の薬学的乾燥粉末組成物 |
| JP7239604B2 (ja) | 2018-04-16 | 2023-03-14 | ツェティ，ユリア | 甲状腺ホルモンを含む吸入用の薬学的乾燥粉末組成物 |
| US11786460B2 (en) | 2018-04-16 | 2023-10-17 | Ioulia Tseti | Pharmaceutical dry powder composition for inhalation comprising a thyroid hormone |
| KR102913096B1 (ko) | 2018-04-16 | 2026-01-14 | 줄리아 세티 | 갑상선 호르몬을 포함하는 흡입용 약학 건조 파우더 조성물(a pharmaceutical dry powder composition for inhalation comprising a thyroid hormone) |
Also Published As
| Publication number | Publication date |
|---|---|
| US8337816B2 (en) | 2012-12-25 |
| EP1487417A2 (en) | 2004-12-22 |
| AU2002333644A1 (en) | 2003-04-01 |
| US20040241232A1 (en) | 2004-12-02 |
| WO2003024396A2 (en) | 2003-03-27 |
| WO2003024396A3 (en) | 2004-09-30 |
| EP1487417A4 (en) | 2010-03-17 |
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