JP2004520293A5 - - Google Patents
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- Publication number
- JP2004520293A5 JP2004520293A5 JP2002547935A JP2002547935A JP2004520293A5 JP 2004520293 A5 JP2004520293 A5 JP 2004520293A5 JP 2002547935 A JP2002547935 A JP 2002547935A JP 2002547935 A JP2002547935 A JP 2002547935A JP 2004520293 A5 JP2004520293 A5 JP 2004520293A5
- Authority
- JP
- Japan
- Prior art keywords
- mmol
- aminothiazol
- methoxyimino
- thia
- aza
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- YMWUJEATGCHHMB-UHFFFAOYSA-N Dichloromethane Chemical compound ClCCl YMWUJEATGCHHMB-UHFFFAOYSA-N 0.000 description 6
- -1 2-aminothiazol-4-yl Chemical group 0.000 description 2
- NFHFRUOZVGFOOS-UHFFFAOYSA-N palladium;triphenylphosphane Chemical compound [Pd].C1=CC=CC=C1P(C=1C=CC=CC=1)C1=CC=CC=C1.C1=CC=CC=C1P(C=1C=CC=CC=1)C1=CC=CC=C1.C1=CC=CC=C1P(C=1C=CC=CC=1)C1=CC=CC=C1.C1=CC=CC=C1P(C=1C=CC=CC=1)C1=CC=CC=C1 NFHFRUOZVGFOOS-UHFFFAOYSA-N 0.000 description 2
- RIOQSEWOXXDEQQ-UHFFFAOYSA-N triphenylphosphine Chemical compound C1=CC=CC=C1P(C=1C=CC=CC=1)C1=CC=CC=C1 RIOQSEWOXXDEQQ-UHFFFAOYSA-N 0.000 description 2
- SCNWTQPZTZMXBG-UHFFFAOYSA-N 2-methyloct-2-enoic acid Chemical compound CCCCCC=C(C)C(O)=O SCNWTQPZTZMXBG-UHFFFAOYSA-N 0.000 description 1
- VJZGUVFXFMVTRC-UHFFFAOYSA-N C1(=CC=CC=C1)S(=O)O.CC(=CCCCCC)C(=O)O Chemical compound C1(=CC=CC=C1)S(=O)O.CC(=CCCCCC)C(=O)O VJZGUVFXFMVTRC-UHFFFAOYSA-N 0.000 description 1
- JEHKKBHWRAXMCH-UHFFFAOYSA-N benzenesulfinic acid Chemical class O[S@@](=O)C1=CC=CC=C1 JEHKKBHWRAXMCH-UHFFFAOYSA-N 0.000 description 1
- 239000003054 catalyst Substances 0.000 description 1
- 239000011521 glass Substances 0.000 description 1
- 238000004128 high performance liquid chromatography Methods 0.000 description 1
- 238000000034 method Methods 0.000 description 1
- 239000012299 nitrogen atmosphere Substances 0.000 description 1
- 239000000047 product Substances 0.000 description 1
- 239000012265 solid product Substances 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25101400P | 2000-12-04 | 2000-12-04 | |
| PCT/IB2001/002225 WO2002046198A1 (en) | 2000-12-04 | 2001-11-22 | Coupling process and intermediates useful for preparing cephalosphorins |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004520293A JP2004520293A (ja) | 2004-07-08 |
| JP2004520293A5 true JP2004520293A5 (enExample) | 2007-11-15 |
Family
ID=22950114
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002547935A Pending JP2004520293A (ja) | 2000-12-04 | 2001-11-22 | セファロスポリン調製に有用なカップリング方法と中間体 |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US20020198375A1 (enExample) |
| EP (1) | EP1339722A1 (enExample) |
| JP (1) | JP2004520293A (enExample) |
| KR (1) | KR100526379B1 (enExample) |
| CN (1) | CN1243755C (enExample) |
| AR (1) | AR035511A1 (enExample) |
| AU (2) | AU2394302A (enExample) |
| BR (1) | BR0115870A (enExample) |
| CA (1) | CA2436848C (enExample) |
| CZ (1) | CZ20031525A3 (enExample) |
| HU (1) | HUP0400642A3 (enExample) |
| IL (1) | IL155714A0 (enExample) |
| MX (1) | MXPA03004937A (enExample) |
| PL (1) | PL362144A1 (enExample) |
| RU (1) | RU2237670C1 (enExample) |
| WO (1) | WO2002046198A1 (enExample) |
| ZA (1) | ZA200303670B (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20030051895A (ko) * | 2000-12-04 | 2003-06-25 | 후지사와 야꾸힝 고교 가부시키가이샤 | 아미노티아졸 유도체의 무수물의 제조 방법 |
| US7378408B2 (en) * | 2001-11-30 | 2008-05-27 | Pfizer Inc. | Methods of treatment and formulations of cephalosporin |
| RU2321590C1 (ru) * | 2004-03-09 | 2008-04-10 | Пфайзер Продактс Инк. | Способ получения промежуточных соединений цефалоспорина с использованием сложных эфиров альфа-йод-1-азетидинуксусной кислоты и триалкилфосфитов |
| SG194779A1 (en) | 2011-05-04 | 2013-12-30 | Univ Cornell | Multiblock copolymer films, methods of making same, and uses thereof |
| EP2740730B1 (en) | 2011-08-03 | 2016-11-16 | Kyowa Hakko Kirin Co., Ltd. | Dibenzooxepin derivative |
| CN102718779B (zh) * | 2012-05-25 | 2015-07-29 | 深圳致君制药有限公司 | 注射用头孢唑肟钠及其制备方法、原料药头孢唑肟钠的合成方法 |
| CN105254648B (zh) * | 2015-11-13 | 2018-04-03 | 广东温氏大华农生物科技有限公司 | 一种头孢维星及其钠盐的合成方法 |
| WO2018229580A1 (en) * | 2017-06-14 | 2018-12-20 | Aurobindo Pharma Ltd | An improved process for the preparation of cefovecin sodium |
| EP3697524A4 (en) | 2017-09-19 | 2021-09-01 | Terapore Technologies, Inc. | CHEMICALLY RESISTANT ISOPOROUS CROSS-LINKED BLOCK COPOLYMER STRUCTURE |
| EP3774003A4 (en) * | 2018-04-04 | 2022-01-05 | Terapore Technologies, Inc. | ENCAPSULATION PARTICLE FRACTIONATION DEVICES AND SYSTEMS AND THEIR METHODS OF USE |
| GB2575261B (en) | 2018-07-02 | 2022-03-09 | Norbrook Lab Ltd | Intermediates in the synthesis of C3-substituted cephalosporins |
| US11051804B2 (en) * | 2018-07-02 | 2021-07-06 | DePuy Synthes Products, Inc. | Orthopedic fixation system and method of use thereof |
| CN110396034A (zh) * | 2019-07-31 | 2019-11-01 | 上海应用技术大学 | 一种烯丙基化合物的制备方法 |
| CN111187284A (zh) * | 2020-03-10 | 2020-05-22 | 赵俊瑶 | 一种头孢克洛的制备方法 |
| CN111892612A (zh) * | 2020-07-31 | 2020-11-06 | 重庆医药高等专科学校 | 一种以青霉素钾盐为原料制备头孢维星的中间体异构化物及其制备方法 |
| CN112321611B (zh) * | 2020-10-29 | 2022-05-06 | 湖北凌晟药业有限公司 | 一种头孢沙定母核的制备方法 |
| CN115873021A (zh) * | 2022-12-19 | 2023-03-31 | 华北制药集团动物保健品有限责任公司 | 一种头孢维星钠的制备方法 |
| CN116731039B (zh) * | 2023-06-12 | 2025-02-18 | 重庆汉佩生物科技有限公司 | 头孢维星衍生物的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY106399A (en) * | 1990-07-24 | 1995-05-30 | Pfizer | Cephalosporins and homologeus, preparation and pharmaceutical composition |
| US6001997A (en) * | 1990-07-24 | 1999-12-14 | Bateson; John Hargreaves | Cephalosporins and homologues, preparations and pharmaceutical compositions |
| GB9212609D0 (en) * | 1992-06-13 | 1992-07-29 | Smithkline Beecham Plc | Novel compounds |
| GB9424847D0 (en) * | 1994-12-09 | 1995-02-08 | Smithkline Beecham Plc | Novel process |
| GB2300856A (en) * | 1995-05-16 | 1996-11-20 | Pfizer Ltd | Beta-lactam preparation |
| GB0019124D0 (en) * | 2000-08-03 | 2000-09-27 | Pfizer | Novel process |
| DE60117876T2 (de) * | 2000-12-04 | 2006-08-31 | Pfizer Products Inc., Groton | Verfahren und esterderivate zur herstellung von cephalosphorinen |
-
2001
- 2001-11-22 JP JP2002547935A patent/JP2004520293A/ja active Pending
- 2001-11-22 IL IL15571401A patent/IL155714A0/xx unknown
- 2001-11-22 CZ CZ20031525A patent/CZ20031525A3/cs unknown
- 2001-11-22 PL PL01362144A patent/PL362144A1/xx not_active Application Discontinuation
- 2001-11-22 HU HU0400642A patent/HUP0400642A3/hu unknown
- 2001-11-22 BR BR0115870-8A patent/BR0115870A/pt not_active IP Right Cessation
- 2001-11-22 AU AU2394302A patent/AU2394302A/xx active Pending
- 2001-11-22 KR KR10-2003-7007396A patent/KR100526379B1/ko not_active Expired - Fee Related
- 2001-11-22 CN CNB018199623A patent/CN1243755C/zh not_active Expired - Fee Related
- 2001-11-22 WO PCT/IB2001/002225 patent/WO2002046198A1/en not_active Ceased
- 2001-11-22 AU AU2002223943A patent/AU2002223943B2/en not_active Ceased
- 2001-11-22 RU RU2003116519/04A patent/RU2237670C1/ru active
- 2001-11-22 EP EP01999227A patent/EP1339722A1/en not_active Withdrawn
- 2001-11-22 MX MXPA03004937A patent/MXPA03004937A/es active IP Right Grant
- 2001-11-22 CA CA002436848A patent/CA2436848C/en not_active Expired - Fee Related
- 2001-12-03 AR ARP010105609A patent/AR035511A1/es not_active Application Discontinuation
- 2001-12-04 US US10/006,279 patent/US20020198375A1/en not_active Abandoned
-
2003
- 2003-05-13 ZA ZA200303670A patent/ZA200303670B/en unknown
-
2004
- 2004-02-11 US US10/776,795 patent/US7129350B2/en not_active Expired - Lifetime
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