JP2004509079A - 効力が増大した修飾生体ペプチド - Google Patents
効力が増大した修飾生体ペプチド Download PDFInfo
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- JP2004509079A JP2004509079A JP2002515924A JP2002515924A JP2004509079A JP 2004509079 A JP2004509079 A JP 2004509079A JP 2002515924 A JP2002515924 A JP 2002515924A JP 2002515924 A JP2002515924 A JP 2002515924A JP 2004509079 A JP2004509079 A JP 2004509079A
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- C07K14/575—Hormones
- C07K14/585—Calcitonins
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- C07K14/595—Gastrins; Cholecystokinins [CCK]
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- C07K14/60—Growth hormone-releasing factor [GH-RF], i.e. somatoliberin
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- C07K14/575—Hormones
- C07K14/605—Glucagons
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- C07K14/575—Hormones
- C07K14/635—Parathyroid hormone, i.e. parathormone; Parathyroid hormone-related peptides
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- C07K14/575—Hormones
- C07K14/65—Insulin-like growth factors, i.e. somatomedins, e.g. IGF-1, IGF-2
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- C07K14/575—Hormones
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- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
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- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/675—Beta-endorphins
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- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/68—Melanocyte-stimulating hormone [MSH]
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/695—Corticotropin [ACTH]
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- C—CHEMISTRY; METALLURGY
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/78—Connective tissue peptides, e.g. collagen, elastin, laminin, fibronectin, vitronectin or cold insoluble globulin [CIG]
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- C—CHEMISTRY; METALLURGY
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- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
- C07K7/086—Bombesin; Related peptides
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- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US22261900P | 2000-08-02 | 2000-08-02 | |
| PCT/CA2001/001119 WO2002010195A2 (en) | 2000-08-02 | 2001-08-02 | Modified peptides with increased potency |
Publications (2)
| Publication Number | Publication Date |
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| JP2004509079A true JP2004509079A (ja) | 2004-03-25 |
| JP2004509079A5 JP2004509079A5 (enExample) | 2005-08-18 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2002515924A Pending JP2004509079A (ja) | 2000-08-02 | 2001-08-02 | 効力が増大した修飾生体ペプチド |
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| US (1) | US20030204063A1 (enExample) |
| EP (1) | EP1305338A2 (enExample) |
| JP (1) | JP2004509079A (enExample) |
| CN (1) | CN1454214A (enExample) |
| AU (1) | AU2001279526A1 (enExample) |
| BR (1) | BR0113178A (enExample) |
| CA (1) | CA2417100A1 (enExample) |
| WO (1) | WO2002010195A2 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004508410A (ja) * | 2000-09-18 | 2004-03-18 | オステオミーター・ビオテク・エー／エス | Ｇｌｐ−１及びｇｌｐ−２ペプチドの使用方法 |
| JP2011508728A (ja) * | 2007-12-21 | 2011-03-17 | ビーエーエスエフ ソシエタス・ヨーロピア | ペプチドを含有するフケ防止組成物 |
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| US7186683B2 (en) | 2000-09-18 | 2007-03-06 | Sanos Bioscience A/S | Use of GLP for the treatment, prevention, diagnosis, and prognosis of bone-related and nutrition-related disorders |
| WO2002048192A2 (en) * | 2000-12-13 | 2002-06-20 | Eli Lilly And Company | Amidated glucagon-like peptide-1 |
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| EP1837031B1 (en) | 2002-06-07 | 2009-10-14 | Waratah Pharmaceuticals, Inc. | Compositions and methods for treating diabetes |
| US20080214437A1 (en) * | 2002-09-06 | 2008-09-04 | Mohapatra Shyam S | Methods and compositions for reducing activity of the atrial natriuretic peptide receptor and for treatment of diseases |
| WO2004022003A2 (en) * | 2002-09-06 | 2004-03-18 | University Of South Florida | Materials and methods for treatment of allergic diseases |
| WO2004022579A2 (en) * | 2002-09-06 | 2004-03-18 | University Of South Florida | Cellular delivery of natriuretic peptides |
| WO2004027064A2 (en) * | 2002-09-18 | 2004-04-01 | Centre Hospitalier De L'universite De Montreal (Chum) | Ghrh analogues |
| US7067488B2 (en) | 2002-09-25 | 2006-06-27 | Theratechnologies Inc. | Modified GLP-1 peptides with increased biological potency |
| US8603969B2 (en) * | 2004-02-11 | 2013-12-10 | Amylin Pharmaceuticals, Llc | Pancreatic polypeptide family motifs and polypeptides comprising the same |
| WO2005094420A2 (en) * | 2004-02-17 | 2005-10-13 | University Of South Florida | Materials and methods for treatment of inflammatory and cell proliferation disorders |
| CA2580919A1 (en) | 2004-10-25 | 2006-05-04 | Cytos Biotechnology Ag | Gastric inhibitory polypeptide (gip) antigen arrays and uses thereof |
| GB0426146D0 (en) | 2004-11-29 | 2004-12-29 | Bioxell Spa | Therapeutic peptides and method |
| WO2006086769A2 (en) | 2005-02-11 | 2006-08-17 | Amylin Pharmaceuticals, Inc. | Gip analog and hybrid polypeptides with selectable properties |
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| WO2007028632A2 (en) * | 2005-09-08 | 2007-03-15 | Uutech Limited | Analogs of gastric inhibitory polypeptide as a treatment for age related decreased pancreatic beta cell function |
| EP1943274A2 (en) * | 2005-09-08 | 2008-07-16 | Uutech Limited | Treatment of diabetes related obesity |
| EP1782819A1 (en) * | 2005-11-03 | 2007-05-09 | Cognis IP Management GmbH | Oligopeptides and their use |
| WO2007056362A2 (en) | 2005-11-07 | 2007-05-18 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting physiological solubility and stability |
| CA2656990A1 (en) * | 2006-04-28 | 2007-11-08 | University Of South Florida | Materials and methods for reducing inflammation by inhibition of the atrial natriuretic peptide receptor |
| US8497240B2 (en) | 2006-08-17 | 2013-07-30 | Amylin Pharmaceuticals, Llc | DPP-IV resistant GIP hybrid polypeptides with selectable properties |
| US20100190697A1 (en) * | 2006-09-13 | 2010-07-29 | The Trustees Of Columbia University In The City If | Undercarboxylated/uncarboxylated osteocalcin increases beta-cell proliferation, insulin secretion, insulin sensitivity, glucose tolerance and decreases fat mass |
| AU2006350707A1 (en) * | 2006-11-08 | 2008-05-15 | Chongxi Yu | Transdermal delivery systems of peptides and related compounds |
| CA2674354A1 (en) * | 2007-01-05 | 2008-07-17 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting enhanced solubility in physiological ph buffers |
| EP2118123B1 (en) | 2007-01-31 | 2015-10-14 | Dana-Farber Cancer Institute, Inc. | Stabilized p53 peptides and uses thereof |
| EA017849B1 (ru) | 2007-02-15 | 2013-03-29 | Индиана Юниверсити Рисерч Энд Текнолоджи Корпорейшн | Соагонисты глюкагоновых/glp-1-рецепторов |
| EP3159352B1 (en) | 2007-03-28 | 2023-08-02 | President and Fellows of Harvard College | Stitched polypeptides |
| WO2008145701A1 (en) * | 2007-05-29 | 2008-12-04 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Method for predicting the outcome of a critically ill patient |
| WO2009040006A1 (en) * | 2007-09-11 | 2009-04-02 | Mondobiotech Laboratories Ag | Spantide for therapeutic uses |
| WO2009058734A1 (en) * | 2007-10-30 | 2009-05-07 | Indiana University Research And Technology Corporation | Compounds exhibiting glucagon antagonist and glp-1 agonist activity |
| AU2008318986B2 (en) | 2007-10-30 | 2014-12-04 | Indiana University Research And Technology Corporation | Glucagon antagonists |
| JP2011511778A (ja) * | 2008-01-30 | 2011-04-14 | インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーション | エステルに基づいたペプチドプロドラッグ |
| US8450270B2 (en) | 2008-06-17 | 2013-05-28 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting enhanced solubility and stability in physiological pH buffers |
| PA8830501A1 (es) | 2008-06-17 | 2010-07-27 | Univ Indiana Res & Tech Corp | Co-agonistas del receptor de glucagon/glp-1 |
| EA020326B9 (ru) | 2008-06-17 | 2015-03-31 | Индиана Юниверсити Рисерч Энд Текнолоджи Корпорейшн | Агонисты смешанного действия на основе глюкозозависимого инсулинотропного пептида для лечения нарушений обмена веществ и ожирения |
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| CN102325539A (zh) | 2008-12-19 | 2012-01-18 | 印第安纳大学研究及科技有限公司 | 基于酰胺的胰高血糖素超家族肽前药 |
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| US8703701B2 (en) | 2009-12-18 | 2014-04-22 | Indiana University Research And Technology Corporation | Glucagon/GLP-1 receptor co-agonists |
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| RU2580317C2 (ru) | 2010-06-24 | 2016-04-10 | Индиана Юниверсити Рисерч Энд Текнолоджи Корпорейшн | Пептидные пролекарства, принадлежащие к суперсемейству амид-содержащих глюкагонов |
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-
2001
- 2001-08-02 BR BR0113178-8A patent/BR0113178A/pt not_active Application Discontinuation
- 2001-08-02 CA CA002417100A patent/CA2417100A1/en not_active Abandoned
- 2001-08-02 JP JP2002515924A patent/JP2004509079A/ja active Pending
- 2001-08-02 AU AU2001279526A patent/AU2001279526A1/en not_active Abandoned
- 2001-08-02 EP EP01957662A patent/EP1305338A2/en not_active Withdrawn
- 2001-08-02 CN CN01813865A patent/CN1454214A/zh active Pending
- 2001-08-02 WO PCT/CA2001/001119 patent/WO2002010195A2/en not_active Ceased
- 2001-08-02 US US10/343,654 patent/US20030204063A1/en not_active Abandoned
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004508410A (ja) * | 2000-09-18 | 2004-03-18 | オステオミーター・ビオテク・エー／エス | Ｇｌｐ−１及びｇｌｐ−２ペプチドの使用方法 |
| JP2004524268A (ja) * | 2000-09-18 | 2004-08-12 | オステオミーター・ビオテク・エー／エス | 骨関連疾患及び栄養関連疾患の治療、予防、診断及び予後のためにｇｌｐを使用する方法 |
| JP2011508728A (ja) * | 2007-12-21 | 2011-03-17 | ビーエーエスエフ ソシエタス・ヨーロピア | ペプチドを含有するフケ防止組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| BR0113178A (pt) | 2004-04-06 |
| WO2002010195A2 (en) | 2002-02-07 |
| CN1454214A (zh) | 2003-11-05 |
| EP1305338A2 (en) | 2003-05-02 |
| CA2417100A1 (en) | 2002-02-07 |
| AU2001279526A1 (en) | 2002-02-13 |
| US20030204063A1 (en) | 2003-10-30 |
| WO2002010195A3 (en) | 2002-10-03 |
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| Date | Code | Title | Description |
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| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20031212 |