JP2004508330A5 - - Google Patents
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- Publication number
- JP2004508330A5 JP2004508330A5 JP2002524497A JP2002524497A JP2004508330A5 JP 2004508330 A5 JP2004508330 A5 JP 2004508330A5 JP 2002524497 A JP2002524497 A JP 2002524497A JP 2002524497 A JP2002524497 A JP 2002524497A JP 2004508330 A5 JP2004508330 A5 JP 2004508330A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- alkyl
- pyridin
- pyrazolo
- piperidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23040700P | 2000-09-06 | 2000-09-06 | |
| US09/927,188 US6635633B2 (en) | 2000-08-14 | 2001-08-10 | Substituted pyrazoles |
| PCT/US2001/027480 WO2002020013A2 (en) | 2000-09-06 | 2001-09-05 | A method for treating allergies using substituted pyrazoles |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2004508330A JP2004508330A (ja) | 2004-03-18 |
| JP2004508330A5 true JP2004508330A5 (enExample) | 2005-08-18 |
| JP4129391B2 JP4129391B2 (ja) | 2008-08-06 |
Family
ID=26924202
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002524497A Expired - Fee Related JP4129391B2 (ja) | 2000-09-06 | 2001-09-05 | 置換ピラゾールを用いてアレルギーを治療する方法 |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1315492B1 (enExample) |
| JP (1) | JP4129391B2 (enExample) |
| CN (1) | CN1321641C (enExample) |
| AT (1) | ATE402699T1 (enExample) |
| AU (2) | AU8873101A (enExample) |
| CA (1) | CA2421510A1 (enExample) |
| DE (1) | DE60135130D1 (enExample) |
| DK (1) | DK1315492T3 (enExample) |
| ES (1) | ES2309088T3 (enExample) |
| HK (1) | HK1052881B (enExample) |
| MX (1) | MXPA03001962A (enExample) |
| NZ (1) | NZ524682A (enExample) |
| PT (1) | PT1315492E (enExample) |
| WO (1) | WO2002020013A2 (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004531456A (ja) * | 2000-09-06 | 2004-10-14 | オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド | 置換ピラゾールを用いてアレルギーを治療する方法 |
| ES2201899B1 (es) * | 2002-04-01 | 2005-06-01 | Almirall Prodesfarma, S.A. | Derivados de la azaindolilpiperidina como agentes antihistaminicos y antialergicos. |
| ES2201907B1 (es) | 2002-05-29 | 2005-06-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos. |
| DK1753764T3 (da) | 2004-06-09 | 2009-02-16 | Glaxo Group Ltd | Pyrrolopyridin-derivater |
| GEP20207129B (en) | 2009-06-17 | 2020-07-10 | Vertex Pharma | Inhibitors of influenza viruses replication |
| RU2013132681A (ru) | 2010-12-16 | 2015-01-27 | Вертекс Фармасьютикалз Инкорпорейтед | Ингибиторы репликации вирусов гриппа |
| UA118010C2 (uk) | 2011-08-01 | 2018-11-12 | Вертекс Фармасьютікалз Інкорпорейтед | Інгібітори реплікації вірусів грипу |
| US9260425B2 (en) | 2011-08-12 | 2016-02-16 | Genetech, Inc. | Pyrazolo[3,4-c]pyridine compounds and methods of use |
| PT3068776T (pt) | 2013-11-13 | 2019-08-26 | Vertex Pharma | Inibidores da replicação de vírus da gripe |
| HUE038820T2 (hu) | 2013-11-13 | 2018-11-28 | Vertex Pharma | Eljárás influenzavírusok replikációjának inhibitorai elõállítására |
| WO2016183120A1 (en) | 2015-05-13 | 2016-11-17 | Vertex Pharmaceuticals Incorporated | Inhibitors of influenza viruses replication |
| EP3294717B1 (en) | 2015-05-13 | 2020-07-29 | Vertex Pharmaceuticals Inc. | Methods of preparing inhibitors of influenza viruses replication |
| LT3860998T (lt) | 2018-10-05 | 2024-06-25 | Annapurna Bio Inc. | Junginiai ir kompozicijos, skirti gydyti būkles, susijusias su apj receptoriaus aktyvumu |
| CN111518019B (zh) * | 2019-02-01 | 2023-10-24 | 江苏豪森药业集团有限公司 | 一种棕榈酸帕里哌酮中间体的制备方法 |
| CN112142744A (zh) * | 2019-06-28 | 2020-12-29 | 上海瑛派药业有限公司 | 取代的稠合杂芳双环化合物作为激酶抑制剂及其应用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE789948A (fr) * | 1971-10-13 | 1973-04-11 | Sandoz Sa | Nouveaux derives du pyrazole, leur preparation et leur application comme medicaments |
| JPH0615542B2 (ja) * | 1986-07-22 | 1994-03-02 | 吉富製薬株式会社 | ピラゾロピリジン化合物 |
| JP3907220B2 (ja) * | 1994-06-30 | 2007-04-18 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 複素環含有化合物 |
| JP3964478B2 (ja) * | 1995-06-30 | 2007-08-22 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ヘテロ環含有カルボン酸誘導体及びそれを含有する医薬 |
| AU7553198A (en) * | 1997-06-12 | 1998-12-30 | Sumitomo Pharmaceuticals Company, Limited | Pyrazole derivatives |
-
2001
- 2001-09-05 AT AT01968487T patent/ATE402699T1/de not_active IP Right Cessation
- 2001-09-05 CN CNB018185045A patent/CN1321641C/zh not_active Expired - Lifetime
- 2001-09-05 WO PCT/US2001/027480 patent/WO2002020013A2/en not_active Ceased
- 2001-09-05 AU AU8873101A patent/AU8873101A/xx active Pending
- 2001-09-05 CA CA002421510A patent/CA2421510A1/en not_active Abandoned
- 2001-09-05 HK HK03105185.1A patent/HK1052881B/en not_active IP Right Cessation
- 2001-09-05 EP EP01968487A patent/EP1315492B1/en not_active Expired - Lifetime
- 2001-09-05 NZ NZ524682A patent/NZ524682A/en unknown
- 2001-09-05 MX MXPA03001962A patent/MXPA03001962A/es active IP Right Grant
- 2001-09-05 AU AU2001288731A patent/AU2001288731B8/en not_active Expired
- 2001-09-05 PT PT01968487T patent/PT1315492E/pt unknown
- 2001-09-05 DK DK01968487T patent/DK1315492T3/da active
- 2001-09-05 JP JP2002524497A patent/JP4129391B2/ja not_active Expired - Fee Related
- 2001-09-05 DE DE60135130T patent/DE60135130D1/de not_active Expired - Lifetime
- 2001-09-05 ES ES01968487T patent/ES2309088T3/es not_active Expired - Lifetime
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