JP2004506632A5 - - Google Patents

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Publication number
JP2004506632A5
JP2004506632A5 JP2002519452A JP2002519452A JP2004506632A5 JP 2004506632 A5 JP2004506632 A5 JP 2004506632A5 JP 2002519452 A JP2002519452 A JP 2002519452A JP 2002519452 A JP2002519452 A JP 2002519452A JP 2004506632 A5 JP2004506632 A5 JP 2004506632A5
Authority
JP
Japan
Prior art keywords
methyl
tetrazol
phenyl
thiazol
cyclopentyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2002519452A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004506632A (ja
JP3961948B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2001/009207 external-priority patent/WO2002014312A1/en
Publication of JP2004506632A publication Critical patent/JP2004506632A/ja
Publication of JP2004506632A5 publication Critical patent/JP2004506632A5/ja
Application granted granted Critical
Publication of JP3961948B2 publication Critical patent/JP3961948B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2002519452A 2000-08-15 2001-08-09 テトラゾリル−フェニルアセトアミドであるグルコキナーゼ活性化物質 Expired - Fee Related JP3961948B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22549400P 2000-08-15 2000-08-15
PCT/EP2001/009207 WO2002014312A1 (en) 2000-08-15 2001-08-09 Tetrazolyl-phenyl acetamide glucokinase activators

Publications (3)

Publication Number Publication Date
JP2004506632A JP2004506632A (ja) 2004-03-04
JP2004506632A5 true JP2004506632A5 (cg-RX-API-DMAC10.html) 2005-03-17
JP3961948B2 JP3961948B2 (ja) 2007-08-22

Family

ID=22845106

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002519452A Expired - Fee Related JP3961948B2 (ja) 2000-08-15 2001-08-09 テトラゾリル−フェニルアセトアミドであるグルコキナーゼ活性化物質

Country Status (20)

Country Link
US (3) US6369232B1 (cg-RX-API-DMAC10.html)
EP (1) EP1311504B1 (cg-RX-API-DMAC10.html)
JP (1) JP3961948B2 (cg-RX-API-DMAC10.html)
KR (1) KR100518061B1 (cg-RX-API-DMAC10.html)
CN (1) CN1209362C (cg-RX-API-DMAC10.html)
AR (1) AR031718A1 (cg-RX-API-DMAC10.html)
AT (1) ATE297921T1 (cg-RX-API-DMAC10.html)
AU (2) AU2001283998B2 (cg-RX-API-DMAC10.html)
BR (1) BR0113312A (cg-RX-API-DMAC10.html)
CA (1) CA2419416C (cg-RX-API-DMAC10.html)
DE (1) DE60111540T2 (cg-RX-API-DMAC10.html)
DK (1) DK1311504T3 (cg-RX-API-DMAC10.html)
ES (1) ES2243541T3 (cg-RX-API-DMAC10.html)
MX (1) MXPA03001275A (cg-RX-API-DMAC10.html)
PA (1) PA8525201A1 (cg-RX-API-DMAC10.html)
PE (1) PE20020386A1 (cg-RX-API-DMAC10.html)
PT (1) PT1311504E (cg-RX-API-DMAC10.html)
UY (1) UY26885A1 (cg-RX-API-DMAC10.html)
WO (1) WO2002014312A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA200300904B (cg-RX-API-DMAC10.html)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0102299D0 (sv) 2001-06-26 2001-06-26 Astrazeneca Ab Compounds
SE0102764D0 (sv) 2001-08-17 2001-08-17 Astrazeneca Ab Compounds
US7087631B2 (en) * 2002-07-18 2006-08-08 Inotek Pharmaceuticals Corporation Aryltetrazole compounds, and compositions thereof
US7078423B2 (en) * 2002-07-18 2006-07-18 Inotek Pharmaceuticals Corporation 5-Aryltetrazole compounds, compositions thereof, and uses therefor
NZ539013A (en) * 2002-10-03 2007-05-31 Novartis Ag Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in the treatment of type 2 diabetes
GB0226931D0 (en) 2002-11-19 2002-12-24 Astrazeneca Ab Chemical compounds
MY141521A (en) 2002-12-12 2010-05-14 Hoffmann La Roche 5-substituted-six-membered heteroaromatic glucokinase activators
WO2004063194A1 (en) * 2003-01-06 2004-07-29 Eli Lilly And Company Heteroaryl compounds
WO2004072066A1 (en) * 2003-02-11 2004-08-26 Prosidion Limited Tri(cyclo) substituted amide glucokinase activator compounds
PL378117A1 (pl) * 2003-02-11 2006-03-06 Prosidion Limited Tricyklopodstawione związki amidowe
CA2561157A1 (en) * 2004-04-02 2005-10-13 Novartis Ag Thiazolopyridine derivatives, pharmaceutical conditions containing them and methods of treating glucokinase mediated conditions
RU2412192C2 (ru) * 2004-04-02 2011-02-20 Новартис Аг Сульфонамидтиазолпиридиновые производные как активаторы глюкокиназы, пригодные для лечения диабета типа 2
JP4651714B2 (ja) 2005-07-09 2011-03-16 アストラゼネカ アクチボラグ 糖尿病の治療においてglk活性化剤として使用するためのヘテロアリールベンズアミド誘導体
US7514439B2 (en) 2005-07-11 2009-04-07 Mitsubishi Tanabe Pharma Corporation Oxime derivative and preparations thereof
AU2006285834A1 (en) 2005-08-31 2007-03-08 Astellas Pharma Inc. Thiazole derivative
JP2007063225A (ja) * 2005-09-01 2007-03-15 Takeda Chem Ind Ltd イミダゾピリジン化合物
WO2007039177A2 (en) 2005-09-29 2007-04-12 Sanofi-Aventis Phenyl- and pyridinyl- 1, 2 , 4 - oxadiazolone derivatives, processes for their preparation and their use as pharmaceuticals
GT200600429A (es) * 2005-09-30 2007-04-30 Compuestos organicos
GT200600428A (es) * 2005-09-30 2007-05-21 Compuestos organicos
CA2626475A1 (en) * 2005-11-03 2007-05-10 Prosidion Limited Tricyclo substituted amides
JP2009515997A (ja) * 2005-11-18 2009-04-16 タケダ サン ディエゴ インコーポレイテッド グルコキナーゼ活性剤
WO2007069684A1 (ja) * 2005-12-15 2007-06-21 Nihon Nohyaku Co., Ltd. フタルアミド誘導体及び農園芸用殺虫剤並びにその使用方法
US8034822B2 (en) 2006-03-08 2011-10-11 Takeda San Diego, Inc. Glucokinase activators
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
EP2049518B1 (en) * 2006-05-31 2011-08-31 Takeda San Diego, Inc. Indazole and isoindole derivatives as glucokinase activating agents.
US7910747B2 (en) * 2006-07-06 2011-03-22 Bristol-Myers Squibb Company Phosphonate and phosphinate pyrazolylamide glucokinase activators
US7902248B2 (en) 2006-12-14 2011-03-08 Hoffmann-La Roche Inc. Oxime glucokinase activators
WO2008079787A2 (en) 2006-12-20 2008-07-03 Takeda San Diego, Inc. Glucokinase activators
TW200831081A (en) * 2006-12-25 2008-08-01 Kyorin Seiyaku Kk Glucokinase activator
EP2105435A4 (en) * 2007-01-10 2011-06-15 Mitsubishi Tanabe Pharma Corp Hydrazone derivative
EP2116533B1 (en) * 2007-03-07 2013-07-10 Kyorin Pharmaceutical Co., Ltd. Glucokinase activator
WO2008116107A2 (en) * 2007-03-21 2008-09-25 Takeda San Diego, Inc. Piperazine derivatives as glucokinase activators
EP2195304B1 (en) * 2007-10-08 2014-01-08 Advinus Therapeutics Private Limited Acetamide derivatives as glucokinase activators, their process and medicinal applications
AR070107A1 (es) * 2008-01-15 2010-03-17 Lilly Co Eli R-2-(4-ciclopropansulfonil-fenil)-n-pirazin-2-il-3-(tetrahidropiran-4-il)-propionamida en forma cristalina, composicion farmaceutica que la comprende y su uso para la manufactura de un medicamento util para la prevencion o tratamiento de hiperglicemia
RU2010134411A (ru) * 2008-01-18 2012-02-27 Астеллас Фарма Инк. (Jp) Фенилацетамидное производное
NZ588462A (en) 2008-04-28 2012-07-27 Kyorin Seiyaku Kk Cyclopentylacrylic acid amide derivative
CN105176930B (zh) 2010-03-31 2021-05-04 斯克里普斯研究所 重编程细胞

Family Cites Families (7)

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Publication number Priority date Publication date Assignee Title
US3776917A (en) * 1972-06-05 1973-12-04 Schering Corp 2-amino-6-phenalkyl-aminopyridines and derivatives thereof
GB8909574D0 (en) 1989-04-26 1989-06-14 Ici Plc Chemical process
US5859052A (en) * 1993-01-14 1999-01-12 G. D. Searle & Co. Fatty acid analogs and prodrugs
US5461049A (en) * 1994-05-27 1995-10-24 Warner-Lambert Company Amide tetrazole ACAT inhibitors
US5468867A (en) * 1994-05-27 1995-11-21 Syntex (U.S.A.) Inc. Process for preparing1-butyl-2-[2'-(2H-tetrazol-5-yl)biphenyl-4-ylmethyl1-1H-indole-3-carboxylic acid
KR20000070568A (ko) * 1997-01-28 2000-11-25 폴락 돈나 엘. 당뇨병 및 비만 치료를 위한 β3 효능제로서의 티아졸 벤젠설폰아미드
TR200102805T2 (tr) * 1999-03-29 2002-04-22 F.Hoffmann-La Roche Ag Glikokinaz aktivatörleri

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