JP2003201284A - 置換チアゾリン類およびその中間体の製造方法 - Google Patents

置換チアゾリン類およびその中間体の製造方法

Info

Publication number
JP2003201284A
JP2003201284A JP2002300807A JP2002300807A JP2003201284A JP 2003201284 A JP2003201284 A JP 2003201284A JP 2002300807 A JP2002300807 A JP 2002300807A JP 2002300807 A JP2002300807 A JP 2002300807A JP 2003201284 A JP2003201284 A JP 2003201284A
Authority
JP
Japan
Prior art keywords
formula
hcl
methylcysteine
solution
lipase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2002300807A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003201284A5 (enExample
Inventor
Sylvia Krich
シルヴィア・クリヒ
Alexander Rieder
アレクザンダー・リーダー
Ferdinand Heu
フェルデイナンド・ホイ
Gerhard Steinbauer
ゲルハルト・シュタインバウアー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Patheon Austria GmbH and Co KG
Original Assignee
DSM Fine Chemicals Austria Nfg GmbH and Co KG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by DSM Fine Chemicals Austria Nfg GmbH and Co KG filed Critical DSM Fine Chemicals Austria Nfg GmbH and Co KG
Publication of JP2003201284A publication Critical patent/JP2003201284A/ja
Publication of JP2003201284A5 publication Critical patent/JP2003201284A5/ja
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/02—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
JP2002300807A 2001-10-16 2002-10-15 置換チアゾリン類およびその中間体の製造方法 Withdrawn JP2003201284A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT1639/2001 2001-10-16
AT0163901A AT500490A1 (de) 2001-10-16 2001-10-16 Verfahren zur herstellung von substituierten thiazolinen und deren zwischenprodukte

Publications (2)

Publication Number Publication Date
JP2003201284A true JP2003201284A (ja) 2003-07-18
JP2003201284A5 JP2003201284A5 (enExample) 2005-11-04

Family

ID=3688515

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002300807A Withdrawn JP2003201284A (ja) 2001-10-16 2002-10-15 置換チアゾリン類およびその中間体の製造方法

Country Status (4)

Country Link
US (2) US6894170B2 (enExample)
EP (1) EP1302467A3 (enExample)
JP (1) JP2003201284A (enExample)
AT (1) AT500490A1 (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6794515B2 (en) * 2002-05-15 2004-09-21 Genzyme Corporation Synthesis of 2-alkylcysteine via substituted thiazoline amide
JPWO2004031163A1 (ja) * 2002-10-01 2006-02-02 株式会社カネカ 光学活性α−置換システインまたはその塩の製造方法並びにその合成中間体及びその製造方法
DE10308580B3 (de) * 2003-02-27 2004-09-09 Consortium für elektrochemische Industrie GmbH Verfahren zur elektrophilen Substitution von Thiazolidinen oder Oxazolidinen
DE10317878A1 (de) * 2003-04-17 2004-11-11 Consortium für elektrochemische Industrie GmbH Verfahren zur Herstellung von alpha-methylierten Cystein und Serin-Derivaten
WO2005055931A2 (en) * 2003-12-03 2005-06-23 University Of Medicine And Dentistry Of New Jersey Method of preventing survival of retrovirally cells and of inhibiting formation of infectious retroviruses
JP2006312614A (ja) * 2005-05-09 2006-11-16 Ajinomoto Co Inc チアゾリン化合物および光学活性α−アルキルシステインの製造方法
CN103435569B (zh) 2008-07-14 2015-08-19 法罗肯生物科学公司 作为金属螯合剂的脱氮杂去铁硫辛聚醚类似物的新型盐和多晶型物
EP2459544A4 (en) * 2009-07-27 2012-12-05 Ferrokin Biosciences Inc DESDAADESFERROTHIOCIN POLYETHERAL ANALOGUE PROGRUGS USING METAL CHLORIDE
JP2013525495A (ja) 2010-05-04 2013-06-20 シャイアー・リミテッド・ライアビリティ・カンパニー 金属キレート化剤としてのデスアザデスフェリチオシン類似体
PT2624695E (pt) 2010-10-08 2015-12-01 Nivalis Therapeutics Inc Novos compostos de quinolina substituídos como inibidores de s-nitrosoglutationa redutase
US8785643B2 (en) 2010-12-16 2014-07-22 N30 Pharmaceuticals, Inc. Substituted bicyclic aromatic compounds as S-nitrosoglutathione reductase inhibitors
CN104892477A (zh) * 2015-06-15 2015-09-09 尚科生物医药（上海）有限公司 手性2-甲基半胱氨酸及其盐酸盐的制备方法
WO2017044766A1 (en) 2015-09-10 2017-03-16 Nivalis Therapeutics, Inc. Solid forms of an s-nitrosoglutathione reductase inhibitor

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US220504A (en) * 1879-10-14 Improvement in globe-holders for gas-fixtures
EP0045281B1 (de) * 1980-07-28 1985-05-08 Ciba-Geigy Ag Thiazolinderivate und Verfahren zu ihrer Herstellung
US6794515B2 (en) * 2002-05-15 2004-09-21 Genzyme Corporation Synthesis of 2-alkylcysteine via substituted thiazoline amide

Also Published As

Publication number Publication date
AT500490A1 (de) 2006-01-15
US6894170B2 (en) 2005-05-17
EP1302467A2 (de) 2003-04-16
US20050101782A1 (en) 2005-05-12
US20030088105A1 (en) 2003-05-08
EP1302467A3 (de) 2003-05-02

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