JP2002507576A5 - - Google Patents

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Publication number
JP2002507576A5
JP2002507576A5 JP2000537561A JP2000537561A JP2002507576A5 JP 2002507576 A5 JP2002507576 A5 JP 2002507576A5 JP 2000537561 A JP2000537561 A JP 2000537561A JP 2000537561 A JP2000537561 A JP 2000537561A JP 2002507576 A5 JP2002507576 A5 JP 2002507576A5
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JP
Japan
Prior art keywords
seq
formula
peptide
fmoc
side chain
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2000537561A
Other languages
English (en)
Japanese (ja)
Other versions
JP4602547B2 (ja
JP2002507576A (ja
Filing date
Publication date
Priority claimed from US09/045,920 external-priority patent/US6281331B1/en
Application filed filed Critical
Priority claimed from PCT/US1999/006230 external-priority patent/WO1999048513A1/en
Publication of JP2002507576A publication Critical patent/JP2002507576A/ja
Publication of JP2002507576A5 publication Critical patent/JP2002507576A5/ja
Application granted granted Critical
Publication of JP4602547B2 publication Critical patent/JP4602547B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2000537561A 1998-03-23 1999-03-22 ペプチド合成のための方法および組成物 Expired - Fee Related JP4602547B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US09/045,920 US6281331B1 (en) 1998-03-23 1998-03-23 Methods and compositions for peptide synthesis
US09/045,920 1998-03-23
US09/071,877 1998-05-01
US09/071,877 US6015881A (en) 1998-03-23 1998-05-01 Methods and compositions for peptide synthesis
PCT/US1999/006230 WO1999048513A1 (en) 1998-03-23 1999-03-22 Methods and compositions for peptide synthesis

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2009247579A Division JP4755713B2 (ja) 1998-03-23 2009-10-28 ペプチド合成のための方法および組成物

Publications (3)

Publication Number Publication Date
JP2002507576A JP2002507576A (ja) 2002-03-12
JP2002507576A5 true JP2002507576A5 (enExample) 2006-06-08
JP4602547B2 JP4602547B2 (ja) 2010-12-22

Family

ID=26723345

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000537561A Expired - Fee Related JP4602547B2 (ja) 1998-03-23 1999-03-22 ペプチド合成のための方法および組成物

Country Status (13)

Country Link
EP (1) EP1071442B9 (enExample)
JP (1) JP4602547B2 (enExample)
CN (1) CN100383158C (enExample)
AT (1) ATE299029T1 (enExample)
AU (1) AU751358B2 (enExample)
BR (1) BR9909018A (enExample)
CA (1) CA2324348C (enExample)
DE (1) DE69926061T2 (enExample)
DK (1) DK1071442T3 (enExample)
ES (1) ES2245505T3 (enExample)
NZ (1) NZ507083A (enExample)
TW (1) TWI233931B (enExample)
WO (1) WO1999048513A1 (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6281331B1 (en) * 1998-03-23 2001-08-28 Trimeris, Inc. Methods and compositions for peptide synthesis
US6469136B1 (en) * 1999-07-07 2002-10-22 Trimeris, Inc. Methods and composition for peptide synthesis
CA2450548C (en) 2001-06-15 2012-05-01 F. Hoffmann-La Roche Ag Method for the recombinant production of peptidic antiviral fusion inhibitors, and acetylation of gb41 fragments
KR100637981B1 (ko) * 2002-07-24 2006-10-23 에프. 호프만-라 로슈 아게 페길화된 t20 폴리펩타이드
ATE376556T1 (de) 2003-12-31 2007-11-15 Hoffmann La Roche Verfahren zur peptidsynthese unter verwendung einer reduzierten menge an entschützungsmittel
WO2005063799A2 (en) * 2003-12-31 2005-07-14 F.Hoffmann-La Roche Ag Peptide synthesis and deprotection with co-solvent
ATE410437T1 (de) 2003-12-31 2008-10-15 Hoffmann La Roche Verfahren und systeme zur rückgewinnung von peptiden
MX2007007917A (es) * 2004-12-30 2007-08-14 Hoffmann La Roche Sintesis del peptido t-20 utilizando fragmentos peptidicos intermediarios.
JP2009535402A (ja) 2006-05-03 2009-10-01 マリンクロッド・インコーポレイテッド 保護ペプチドを樹脂から放出するための組成物および方法
JP5515738B2 (ja) * 2007-07-25 2014-06-11 味の素株式会社 ジベンゾフルベン誘導体の淘汰方法
DK2205624T3 (da) * 2007-10-27 2017-01-02 Corden Pharma Colorado Inc Insulinotropisk peptidsyntese under anvendelse af faststof- og opløsningsfasekombinationsteknikker
MX2010006044A (es) * 2007-12-11 2010-06-23 Hoffmann La Roche Sintesis de peptidos insulinotropicos utilizando una combinacion de tecnicas en fase solida y en solucion.
JP5445456B2 (ja) 2008-08-06 2014-03-19 味の素株式会社 ジベンゾフルベンの除去方法
US20110288235A1 (en) * 2008-09-03 2011-11-24 Scinopharm Taiwan Ltd. Process for the Preparation of Pramlintide
JP2012502045A (ja) * 2008-09-03 2012-01-26 サイノファーム タイワン リミテッド プラムリンチドの製造方法
WO2011095989A2 (en) * 2010-02-04 2011-08-11 Matrix Laboratories Ltd An improved process for the preparation of enfuvirtide
PL219569B1 (pl) * 2010-02-19 2015-05-29 Peptaderm Spółka Z Ograniczoną Odpowiedzialnością Cykliczne tetrapeptydy i ich zastosowanie
CN103374054B (zh) * 2012-04-28 2014-12-24 上海第一生化药业有限公司 一步法固相合成多肽的方法
GB201315335D0 (en) 2013-08-29 2013-10-09 Of Singapore Amino diacids containing peptide modifiers
EP4100417A2 (en) * 2020-02-05 2022-12-14 Eli Lilly and Company Resin reactors in series peptide synthesizer
CN114315957B (zh) * 2021-12-30 2023-07-07 深圳瑞德林生物技术有限公司 一种多肽的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU617088B2 (en) * 1986-06-12 1991-11-21 Biogen, Inc. Peptides involved in the pathogenesis of hiv infection
US4787222A (en) * 1986-11-24 1988-11-29 Novatek Medical Inc. Combination lock for blood identification system
US5444044A (en) * 1992-03-26 1995-08-22 New York Blood Center Synthetic polypeptides as inhibitors of HIV-1
US5464933A (en) * 1993-06-07 1995-11-07 Duke University Synthetic peptide inhibitors of HIV transmission
US5864027A (en) * 1993-06-07 1999-01-26 Genentech, Inc. HIV envelope polypeptides
US6479055B1 (en) * 1993-06-07 2002-11-12 Trimeris, Inc. Methods for inhibition of membrane fusion-associated events, including respiratory syncytial virus transmission
DE69426725T2 (de) * 1993-09-11 2001-09-06 Polimun Scientific Immunbiologische Forschungsgesellschaft Mbh, Wien Peptide, die neutralisierende antikörper gegen genetisch divergierende hiv-1 stämme, induzieren
DE69735991D1 (de) * 1996-02-09 2006-07-06 Hoffmann La Roche Herstellung eines vip-analogen

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