JP2001500878A5 - - Google Patents

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Publication number
JP2001500878A5
JP2001500878A5 JP1998514881A JP51488198A JP2001500878A5 JP 2001500878 A5 JP2001500878 A5 JP 2001500878A5 JP 1998514881 A JP1998514881 A JP 1998514881A JP 51488198 A JP51488198 A JP 51488198A JP 2001500878 A5 JP2001500878 A5 JP 2001500878A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP1998514881A
Other languages
English (en)
Japanese (ja)
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JP2001500878A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/016586 external-priority patent/WO1998011893A1/en
Publication of JP2001500878A publication Critical patent/JP2001500878A/ja
Publication of JP2001500878A5 publication Critical patent/JP2001500878A5/ja
Withdrawn legal-status Critical Current

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JP10514881A 1996-09-23 1997-09-18 オランザピン二水和物d Withdrawn JP2001500878A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2648696P 1996-09-23 1996-09-23
US60/026,486 1996-09-23
PCT/US1997/016586 WO1998011893A1 (en) 1996-09-23 1997-09-18 Olanzapine dihydrate d

Publications (2)

Publication Number Publication Date
JP2001500878A JP2001500878A (ja) 2001-01-23
JP2001500878A5 true JP2001500878A5 (https=) 2005-05-12

Family

ID=21832112

Family Applications (1)

Application Number Title Priority Date Filing Date
JP10514881A Withdrawn JP2001500878A (ja) 1996-09-23 1997-09-18 オランザピン二水和物d

Country Status (34)

Country Link
US (1) US6251895B1 (https=)
EP (1) EP0831097B1 (https=)
JP (1) JP2001500878A (https=)
KR (1) KR100516088B1 (https=)
CN (1) CN1146567C (https=)
AR (1) AR009801A1 (https=)
AT (1) ATE221074T1 (https=)
AU (1) AU720366B2 (https=)
BR (1) BR9711541A (https=)
CA (1) CA2266444C (https=)
CO (1) CO4900057A1 (https=)
CZ (1) CZ299247B6 (https=)
DE (1) DE69714165T2 (https=)
DK (1) DK0831097T3 (https=)
EA (1) EA001881B1 (https=)
EG (1) EG23815A (https=)
ES (1) ES2180899T3 (https=)
HU (1) HU226167B1 (https=)
ID (1) ID21924A (https=)
IL (1) IL128956A0 (https=)
MY (1) MY125467A (https=)
NO (1) NO323979B1 (https=)
NZ (1) NZ334346A (https=)
PE (1) PE110298A1 (https=)
PL (1) PL194074B1 (https=)
PT (1) PT831097E (https=)
RS (1) RS49597B (https=)
SI (1) SI0831097T1 (https=)
SV (1) SV1997000079A (https=)
TR (1) TR199900639T2 (https=)
TW (1) TW518335B (https=)
UA (1) UA56184C2 (https=)
WO (1) WO1998011893A1 (https=)
ZA (1) ZA978512B (https=)

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US20060074088A1 (en) 2004-08-14 2006-04-06 Boehringer Ingelheim International Gmbh Dihydropteridinones for the treatment of cancer diseases
US20060058311A1 (en) 2004-08-14 2006-03-16 Boehringer Ingelheim International Gmbh Combinations for the treatment of diseases involving cell proliferation
US7759485B2 (en) 2004-08-14 2010-07-20 Boehringer Ingelheim International Gmbh Process for the manufacture of dihydropteridinones
US7728134B2 (en) 2004-08-14 2010-06-01 Boehringer Ingelheim International Gmbh Hydrates and polymorphs of 4[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, process for their manufacture and their use as medicament
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WO2006027800A1 (en) * 2004-09-06 2006-03-16 Shasun Chemicals And Drugs Limited A novel process for preparation of a pharmaceutically pure polymorphic form 1 of olanzapine
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US7834176B2 (en) * 2006-01-26 2010-11-16 Sandoz Ag Polymorph E of Olanzapine and preparation of anhydrous non-solvated crystalline polymorphic Form I of 2-methyl-4(4-methyl-1-piperazinyl)-10H-thieno[2,3-b][1,5] benzodiazepine (Olanzapine Form I) from the polymorphic Olanzapine Form E
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CN102149407A (zh) 2008-09-10 2011-08-10 贝林格尔.英格海姆国际有限公司 治疗糖尿病和相关病症的组合疗法
US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
CN102256976A (zh) 2008-12-23 2011-11-23 贝林格尔.英格海姆国际有限公司 有机化合物的盐形式
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CN102946875A (zh) 2010-05-05 2013-02-27 贝林格尔.英格海姆国际有限公司 组合疗法
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US8546566B2 (en) 2010-10-12 2013-10-01 Boehringer Ingelheim International Gmbh Process for manufacturing dihydropteridinones and intermediates thereof
AR083878A1 (es) 2010-11-15 2013-03-27 Boehringer Ingelheim Int Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento
US9358233B2 (en) 2010-11-29 2016-06-07 Boehringer Ingelheim International Gmbh Method for treating acute myeloid leukemia
US9370535B2 (en) 2011-05-17 2016-06-21 Boehringer Ingelheim International Gmbh Method for treatment of advanced solid tumors
US8883800B2 (en) 2011-07-15 2014-11-11 Boehringer Ingelheim International Gmbh Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US9555001B2 (en) 2012-03-07 2017-01-31 Boehringer Ingelheim International Gmbh Pharmaceutical composition and uses thereof
JP6224084B2 (ja) 2012-05-14 2017-11-01 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 糸球体上皮細胞関連障害及び/又はネフローゼ症候群の治療に用いるdpp−4阻害薬としてのキサンチン誘導体
JP6218811B2 (ja) 2012-05-14 2017-10-25 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Sirs及び/又は敗血症の治療に用いるdpp−4阻害薬としてのキサンチン誘導体
WO2013174767A1 (en) 2012-05-24 2013-11-28 Boehringer Ingelheim International Gmbh A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference
US20140206667A1 (en) 2012-11-14 2014-07-24 Michela Gallagher Methods and compositions for treating schizophrenia
JP2016027003A (ja) * 2012-11-20 2016-02-18 大蔵製薬株式会社 長期間安定なオランザピンの水性医薬製剤
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EP3110449B1 (en) 2014-02-28 2023-06-28 Boehringer Ingelheim International GmbH Medical use of a dpp-4 inhibitor
US9867831B2 (en) 2014-10-01 2018-01-16 Boehringer Ingelheim International Gmbh Combination treatment of acute myeloid leukemia and myelodysplastic syndrome
CN109310697A (zh) 2016-06-10 2019-02-05 勃林格殷格翰国际有限公司 利格列汀和二甲双胍的组合

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