AR009801A1 - Dihidrato d polimorfo de olanzapina, formulaciones farmaceuticas que los contienen como ingrediente activo y metodo para tratar patologias psicoticas,tales como esquizofrenia, ansiedad, trastornos intestinales funcionales y psicosis aplicando dichas formulaciones - Google Patents

Dihidrato d polimorfo de olanzapina, formulaciones farmaceuticas que los contienen como ingrediente activo y metodo para tratar patologias psicoticas,tales como esquizofrenia, ansiedad, trastornos intestinales funcionales y psicosis aplicando dichas formulaciones

Info

Publication number
AR009801A1
AR009801A1 ARP970104361A ARP970104361A AR009801A1 AR 009801 A1 AR009801 A1 AR 009801A1 AR P970104361 A ARP970104361 A AR P970104361A AR P970104361 A ARP970104361 A AR P970104361A AR 009801 A1 AR009801 A1 AR 009801A1
Authority
AR
Argentina
Prior art keywords
dihydrate
pathologies
psychosis
schizophrenia
anxiety
Prior art date
Application number
ARP970104361A
Other languages
English (en)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21832112&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR009801(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of AR009801A1 publication Critical patent/AR009801A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/38—[b, e]- or [b, f]-condensed with six-membered rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Dihidrato D 2-metil-tieno-benzodiazepina novedoso (olanzapina), con el siguiente patron RX (en polvo) d 9.4511 - 7.7098 - 7.4482 - 6.9807 - 6.5252 -5.7076 - 5.5539 - 5.223 - 4.9803 - 4.8908 - 4.784 - 4.6947 - 4.4271 - 4.3956 - 4.3492 - 4.2834 -4.1156 - 3.7837 - 3.7118 - 3.5757 - 3.482 - 3.3758 - 3.3274 -3.2413 - 3.1879 - 3.135 - 3.0979 - 3.016 - 2.9637 - 2.907 - 2.8256 - 2.7914 - 2.7317 - 2.6732 - 2.5863. También se proponen composiciones formuladas condicho dihidrato y el tratamiento de diversas patologías psicoticas utilizando dichas formulaciones.
ARP970104361A 1996-09-23 1997-09-23 Dihidrato d polimorfo de olanzapina, formulaciones farmaceuticas que los contienen como ingrediente activo y metodo para tratar patologias psicoticas,tales como esquizofrenia, ansiedad, trastornos intestinales funcionales y psicosis aplicando dichas formulaciones AR009801A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2648696P 1996-09-23 1996-09-23

Publications (1)

Publication Number Publication Date
AR009801A1 true AR009801A1 (es) 2000-05-03

Family

ID=21832112

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP970104361A AR009801A1 (es) 1996-09-23 1997-09-23 Dihidrato d polimorfo de olanzapina, formulaciones farmaceuticas que los contienen como ingrediente activo y metodo para tratar patologias psicoticas,tales como esquizofrenia, ansiedad, trastornos intestinales funcionales y psicosis aplicando dichas formulaciones

Country Status (35)

Country Link
US (1) US6251895B1 (es)
EP (1) EP0831097B1 (es)
JP (1) JP2001500878A (es)
KR (1) KR100516088B1 (es)
CN (1) CN1146567C (es)
AR (1) AR009801A1 (es)
AT (1) ATE221074T1 (es)
AU (1) AU720366B2 (es)
BR (1) BR9711541A (es)
CA (1) CA2266444C (es)
CO (1) CO4900057A1 (es)
CZ (1) CZ299247B6 (es)
DE (1) DE69714165T2 (es)
DK (1) DK0831097T3 (es)
EA (1) EA001881B1 (es)
EG (1) EG23815A (es)
ES (1) ES2180899T3 (es)
HK (1) HK1009809A1 (es)
HU (1) HU226167B1 (es)
ID (1) ID21924A (es)
IL (1) IL128956A0 (es)
MY (1) MY125467A (es)
NO (1) NO323979B1 (es)
NZ (1) NZ334346A (es)
PE (1) PE110298A1 (es)
PL (1) PL194074B1 (es)
PT (1) PT831097E (es)
RS (1) RS49597B (es)
SI (1) SI0831097T1 (es)
SV (1) SV1997000079A (es)
TR (1) TR199900639T2 (es)
TW (1) TW518335B (es)
UA (1) UA56184C2 (es)
WO (1) WO1998011893A1 (es)
ZA (1) ZA978512B (es)

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Also Published As

Publication number Publication date
NZ334346A (en) 2000-05-26
PT831097E (pt) 2002-10-31
SV1997000079A (es) 1999-01-13
MY125467A (en) 2006-08-30
EA199900325A1 (ru) 1999-08-26
TW518335B (en) 2003-01-21
NO991339L (no) 1999-03-19
DE69714165T2 (de) 2003-01-23
CA2266444C (en) 2007-01-09
NO991339D0 (no) 1999-03-19
PL332541A1 (en) 1999-09-13
RS49597B (sr) 2007-06-04
KR100516088B1 (ko) 2005-09-22
CA2266444A1 (en) 1998-03-26
EP0831097B1 (en) 2002-07-24
EP0831097A3 (en) 1998-04-29
ES2180899T3 (es) 2003-02-16
NO323979B1 (no) 2007-07-30
YU15499A (sh) 2000-03-21
HUP0000065A3 (en) 2000-11-28
HU226167B1 (hu) 2008-05-28
KR20000048519A (ko) 2000-07-25
HK1009809A1 (en) 1999-06-11
PE110298A1 (es) 1999-01-18
CZ299247B6 (cs) 2008-05-28
CN1146567C (zh) 2004-04-21
AU4424197A (en) 1998-04-14
BR9711541A (pt) 1999-08-24
DE69714165D1 (de) 2002-08-29
ID21924A (id) 1999-08-12
ZA978512B (en) 1999-03-23
SI0831097T1 (en) 2003-02-28
EA001881B1 (ru) 2001-10-22
CZ98999A3 (cs) 1999-08-11
CO4900057A1 (es) 2000-03-27
WO1998011893A1 (en) 1998-03-26
CN1234738A (zh) 1999-11-10
UA56184C2 (uk) 2003-05-15
ATE221074T1 (de) 2002-08-15
EP0831097A2 (en) 1998-03-25
AU720366B2 (en) 2000-06-01
DK0831097T3 (da) 2002-09-02
JP2001500878A (ja) 2001-01-23
TR199900639T2 (xx) 1999-06-21
EG23815A (en) 2007-08-19
IL128956A0 (en) 2000-02-17
PL194074B1 (pl) 2007-04-30
US6251895B1 (en) 2001-06-26
HUP0000065A2 (hu) 2000-06-28

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