IT1206505B - Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono. - Google Patents

Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono.

Info

Publication number
IT1206505B
IT1206505B IT8322185A IT2218583A IT1206505B IT 1206505 B IT1206505 B IT 1206505B IT 8322185 A IT8322185 A IT 8322185A IT 2218583 A IT2218583 A IT 2218583A IT 1206505 B IT1206505 B IT 1206505B
Authority
IT
Italy
Prior art keywords
benzothiazepinonic
derivatives
contain
preparation
new
Prior art date
Application number
IT8322185A
Other languages
English (en)
Other versions
IT8322185A0 (it
Inventor
Stefano Maiorana
Diego Brocchetti
Giuseppe Piacenza
Amedea Manfredi
Original Assignee
Schiapparelli Farma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schiapparelli Farma filed Critical Schiapparelli Farma
Publication of IT8322185A0 publication Critical patent/IT8322185A0/it
Priority to IT8322185A priority Critical patent/IT1206505B/it
Priority to NZ208761A priority patent/NZ208761A/en
Priority to ZA845095A priority patent/ZA845095B/xx
Priority to US06/628,730 priority patent/US4547495A/en
Priority to IL72368A priority patent/IL72368A/xx
Priority to NL8402255A priority patent/NL8402255A/nl
Priority to AT0232384A priority patent/AT392070B/de
Priority to FR8411380A priority patent/FR2567882B1/fr
Priority to KR1019840004202A priority patent/KR910005708B1/ko
Priority to PT78955A priority patent/PT78955B/pt
Priority to JP59149766A priority patent/JPS6042374A/ja
Priority to BE2/60463A priority patent/BE900192A/fr
Priority to CH3557/84A priority patent/CH661508A5/de
Priority to AU30923/84A priority patent/AU560729B2/en
Priority to IE1881/84A priority patent/IE57663B1/en
Priority to DE19843426821 priority patent/DE3426821A1/de
Priority to LU85473A priority patent/LU85473A1/fr
Priority to GR75393A priority patent/GR79983B/el
Priority to DK356484A priority patent/DK165117C/da
Priority to CA000459353A priority patent/CA1223583A/en
Priority to FI842927A priority patent/FI80881C/fi
Priority to SE8403801A priority patent/SE461219B/sv
Priority to ES534539A priority patent/ES8507090A1/es
Priority to GB08418744A priority patent/GB2143532B/en
Application granted granted Critical
Publication of IT1206505B publication Critical patent/IT1206505B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
IT8322185A 1983-07-22 1983-07-22 Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono. IT1206505B (it)

Priority Applications (24)

Application Number Priority Date Filing Date Title
IT8322185A IT1206505B (it) 1983-07-22 1983-07-22 Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono.
NZ208761A NZ208761A (en) 1983-07-22 1984-07-03 1,5-benzothiazepines and pharmaceutial compositions
ZA845095A ZA845095B (en) 1983-07-22 1984-07-03 New benzothiazepines with cardiovascular utility,methods for their preparations and pharmaceutical compositions containing them
US06/628,730 US4547495A (en) 1983-07-22 1984-07-09 1,5-Benzothiazepines with cardiovascular utility, and pharmaceutical compositions containing them
IL72368A IL72368A (en) 1983-07-22 1984-07-10 5-2(dialkylaminoethyl)-4-oxo-2-(substituted phenyl)-1,5-benzothiazepin-3-ol-esters with cardiovascular utility,methods for their preparation and pharmaceutical compositions containing them
NL8402255A NL8402255A (nl) 1983-07-22 1984-07-17 Nieuwe 1,5-benzothiazepinen met cardiovasculaire toepassing, werkwijzen voor hun bereiding en farmaceutische preparaten die ze bevatten.
AT0232384A AT392070B (de) 1983-07-22 1984-07-18 Verfahren zur herstellung neuer 1,5-benzothiazepine
FR8411380A FR2567882B1 (fr) 1983-07-22 1984-07-18 Nouvelles 1,5-benzothiazepines a activite cardiovasculaire, procedes pour leur preparation et compositions pharmaceutiques les contenant
KR1019840004202A KR910005708B1 (ko) 1983-07-22 1984-07-18 1,5-벤조티아제핀 유도체의 제조방법
CH3557/84A CH661508A5 (de) 1983-07-22 1984-07-20 1,5-benzothiazepine mit cardiovascularer wirksamkeit, verfahren zu ihrer herstellung und pharmazeutische praeparate, welche diese verbindungen enthalten.
DK356484A DK165117C (da) 1983-07-22 1984-07-20 1,5-benzothiazepin, fremgangsmaade til fremstilling deraf og farmaceutisk praeparat indeholdende en saadan forbindelse
BE2/60463A BE900192A (fr) 1983-07-22 1984-07-20 Nouvelles 1,5-benzothiazepines d'utilite cardiovasculaire, procedes pour leur preparation et compositions pharmaceutiques en contenant.
PT78955A PT78955B (en) 1983-07-22 1984-07-20 New 1,5-benzothiazepines with cardiovascular utility methods for their preparations and pharmaceutical compositions containing them
AU30923/84A AU560729B2 (en) 1983-07-22 1984-07-20 1,5-benzothiazepine derivatives
IE1881/84A IE57663B1 (en) 1983-07-22 1984-07-20 1,-5 benzothiazepine derivatives,their preparation and pharmaceutical compositions containing them
DE19843426821 DE3426821A1 (de) 1983-07-22 1984-07-20 1,5-benzothiazepin-verbindungen und ihre salze, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln
LU85473A LU85473A1 (fr) 1983-07-22 1984-07-20 Nouvelles 1,5-benzothiazepines d'utilite cardiovasculaire,procedes pour leur preparation et compositions pharmaceutiques en contenant
GR75393A GR79983B (it) 1983-07-22 1984-07-20
JP59149766A JPS6042374A (ja) 1983-07-22 1984-07-20 新規な1,5−ベンゾチアゼピン類、それらの製造方法およびそれらを含有している製薬学的組成物
CA000459353A CA1223583A (en) 1983-07-22 1984-07-20 1,5-benzothiozepines with cardiovascular activity, methods for their preparations and pharmaceutical compositions containing them
FI842927A FI80881C (fi) 1983-07-22 1984-07-20 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1,5-bentsotiazepinderivat.
SE8403801A SE461219B (sv) 1983-07-22 1984-07-20 1,5-bensotiazepiner med kardiovaskulaer anvaendbarhet, foerfarande foer framstaellning daerav samt farmaceutiska kompositioner som innehaaller dem
ES534539A ES8507090A1 (es) 1983-07-22 1984-07-21 Procedimiento para la obtencion de nuevas 1, 5-benzotiacepinas
GB08418744A GB2143532B (en) 1983-07-22 1984-07-23 1,-5 benzothiazepine derivatives, their preparation and pharmaceutical compositions containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8322185A IT1206505B (it) 1983-07-22 1983-07-22 Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono.

Publications (2)

Publication Number Publication Date
IT8322185A0 IT8322185A0 (it) 1983-07-22
IT1206505B true IT1206505B (it) 1989-04-27

Family

ID=11192749

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8322185A IT1206505B (it) 1983-07-22 1983-07-22 Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono.

Country Status (24)

Country Link
US (1) US4547495A (it)
JP (1) JPS6042374A (it)
KR (1) KR910005708B1 (it)
AT (1) AT392070B (it)
AU (1) AU560729B2 (it)
BE (1) BE900192A (it)
CA (1) CA1223583A (it)
CH (1) CH661508A5 (it)
DE (1) DE3426821A1 (it)
DK (1) DK165117C (it)
ES (1) ES8507090A1 (it)
FI (1) FI80881C (it)
FR (1) FR2567882B1 (it)
GB (1) GB2143532B (it)
GR (1) GR79983B (it)
IE (1) IE57663B1 (it)
IL (1) IL72368A (it)
IT (1) IT1206505B (it)
LU (1) LU85473A1 (it)
NL (1) NL8402255A (it)
NZ (1) NZ208761A (it)
PT (1) PT78955B (it)
SE (1) SE461219B (it)
ZA (1) ZA845095B (it)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4925837A (en) * 1984-09-14 1990-05-15 Synthelabo Pharmaceutical compositions
GB2167063A (en) * 1984-11-17 1986-05-21 Tanabe Seiyaku Co 6 or 9-chloro-1, 5-benzothiazepine derivatives
US4584131A (en) * 1985-06-20 1986-04-22 E. R. Squibb & Sons, Inc. Benzothiazepine derivatives
USRE33072E (en) * 1985-06-20 1989-09-26 E. R. Squibb & Sons, Inc. Benzothiazepine derivatives
US4652561A (en) * 1986-02-26 1987-03-24 Hoffmann-La Roche Inc. Naphtho[1,2-b]-1,4-thiazepinones
IL81954A0 (en) * 1986-03-24 1987-10-20 Hoffmann La Roche Naphthothiazocinones,their manufacture and pharmaceutical compositions containing them
JPS63275572A (ja) * 1987-05-01 1988-11-14 Tanabe Seiyaku Co Ltd 1,5−ベンゾチアゼピン誘導体
JP2703564B2 (ja) * 1987-07-31 1998-01-26 田辺製薬株式会社 1,5−ベンゾチアゼピン誘導体
US4808580A (en) * 1987-12-17 1989-02-28 Hoffmann-La Roche Inc. Naphtho[1,2-b][1,4]thiazepin-4(5H)-ones and use thereof in treatment of ischemia and blood pressure lowering
US4912102A (en) * 1988-02-01 1990-03-27 Hoffmann-La Roche Inc. Analogs of naphtho[1,2-β] [1,4] thiazepin-4(5H)-one
JP2674232B2 (ja) * 1989-08-31 1997-11-12 田辺製薬株式会社 1,5―ベンゾチアゼピン誘導体
US5001236A (en) * 1989-11-22 1991-03-19 Marion Laboratories, Inc. Benzothiazepines
IT1240686B (it) * 1990-04-27 1993-12-17 Luso Farmaco Inst Derivati 1,5-benzotiazepinonici, loro preparazione e uso farmaceutico
JP3151163B2 (ja) * 1997-01-24 2001-04-03 ソニーケミカル株式会社 記録用シート及びその記録用シートを使った記録方法
KR100397799B1 (ko) * 2001-07-11 2003-09-13 송기만 조명갓의 표면처리 방법
KR100436262B1 (ko) * 2002-01-04 2004-06-16 삼성전자주식회사 전자레인지용 램프의 제조방법
AU2009332930A1 (en) * 2008-02-01 2009-08-13 The Scripps Research Institute Methods for treating a condition characterized by dysfunction in protein homeostasis

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5899471A (ja) * 1981-12-07 1983-06-13 Tanabe Seiyaku Co Ltd ベンゾチアゼピン誘導体の新規製造法

Also Published As

Publication number Publication date
PT78955B (en) 1986-06-05
ES534539A0 (es) 1985-09-16
SE8403801L (sv) 1985-01-23
CA1223583A (en) 1987-06-30
US4547495A (en) 1985-10-15
KR850001184A (ko) 1985-03-16
AU560729B2 (en) 1987-04-16
DK356484D0 (da) 1984-07-20
FI842927A0 (fi) 1984-07-20
IL72368A (en) 1987-11-30
SE8403801D0 (sv) 1984-07-20
IL72368A0 (en) 1984-11-30
KR910005708B1 (ko) 1991-08-02
SE461219B (sv) 1990-01-22
GB2143532A (en) 1985-02-13
AT392070B (de) 1991-01-25
NL8402255A (nl) 1985-02-18
CH661508A5 (de) 1987-07-31
PT78955A (en) 1984-08-01
GB2143532B (en) 1986-06-25
GR79983B (it) 1984-10-31
NZ208761A (en) 1987-04-30
DK165117C (da) 1993-03-01
DK356484A (da) 1985-01-23
IE57663B1 (en) 1993-02-24
ATA232384A (de) 1990-07-15
DK165117B (da) 1992-10-12
FI842927A (fi) 1985-01-23
FI80881C (fi) 1990-08-10
JPS6042374A (ja) 1985-03-06
DE3426821C2 (it) 1992-01-23
BE900192A (fr) 1984-11-16
IT8322185A0 (it) 1983-07-22
AU3092384A (en) 1985-01-24
FI80881B (fi) 1990-04-30
FR2567882B1 (fr) 1987-08-14
DE3426821A1 (de) 1985-01-31
GB8418744D0 (en) 1984-08-30
FR2567882A1 (fr) 1986-01-24
ES8507090A1 (es) 1985-09-16
LU85473A1 (fr) 1985-04-17
ZA845095B (en) 1985-04-24
IE841881L (en) 1985-01-22

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