IS3970A - Hliðstæð aðferð til framleiðslu á 1,5-benzódíazepín afleiðum - Google Patents

Hliðstæð aðferð til framleiðslu á 1,5-benzódíazepín afleiðum

Info

Publication number
IS3970A
IS3970A IS3970A IS3970A IS3970A IS 3970 A IS3970 A IS 3970A IS 3970 A IS3970 A IS 3970A IS 3970 A IS3970 A IS 3970A IS 3970 A IS3970 A IS 3970A
Authority
IS
Iceland
Prior art keywords
preparation
analogous method
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
IS3970A
Other languages
English (en)
Inventor
Finch Harry
Trist David
Tarzia Giorgio
Original Assignee
Glaxo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Spa filed Critical Glaxo Spa
Publication of IS3970A publication Critical patent/IS3970A/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/121,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
IS3970A 1992-01-21 1993-01-20 Hliðstæð aðferð til framleiðslu á 1,5-benzódíazepín afleiðum IS3970A (is)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929201180A GB9201180D0 (en) 1992-01-21 1992-01-21 Chemical compounds

Publications (1)

Publication Number Publication Date
IS3970A true IS3970A (is) 1993-07-22

Family

ID=10708914

Family Applications (1)

Application Number Title Priority Date Filing Date
IS3970A IS3970A (is) 1992-01-21 1993-01-20 Hliðstæð aðferð til framleiðslu á 1,5-benzódíazepín afleiðum

Country Status (29)

Country Link
US (2) US5580895A (is)
JP (1) JP3253723B2 (is)
KR (1) KR100263625B1 (is)
CN (1) CN1049217C (is)
AP (1) AP369A (is)
AU (2) AU3450193A (is)
BG (1) BG61876B1 (is)
CA (1) CA2087672C (is)
CZ (1) CZ283950B6 (is)
FI (1) FI111632B (is)
GB (1) GB9201180D0 (is)
GE (1) GEP20001968B (is)
HU (2) HU221297B1 (is)
IL (1) IL104447A (is)
IS (1) IS3970A (is)
MX (1) MX9300261A (is)
MY (1) MY131307A (is)
NO (1) NO305952B1 (is)
NZ (1) NZ245715A (is)
OA (1) OA09964A (is)
PH (1) PH30894A (is)
PL (1) PL175340B1 (is)
RO (1) RO114128B1 (is)
RU (1) RU2124009C1 (is)
SK (1) SK280173B6 (is)
TW (1) TW226013B (is)
UA (1) UA29416C2 (is)
WO (1) WO1993014074A1 (is)
ZA (1) ZA93375B (is)

Families Citing this family (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9225492D0 (en) * 1992-12-05 1993-01-27 Glaxo Group Ltd Amine derivatives
CN1120845A (zh) * 1993-04-15 1996-04-17 格拉克索有限公司 具有cck和/或胃泌素拮抗活性的1,5-苯并二氮杂䓬衍生物
GB9307833D0 (en) * 1993-04-15 1993-06-02 Glaxo Inc Modulators of cholecystokinin and gastrin
GB9308421D0 (en) * 1993-04-23 1993-06-09 Glaxo Spa Chemical compounds
GB9308431D0 (en) * 1993-04-23 1993-06-09 Glaxo Spa Chemical compounds
GB9314977D0 (en) * 1993-07-20 1993-09-01 Glaxo Spa Chemical compounds
GB9315018D0 (en) * 1993-07-20 1993-09-01 Glaxo Spa Chemical compounds
GB2280182A (en) * 1993-07-20 1995-01-25 Glaxo Spa Benzodiazepine derivatives
GB9314981D0 (en) * 1993-07-20 1993-09-01 Glaxo Spa Chemical compounds
US5739129A (en) * 1994-04-14 1998-04-14 Glaxo Wellcome Inc. CCK or gastrin modulating 5-heterocyclic-1, 5 benzodiazepines
HUT76135A (en) * 1994-04-14 1997-06-30 Glaxo Wellcome Inc Cholecystokinin and gastrin modulating 5-heterocyclic-1,5-benzodiazepines
PE27497A1 (es) * 1994-04-15 1997-08-07 Glaxo Inc Derivados de 1,5 benzodiazepina
US5780464A (en) * 1994-10-14 1998-07-14 Glaxo Wellcome Inc. Enteric coated compositions of 1,5-benzodiazepine derivatives having CCK antagonistic or agonistic activity
GB9420748D0 (en) * 1994-10-14 1994-11-30 Glaxo Inc 1,5 benzodiazepine derivatives
IL124808A0 (en) 1995-12-11 1999-01-26 New England Medical Center Inc Assay for and uses of peptide hormone receptor ligands
US5750353A (en) * 1995-12-11 1998-05-12 New England Medical Center Hospitals, Inc. Assay for non-peptide agonists to peptide hormone receptors
AU721081B2 (en) * 1996-12-10 2000-06-22 Zeria Pharmaceutical Co., Ltd. 1,5-benzodiazepine derivatives
JP4613157B2 (ja) * 2003-01-14 2011-01-12 サイトキネティクス・インコーポレーテッド 化合物、組成物および方法
GB0307918D0 (en) * 2003-04-05 2003-05-14 Astrazeneca Ab Therapeutic use
CA2545513C (en) * 2003-11-18 2013-01-08 Boehringer Ingelheim International Gmbh Solid pharmaceutical preparation form
PL1765327T3 (pl) 2004-06-17 2015-01-30 Cytokinetics Inc Związki, kompozycje i sposoby
US7538223B2 (en) 2005-08-04 2009-05-26 Cytokinetics, Inc. Compounds, compositions and methods
US7825120B2 (en) 2005-12-15 2010-11-02 Cytokinetics, Inc. Certain substituted ((piperazin-1-ylmethyl)benzyl)ureas
WO2007070683A2 (en) 2005-12-15 2007-06-21 Cytokinetics, Inc. Certain chemical entities, compositions and methods
EP1959962A2 (en) 2005-12-16 2008-08-27 Cytokinetics, Inc. Certain chemical entities, compositions, and methods
US7989455B2 (en) 2005-12-19 2011-08-02 Cytokinetics, Inc. Compounds, compositions and methods
CU20090172A6 (es) 2009-10-09 2011-10-05 Facultad De Quimica Universidad De La Habana Sistemas tricíclicos y tetracíclicos con actividad sobre el sistema nervioso central y vascular
ES2613808T3 (es) 2011-07-29 2017-05-26 Oncotherapy Science, Inc. Péptido derivado de ERAP1 y uso del mismo
CN103435562B (zh) * 2013-08-26 2016-02-24 华东理工大学 6-取代苯并二氮卓-2,4-二酮类化合物及其用途
PL3324977T3 (pl) 2015-07-22 2022-11-14 Enanta Pharmaceuticals, Inc. Pochodne benzodiazepiny jako inhibitory rsv
US20170226129A1 (en) 2016-01-15 2017-08-10 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
ES2923521T3 (es) 2017-02-16 2022-09-28 Enanta Pharm Inc Procesos para la preparación de derivados de benzodiazepina
US10752598B2 (en) * 2017-06-07 2020-08-25 Enanta Pharmaceuticals, Inc. Aryldiazepine derivatives as RSV inhibitors
US10851115B2 (en) 2017-06-30 2020-12-01 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
WO2019006295A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
CA3077309A1 (en) 2017-09-29 2019-04-04 Enanta Pharmaceuticals, Inc. Combination pharmaceutical agents as rsv inhibitors
US10647711B2 (en) 2017-11-13 2020-05-12 Enanta Pharmaceuticals, Inc. Azepin-2-one derivatives as RSV inhibitors
US10975094B2 (en) 2018-04-11 2021-04-13 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
EP3889264A4 (en) 2018-11-30 2022-10-12 Tokushima University BREAST CANCER THERAPEUTIC WITH BIG3-PHB2 INTERACTION INHIBITING PEPTIDE FROM PHB2
US11254664B2 (en) 2019-03-18 2022-02-22 Enanta Pharmaceuticals, Inc. Benzodiazepine derivatives as RSV inhibitors
WO2020210246A1 (en) 2019-04-09 2020-10-15 Enanta Pharmaceuticals, Inc, Heterocyclic compounds as rsv inhibitors
US11505558B1 (en) 2019-10-04 2022-11-22 Enanta Pharmaceuticals, Inc. Antiviral heterocyclic compounds
UY39032A (es) 2020-01-24 2021-07-30 Enanta Pharm Inc Compuestos heterocíclicos como agentes antivirales
US11534439B2 (en) 2020-07-07 2022-12-27 Enanta Pharmaceuticals, Inc. Dihydroquinoxaline and dihydropyridopyrazine derivatives as RSV inhibitors
US11945824B2 (en) 2020-10-19 2024-04-02 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as anti-viral agents

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2641280B1 (fr) * 1988-12-29 1994-01-21 Roussel Uclaf Nouveaux derives de la 2,4-dioxo 2,3,4,5-tetrahydro 1h-1,5-benzodiazepine, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
PL175340B1 (pl) 1998-12-31
US5637697A (en) 1997-06-10
HU221297B1 (en) 2002-09-28
AU3193593A (en) 1993-07-22
IL104447A (en) 1998-02-22
CN1074678A (zh) 1993-07-28
RO114128B1 (ro) 1999-01-29
SK280173B6 (sk) 1999-09-10
CN1049217C (zh) 2000-02-09
NZ245715A (en) 1995-07-26
GB9201180D0 (en) 1992-03-11
AP369A (en) 1994-11-06
ZA93375B (en) 1994-07-18
FI943421A (fi) 1994-07-19
CA2087672C (en) 2003-08-05
OA09964A (en) 1995-12-11
PH30894A (en) 1997-12-23
US5580895A (en) 1996-12-03
CA2087672A1 (en) 1993-07-22
KR100263625B1 (ko) 2000-11-01
GEP20001968B (en) 2000-03-05
FI111632B (fi) 2003-08-29
BG98881A (bg) 1995-03-31
MY131307A (en) 2007-08-30
FI943421A0 (fi) 1994-07-19
CZ173694A3 (en) 1995-09-13
JPH07118244A (ja) 1995-05-09
HUT67375A (en) 1995-03-28
TW226013B (is) 1994-07-01
HU9402150D0 (en) 1994-09-28
RU94037768A (ru) 1996-08-10
NO305952B1 (no) 1999-08-23
SK86494A3 (en) 1995-03-08
AU661749B2 (en) 1995-08-03
HU211295A9 (en) 1995-11-28
NO942720L (no) 1994-07-20
BG61876B1 (bg) 1998-08-31
NO942720D0 (no) 1994-07-20
UA29416C2 (uk) 2000-11-15
CZ283950B6 (cs) 1998-07-15
AU3450193A (en) 1993-08-03
IL104447A0 (en) 1993-05-13
RU2124009C1 (ru) 1998-12-27
MX9300261A (es) 1994-03-31
AP9300478A0 (en) 1993-01-31
JP3253723B2 (ja) 2002-02-04
WO1993014074A1 (en) 1993-07-22

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