IN2014MN01754A - - Google Patents

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Publication number
IN2014MN01754A
IN2014MN01754A IN1754MUN2014A IN2014MN01754A IN 2014MN01754 A IN2014MN01754 A IN 2014MN01754A IN 1754MUN2014 A IN1754MUN2014 A IN 1754MUN2014A IN 2014MN01754 A IN2014MN01754 A IN 2014MN01754A
Authority
IN
India
Prior art keywords
formula
present
compounds
heteroaryl
comounds
Prior art date
Application number
Other languages
English (en)
Inventor
Bhavesh Dave
Rakesh Kumar Banerjee
Samiron Phukan
Abhijit Datta Khoje
Rajkumar Hangarge
Jitendra Sambhaji Jadhav
Venkata P Palle
Rajender Kumar Kamboj
Original Assignee
Lupin Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47997632&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014MN01754(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lupin Ltd filed Critical Lupin Ltd
Priority to IN1754MUN2014 priority Critical patent/IN2014MN01754A/en
Publication of IN2014MN01754A publication Critical patent/IN2014MN01754A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541Non-condensed thiazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61NELECTROTHERAPY; MAGNETOTHERAPY; RADIATION THERAPY; ULTRASOUND THERAPY
    • A61N5/00Radiation therapy
    • A61N5/10X-ray therapy; Gamma-ray therapy; Particle-irradiation therapy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Radiology & Medical Imaging (AREA)
  • Pathology (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
IN1754MUN2014 2012-03-14 2013-03-11 IN2014MN01754A (pm)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IN1754MUN2014 IN2014MN01754A (pm) 2012-03-14 2013-03-11

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN288KO2012 2012-03-14
IN1754MUN2014 IN2014MN01754A (pm) 2012-03-14 2013-03-11
PCT/IB2013/051915 WO2013136254A1 (en) 2012-03-14 2013-03-11 Heterocyclyl compounds

Publications (1)

Publication Number Publication Date
IN2014MN01754A true IN2014MN01754A (pm) 2015-07-03

Family

ID=47997632

Family Applications (2)

Application Number Title Priority Date Filing Date
IN1755MUN2014 IN2014MN01755A (pm) 2012-03-14 2013-03-11
IN1754MUN2014 IN2014MN01754A (pm) 2012-03-14 2013-03-11

Family Applications Before (1)

Application Number Title Priority Date Filing Date
IN1755MUN2014 IN2014MN01755A (pm) 2012-03-14 2013-03-11

Country Status (35)

Country Link
US (5) US9573944B2 (pm)
EP (2) EP2834237B1 (pm)
JP (3) JP6093384B2 (pm)
KR (4) KR20140138911A (pm)
CN (4) CN108383836B (pm)
AP (2) AP3859A (pm)
AU (4) AU2013234014B2 (pm)
BR (1) BR112014022713B1 (pm)
CA (2) CA2865164C (pm)
CL (2) CL2014002412A1 (pm)
CO (2) CO7160029A2 (pm)
CR (2) CR20140463A (pm)
CU (2) CU24335B1 (pm)
DK (2) DK2834237T3 (pm)
DO (2) DOP2014000204A (pm)
EA (2) EA029768B1 (pm)
ES (2) ES2684517T3 (pm)
GE (2) GEP201706671B (pm)
GT (2) GT201400196A (pm)
IL (2) IL234560A (pm)
IN (2) IN2014MN01755A (pm)
MA (2) MA37405A1 (pm)
MX (3) MX355474B (pm)
MY (2) MY174188A (pm)
NI (2) NI201400108A (pm)
NZ (2) NZ629442A (pm)
PE (2) PE20141974A1 (pm)
PH (2) PH12014502040A1 (pm)
PL (1) PL2834237T3 (pm)
SG (2) SG11201405006PA (pm)
TN (2) TN2014000357A1 (pm)
TR (1) TR201811976T4 (pm)
UA (2) UA114907C2 (pm)
WO (2) WO2013136249A1 (pm)
ZA (1) ZA201406186B (pm)

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Also Published As

Publication number Publication date
JP2015514056A (ja) 2015-05-18
AP3859A (en) 2016-10-31
PH12014502040B1 (en) 2014-11-24
US9555035B2 (en) 2017-01-31
CU20140110A7 (es) 2014-11-27
NI201400107A (es) 2014-11-26
IL234559A (en) 2017-06-29
CO7160029A2 (es) 2015-01-15
KR102241111B1 (ko) 2021-04-15
KR20190100472A (ko) 2019-08-28
MX355526B (es) 2018-04-20
JP2018115215A (ja) 2018-07-26
ES2684517T3 (es) 2018-10-03
US20160331753A1 (en) 2016-11-17
AU2017200493A1 (en) 2017-02-16
DOP2014000204A (es) 2015-02-15
MX2014010928A (es) 2015-04-10
EA201491672A1 (ru) 2014-12-30
ZA201406186B (en) 2016-06-29
CA2865164C (en) 2021-06-08
JP6093384B2 (ja) 2017-03-08
CR20140463A (es) 2014-11-28
PH12014502040A1 (en) 2014-11-24
KR20190073597A (ko) 2019-06-26
US9969731B2 (en) 2018-05-15
JP6431770B2 (ja) 2018-11-28
NI201400108A (es) 2014-11-28
IL234560A (en) 2017-06-29
ES2741896T3 (es) 2020-02-12
KR20140138911A (ko) 2014-12-04
CN104203947A (zh) 2014-12-10
NZ629442A (en) 2016-12-23
GEP201706671B (en) 2017-05-25
JP6630771B2 (ja) 2020-01-15
HK1206020A1 (en) 2015-12-31
IN2014MN01755A (pm) 2015-07-03
MY174188A (en) 2020-03-12
CR20140464A (es) 2014-11-28
UA114907C2 (uk) 2017-08-28
CU24272B1 (es) 2017-08-08
SG11201405007QA (en) 2014-10-30
EP2834236A1 (en) 2015-02-11
EP2834237B1 (en) 2018-06-06
PH12014502041B1 (en) 2014-11-24
AU2018202568A1 (en) 2018-05-10
CO7170131A2 (es) 2015-01-28
MA37400B1 (fr) 2019-11-29
DK2834236T3 (da) 2019-08-26
MA37400A1 (fr) 2016-05-31
PE20141973A1 (es) 2014-12-12
CA2865164A1 (en) 2013-09-19
AU2013234009A1 (en) 2014-09-25
CN108383836B (zh) 2021-11-12
AP3834A (en) 2016-09-30
CL2014002411A1 (es) 2015-04-06
AU2017200493B2 (en) 2018-03-29
BR112014022713B1 (pt) 2021-09-08
MX366426B (es) 2019-07-08
CL2014002412A1 (es) 2015-03-06
HK1202538A1 (en) 2015-10-02
MA37405A1 (fr) 2016-03-31
EP2834236B1 (en) 2019-05-22
EA029768B1 (ru) 2018-05-31
GEP201706774B (en) 2017-11-27
US20150299186A1 (en) 2015-10-22
PH12014502041A1 (en) 2014-11-24
US20150133424A1 (en) 2015-05-14
EA028232B1 (ru) 2017-10-31
BR112014022713A2 (pm) 2017-06-20
GT201400196A (es) 2017-09-28
WO2013136254A1 (en) 2013-09-19
KR20140138910A (ko) 2014-12-04
DOP2014000203A (es) 2015-02-15
WO2013136249A1 (en) 2013-09-19
TN2014000357A1 (en) 2015-12-21
MX2014010925A (es) 2015-04-10
US20170112840A1 (en) 2017-04-27
AP2014008008A0 (en) 2014-10-31
CN108383836A (zh) 2018-08-10
CU20140109A7 (es) 2014-11-27
CA2865167A1 (en) 2013-09-19
AU2013234014A1 (en) 2014-09-25
DK2834237T3 (en) 2018-08-27
CN104271577A (zh) 2015-01-07
KR102240101B1 (ko) 2021-04-14
CU24335B1 (es) 2018-04-03
UA114906C2 (uk) 2017-08-28
US20170101408A1 (en) 2017-04-13
NZ629432A (en) 2017-01-27
TR201811976T4 (tr) 2018-09-21
EP2834237A1 (en) 2015-02-11
AU2018202568B2 (en) 2019-05-09
GT201400195A (es) 2017-11-09
SG11201405006PA (en) 2014-10-30
PL2834237T3 (pl) 2018-11-30
MY175950A (en) 2020-07-16
TN2014000356A1 (en) 2015-12-21
US9573944B2 (en) 2017-02-21
EA201491671A1 (ru) 2014-12-30
MX355474B (es) 2018-04-16
CN107698585A (zh) 2018-02-16
CA2865167C (en) 2019-08-06
US9428499B2 (en) 2016-08-30
AU2013234014B2 (en) 2017-02-02
PE20141974A1 (es) 2014-12-12
US9827247B2 (en) 2017-11-28
AP2014008009A0 (en) 2014-10-31
AU2013234009B2 (en) 2016-10-27
JP2015509975A (ja) 2015-04-02

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