IL98599A - Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them - Google Patents

Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them

Info

Publication number
IL98599A
IL98599A IL9859991A IL9859991A IL98599A IL 98599 A IL98599 A IL 98599A IL 9859991 A IL9859991 A IL 9859991A IL 9859991 A IL9859991 A IL 9859991A IL 98599 A IL98599 A IL 98599A
Authority
IL
Israel
Prior art keywords
deoxy
epi
acid
avermectin
blb
Prior art date
Application number
IL9859991A
Other languages
English (en)
Hebrew (he)
Other versions
IL98599A0 (en
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of IL98599A0 publication Critical patent/IL98599A0/xx
Publication of IL98599A publication Critical patent/IL98599A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Fodder In General (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Steroid Compounds (AREA)
  • Silicon Polymers (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
IL9859991A 1990-06-28 1991-06-24 Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them IL98599A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54522990A 1990-06-28 1990-06-28

Publications (2)

Publication Number Publication Date
IL98599A0 IL98599A0 (en) 1992-07-15
IL98599A true IL98599A (en) 1995-06-29

Family

ID=24175383

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9859991A IL98599A (en) 1990-06-28 1991-06-24 Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them

Country Status (21)

Country Link
US (1) US5288710A (da)
EP (1) EP0465121B1 (da)
JP (1) JPH0822870B2 (da)
KR (1) KR100224292B1 (da)
AT (1) ATE134377T1 (da)
AU (1) AU641777B2 (da)
CA (1) CA2045864C (da)
CY (1) CY1949A (da)
DE (1) DE69117223T2 (da)
DK (1) DK0465121T3 (da)
ES (1) ES2084110T3 (da)
FI (1) FI97890C (da)
GR (1) GR3019067T3 (da)
HK (1) HK157096A (da)
IE (1) IE71175B1 (da)
IL (1) IL98599A (da)
LV (1) LV5740B4 (da)
NO (2) NO178339C (da)
NZ (1) NZ238705A (da)
PT (1) PT98117B (da)
ZA (1) ZA914961B (da)

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BR9406627A (pt) * 1993-05-26 1996-02-06 Commw Scient Ind Res Org Composições antiparasiticas
AU687062B2 (en) * 1993-05-26 1998-02-19 Commonwealth Scientific And Industrial Research Organisation Controlled release antiparasitic compositions
US6486195B1 (en) * 1993-08-19 2002-11-26 Merck & Co., Inc. Thermodynamically stable crystal form of 4″-deoxy-4″-epi-methylamino avermectin B1a/B1b benzoic acid salt and processes for its preparation
HU217769B (hu) * 1993-08-19 2000-04-28 Merck & Co. Inc. 4"-Dezoxi-4"-epi-metil-amino-avermektin-B1a/B1b benzoesavas sójának termodinamikailag stabil kristályformája és eljárás annak előállítására, hatóanyagként ezt tartalmazó kompozíció és eljárás rovarok lekűzdésére
US5362863A (en) * 1993-09-29 1994-11-08 Merck & Co., Inc. Process for the preparation of 4"-amino avermectin compounds
JP3529792B2 (ja) * 1995-11-08 2004-05-24 メルク エンド カムパニー インコーポレーテッド 農薬製剤
AU768262B2 (en) * 1995-11-08 2003-12-04 Merck Sharp & Dohme Corp. Pesticidal formulation
CN1281127C (zh) 1995-11-08 2006-10-25 麦克公司 农药制剂
US20050192319A1 (en) * 1996-09-19 2005-09-01 Albert Boeckh Spot-on formulations for combating parasites
US6054140A (en) * 1997-03-21 2000-04-25 Biogenesis S.A. Long acting injectable parasiticidal composition and the process for its preparation
WO1999025187A2 (en) * 1997-11-14 1999-05-27 Novartis Ag Pesticidal compositions of emamectin
NZ505208A (en) * 1997-12-23 2003-07-25 Novartis Ag Use of macrolides in pest control
US6486128B1 (en) 1999-04-08 2002-11-26 Schering-Plough Veterinary Corporation Method of using emamectin to treat fish parasites
AR006063A4 (es) * 1999-04-17 1999-08-11 Romario S R L Bandeja termica para pizzas
GB9926887D0 (en) 1999-11-12 2000-01-12 Novartis Ag Organic compounds
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
JP4701538B2 (ja) 2001-05-21 2011-06-15 住友化学株式会社 農業害虫防除剤組成物
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
DE10203688A1 (de) * 2002-01-31 2003-08-07 Bayer Cropscience Ag Synergistische insektizide Mischungen
DE10207242A1 (de) * 2002-02-21 2003-09-04 Bayer Cropscience Ag Synergistische insektizide Mischungen
DE10207241A1 (de) * 2002-02-21 2003-09-04 Bayer Cropscience Ag Synergistische insektizide Mischungen
EP1497283A4 (en) * 2002-03-22 2006-01-11 Lg Life Sciences Ltd (2S) -N-5-AMINO (IMINO) METHYL-2-THIENYL METHYL-1- (2R) -2- (CARBOXYMETHYL) AMINO) 3,3-DIPHENYLPROPANOYL -2-PYRROLIDINE CARBOXAMIDE MALEIC ACID SALT AND PROCESS OF PREPARATION CORRESPONDING
AR040073A1 (es) 2002-05-07 2005-03-16 Syngenta Participations Ag Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
AR054981A1 (es) 2004-09-23 2007-08-01 Schering Plough Ltd Control de parasitos en animales mediante el uso de nuevos derivados de trifluorometansulfonanilida oxima eter
JP4750126B2 (ja) * 2004-11-19 2011-08-17 シェーリング−プラウ・リミテッド 殺寄生虫薬２−フェニル−３−（１ｈ−ピロール−２−イル）アクリロニトリル誘導体の使用による動物における寄生虫の制御
CA2609574A1 (en) * 2005-06-09 2006-12-21 Schering-Plough Ltd. Control of parasites in animals by n-[(phenyloxy)phenyl]-1,1,1-trifluoromethanesulfonamide and n-[(phenylsulfanyl)phenyl]-1,1,1-trifluoromethanesulfonamide derivatives
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
TWI422328B (zh) 2006-06-19 2014-01-11 Univ California 結合有殺線蟲之種子塗覆物的生物控制劑
FR2906469B1 (fr) * 2006-09-28 2008-11-28 Galderma Sa Utilisation de composes de la famille des avermectines pour le traitement de desordres dermatologiques chez l'homme
CN101600686A (zh) * 2006-12-13 2009-12-09 先灵-普劳有限公司 氯霉素、甲砜霉素及其类似物的水溶性前药
CN101605756A (zh) * 2006-12-13 2009-12-16 先灵-普劳有限公司 氟苯尼考及其类似物的水溶性前药
DE102007002872A1 (de) 2007-01-15 2008-07-17 Alpha-Biocare Gmbh Verwendung von Avermectin-Derivaten zur Behandlung gegen Parasiten von Fischen
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
HUE037127T2 (hu) 2007-06-27 2018-08-28 Du Pont Állati károkozó irtására szolgáló eljárás
TWI556741B (zh) 2007-08-17 2016-11-11 英特威特國際股份有限公司 異唑啉組成物及其作為抗寄生蟲藥上的應用
TWI401023B (zh) 2008-02-06 2013-07-11 Du Pont 中離子農藥
CA2732017A1 (en) * 2008-07-30 2010-02-04 Intervet International B.V. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
CN102355891A (zh) 2009-03-17 2012-02-15 英特威国际有限公司 大环内酯药物递送系统
IN2012DN00709A (da) 2009-08-05 2015-06-19 Du Pont
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
WO2011017347A2 (en) 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
UY33397A (es) 2010-05-27 2011-12-01 Du Pont Forma sólida de un naftaleno carboxamida
AR081970A1 (es) 2010-06-24 2012-10-31 Intervet Int Bv Formulacion inyectable de una lactona macrociclica y levamisol, formulacion y uso veterinario
EP2629772B1 (en) 2010-10-20 2016-05-18 Galderma S.A. Ivermectin for use in the treatment of hemorrhoids
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
EP2658541B1 (en) 2010-12-27 2022-01-26 Intervet International B.V. Topical localized isoxazoline formulation comprising glycofurol
MX356926B (es) 2010-12-27 2018-06-19 Intervet Int Bv Formulación de isoxazolina tópica localizada.
BR112014001950B1 (pt) 2011-07-28 2021-01-12 Syngenta Participations Ag métodos para controle de uma praga de nemátodos e para produzir uma planta de soja protegida contra infestação de nemátodos
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
US9643991B2 (en) * 2015-06-08 2017-05-09 Rotam Agrochem International Company Limited Process for preparing a novel crystalline form of emamectin benzoate and use the same
US9409920B1 (en) * 2015-06-08 2016-08-09 Rotam Agrochem International Company Limited Method for purifying emamectin benzoate and compositions comprising the same
CN107344954B (zh) * 2017-08-07 2020-08-11 河北蓝泰化工科技有限公司 增效型甲氨基阿维菌素b1或b2的盐及制备方法和应用
CN108840893A (zh) * 2018-07-01 2018-11-20 李万强 一种甲氨基阿维菌素苯甲酸盐的新晶型及其制备方法
CN108864230B (zh) * 2018-07-26 2021-05-14 河北威远生物化工有限公司 一种有机磷基团取代的阿维菌素衍生物及其制备方法和应用

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US4366309A (en) * 1980-03-14 1982-12-28 Schering Corporation Derivatives of antibiotic AR-5 components
US4321362A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company De(mycinosyloxy)tylosin and process for its production
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4874749A (en) * 1987-07-31 1989-10-17 Merck & Co., Inc. 4"-Deoxy-4-N-methylamino avermectin Bla/Blb

Also Published As

Publication number Publication date
CY1949A (en) 1991-06-27
JPH05306294A (ja) 1993-11-19
KR100224292B1 (ko) 1999-10-15
DE69117223T2 (de) 1996-09-12
FI97890C (fi) 1997-03-10
NO178339B (no) 1995-11-27
EP0465121B1 (en) 1996-02-21
NO912535D0 (no) 1991-06-27
GR3019067T3 (en) 1996-05-31
DK0465121T3 (da) 1996-03-18
FI913137A0 (fi) 1991-06-27
KR920000781A (ko) 1992-01-29
PT98117B (pt) 1998-12-31
FI913137A (fi) 1991-12-29
IL98599A0 (en) 1992-07-15
EP0465121A1 (en) 1992-01-08
DE69117223D1 (de) 1996-03-28
PT98117A (pt) 1993-10-29
LV5740A4 (lv) 1996-08-20
AU7939291A (en) 1992-01-02
FI97890B (fi) 1996-11-29
NZ238705A (en) 1993-07-27
NO2001007I2 (no) 2007-02-26
ZA914961B (en) 1992-07-29
AU641777B2 (en) 1993-09-30
JPH0822870B2 (ja) 1996-03-06
US5288710A (en) 1994-02-22
ATE134377T1 (de) 1996-03-15
LV5740B4 (lv) 1997-12-20
IE71175B1 (en) 1997-01-29
NO178339C (no) 1996-03-06
NO912535L (no) 1991-12-30
IE912251A1 (en) 1992-01-01
ES2084110T3 (es) 1996-05-01
CA2045864A1 (en) 1991-12-29
HK157096A (en) 1996-08-23
CA2045864C (en) 2001-11-27

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