NO2001007I2 - Stabile salter av 4"-deoksy-4"-epimetylaminoavermectin B1a/B1b med egenskaper som landbruksinsekticid og preparater inneholdende et slikt salt - Google Patents

Stabile salter av 4"-deoksy-4"-epimetylaminoavermectin B1a/B1b med egenskaper som landbruksinsekticid og preparater inneholdende et slikt salt

Info

Publication number
NO2001007I2
NO2001007I2 NO2001007C NO2001007C NO2001007I2 NO 2001007 I2 NO2001007 I2 NO 2001007I2 NO 2001007 C NO2001007 C NO 2001007C NO 2001007 C NO2001007 C NO 2001007C NO 2001007 I2 NO2001007 I2 NO 2001007I2
Authority
NO
Norway
Prior art keywords
acid salt
deoxy
salt
epimethylaminoavermectin
properties
Prior art date
Application number
NO2001007C
Other languages
English (en)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of NO2001007I2 publication Critical patent/NO2001007I2/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Silicon Polymers (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Fodder In General (AREA)
  • Steroid Compounds (AREA)
NO2001007C 1990-06-28 1991-06-27 Stabile salter av 4"-deoksy-4"-epimetylaminoavermectin B1a/B1b med egenskaper som landbruksinsekticid og preparater inneholdende et slikt salt NO2001007I2 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54522990A 1990-06-28 1990-06-28

Publications (1)

Publication Number Publication Date
NO2001007I2 true NO2001007I2 (no) 2007-02-26

Family

ID=24175383

Family Applications (2)

Application Number Title Priority Date Filing Date
NO2001007C NO2001007I2 (no) 1990-06-28 1991-06-27 Stabile salter av 4"-deoksy-4"-epimetylaminoavermectin B1a/B1b med egenskaper som landbruksinsekticid og preparater inneholdende et slikt salt
NO912535A NO178339C (no) 1990-06-28 1991-06-27 Stabile salter av 4''-deoksy-4''-epi-metylaminoavermectin B1a/Blb med egenskaper som landbruksinsekticid og preparater inneholdende et slikt salt

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO912535A NO178339C (no) 1990-06-28 1991-06-27 Stabile salter av 4''-deoksy-4''-epi-metylaminoavermectin B1a/Blb med egenskaper som landbruksinsekticid og preparater inneholdende et slikt salt

Country Status (21)

Country Link
US (1) US5288710A (no)
EP (1) EP0465121B1 (no)
JP (1) JPH0822870B2 (no)
KR (1) KR100224292B1 (no)
AT (1) ATE134377T1 (no)
AU (1) AU641777B2 (no)
CA (1) CA2045864C (no)
CY (1) CY1949A (no)
DE (1) DE69117223T2 (no)
DK (1) DK0465121T3 (no)
ES (1) ES2084110T3 (no)
FI (1) FI97890C (no)
GR (1) GR3019067T3 (no)
HK (1) HK157096A (no)
IE (1) IE71175B1 (no)
IL (1) IL98599A (no)
LV (1) LV5740B4 (no)
NO (2) NO2001007I2 (no)
NZ (1) NZ238705A (no)
PT (1) PT98117B (no)
ZA (1) ZA914961B (no)

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GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
ES2314724T3 (es) 2004-09-23 2009-03-16 Schering-Plough Ltd. Control de parasitos en animales mediante el uso de nuevos derivados de eter de trifluorometanosulfonanilida oxima.
CA2587495A1 (en) * 2004-11-19 2006-05-26 Schering-Plough Ltd. Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives
MX2007015729A (es) * 2005-06-09 2008-02-21 Schering Plough Ltd Control de parasitos en animales con derivados de n-[(feniloxi)fenil]-1,1,1-trifluorometansulfonamida y de n[(fenilsulfanil)fenil]-1,1,1-trifluorometansulfonamida.
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
TWI422328B (zh) 2006-06-19 2014-01-11 Univ California 結合有殺線蟲之種子塗覆物的生物控制劑
FR2906469B1 (fr) * 2006-09-28 2008-11-28 Galderma Sa Utilisation de composes de la famille des avermectines pour le traitement de desordres dermatologiques chez l'homme
WO2008076256A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
MX2009006282A (es) * 2006-12-13 2009-06-23 Schering Plough Ltd Profarmacos solubles en agua de florfenicol y sus analogos.
DE102007002872A1 (de) 2007-01-15 2008-07-17 Alpha-Biocare Gmbh Verwendung von Avermectin-Derivaten zur Behandlung gegen Parasiten von Fischen
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
BRPI0810929B8 (pt) 2007-06-27 2022-12-06 Du Pont uso de um composto de fórmula 1
TWI556741B (zh) 2007-08-17 2016-11-11 英特威特國際股份有限公司 異唑啉組成物及其作為抗寄生蟲藥上的應用
TWI401023B (zh) 2008-02-06 2013-07-11 Du Pont 中離子農藥
US8314252B2 (en) * 2008-07-30 2012-11-20 Intervet Inc. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
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UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
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UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
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ES2566402T3 (es) 2010-05-27 2016-04-12 E. I. Du Pont De Nemours And Company Forma cristalina de 4-[5-[3-cloro-5-(trifluorometil)fenil]-4,5-dihidro-5-(trifluorometil)-3-isoxazolil]-N-[2-oxo-2-[(2,2,2-trifluoroetil)amino]etil]-1-naftalenocarboxamida
AR081970A1 (es) 2010-06-24 2012-10-31 Intervet Int Bv Formulacion inyectable de una lactona macrociclica y levamisol, formulacion y uso veterinario
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MX348079B (es) 2010-12-27 2017-05-25 Intervet Int Bv Formulacion de isoxazolina topica localizada que comprende glucofurol.
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US9643991B2 (en) * 2015-06-08 2017-05-09 Rotam Agrochem International Company Limited Process for preparing a novel crystalline form of emamectin benzoate and use the same
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CN107344954B (zh) * 2017-08-07 2020-08-11 河北蓝泰化工科技有限公司 增效型甲氨基阿维菌素b1或b2的盐及制备方法和应用
CN108840893A (zh) * 2018-07-01 2018-11-20 李万强 一种甲氨基阿维菌素苯甲酸盐的新晶型及其制备方法
CN108864230B (zh) * 2018-07-26 2021-05-14 河北威远生物化工有限公司 一种有机磷基团取代的阿维菌素衍生物及其制备方法和应用

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Also Published As

Publication number Publication date
LV5740B4 (lv) 1997-12-20
HK157096A (en) 1996-08-23
IE71175B1 (en) 1997-01-29
ES2084110T3 (es) 1996-05-01
FI97890C (fi) 1997-03-10
NO912535L (no) 1991-12-30
US5288710A (en) 1994-02-22
ZA914961B (en) 1992-07-29
GR3019067T3 (en) 1996-05-31
DE69117223T2 (de) 1996-09-12
EP0465121A1 (en) 1992-01-08
JPH05306294A (ja) 1993-11-19
PT98117B (pt) 1998-12-31
NO178339B (no) 1995-11-27
NZ238705A (en) 1993-07-27
AU7939291A (en) 1992-01-02
NO912535D0 (no) 1991-06-27
CA2045864A1 (en) 1991-12-29
KR100224292B1 (ko) 1999-10-15
NO178339C (no) 1996-03-06
JPH0822870B2 (ja) 1996-03-06
EP0465121B1 (en) 1996-02-21
IE912251A1 (en) 1992-01-01
FI913137A (fi) 1991-12-29
FI913137A0 (fi) 1991-06-27
FI97890B (fi) 1996-11-29
LV5740A4 (lv) 1996-08-20
DE69117223D1 (de) 1996-03-28
DK0465121T3 (da) 1996-03-18
ATE134377T1 (de) 1996-03-15
IL98599A0 (en) 1992-07-15
IL98599A (en) 1995-06-29
CA2045864C (en) 2001-11-27
CY1949A (en) 1991-06-27
KR920000781A (ko) 1992-01-29
AU641777B2 (en) 1993-09-30
PT98117A (pt) 1993-10-29

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