IL173382A0 - Amino acid prodrugs - Google Patents
Amino acid prodrugsInfo
- Publication number
- IL173382A0 IL173382A0 IL173382A IL17338206A IL173382A0 IL 173382 A0 IL173382 A0 IL 173382A0 IL 173382 A IL173382 A IL 173382A IL 17338206 A IL17338206 A IL 17338206A IL 173382 A0 IL173382 A0 IL 173382A0
- Authority
- IL
- Israel
- Prior art keywords
- amino acid
- acid prodrugs
- prodrugs
- amino
- acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/02—Peptides of undefined number of amino acids; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
- A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/64—Cyclic peptides containing only normal peptide links
- C07K7/645—Cyclosporins; Related peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Pain & Pain Management (AREA)
- Gastroenterology & Hepatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49133103P | 2003-07-29 | 2003-07-29 | |
PCT/US2004/024901 WO2005046575A2 (en) | 2003-07-29 | 2004-07-29 | Amino acid prodrugs |
Publications (1)
Publication Number | Publication Date |
---|---|
IL173382A0 true IL173382A0 (en) | 2006-06-11 |
Family
ID=34590076
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL173382A IL173382A0 (en) | 2003-07-29 | 2006-01-26 | Amino acid prodrugs |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP1660017A4 (de) |
JP (2) | JP2007510621A (de) |
KR (3) | KR20130081319A (de) |
CN (1) | CN101123878A (de) |
AU (1) | AU2004289174B2 (de) |
CA (1) | CA2534342C (de) |
IL (1) | IL173382A0 (de) |
NZ (3) | NZ545570A (de) |
SG (2) | SG145693A1 (de) |
WO (1) | WO2005046575A2 (de) |
ZA (1) | ZA200600660B (de) |
Families Citing this family (108)
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CN116041259A (zh) * | 2023-01-13 | 2023-05-02 | 武汉科技大学 | 一种羟氯喹的衍生物及其制备方法 |
Family Cites Families (11)
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US4650803A (en) * | 1985-12-06 | 1987-03-17 | University Of Kansas | Prodrugs of rapamycin |
US5411947A (en) * | 1989-06-28 | 1995-05-02 | Vestar, Inc. | Method of converting a drug to an orally available form by covalently bonding a lipid to the drug |
CA2102116A1 (en) * | 1991-05-31 | 1992-12-01 | Gary R. Schulte | Use of rapamycin prodrugs as immunosuppressant agents |
US5972379A (en) * | 1995-02-14 | 1999-10-26 | Sequus Pharmaceuticals, Inc. | Liposome composition and method for administering a quinolone |
JPH1143467A (ja) * | 1997-05-14 | 1999-02-16 | Ikeda Mohandou:Kk | 脂肪酸グリセライド誘導体及びグリセライド誘導体、並びにそれらの製造方法 |
IT1294205B1 (it) * | 1997-07-23 | 1999-03-24 | Farmigea Spa | Procedimento per la solubilizzazione in acqua e in veicoli acquosi di sostanze farmacologicamente attive |
US6569842B2 (en) * | 2000-08-18 | 2003-05-27 | Board Of Trustees Of The University Of Illinois, The | Method of preparing and use of prodrugs of betulinic acid derivatives |
US20020160988A1 (en) * | 2001-02-20 | 2002-10-31 | Israel Institute For Biological Research | Compounds co-inducing cholinergic up-regulation and inflammation down-regulation and uses thereof |
US7045543B2 (en) * | 2001-11-05 | 2006-05-16 | Enzrel Inc. | Covalent conjugates of biologically-active compounds with amino acids and amino acid derivatives for targeting to physiologically-protected sites |
JP2006522125A (ja) * | 2003-03-25 | 2006-09-28 | バーテックス ファーマシューティカルズ インコーポレイテッド | プロテインキナーゼのインヒビターとして有用なチアゾール |
SG145693A1 (en) * | 2003-07-29 | 2008-09-29 | Signature R & D Holdings Llc | Amino acid prodrugs |
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2004
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- 2004-07-29 KR KR1020137015399A patent/KR20130081319A/ko not_active Application Discontinuation
- 2004-07-29 KR KR1020127022817A patent/KR20120116991A/ko not_active Application Discontinuation
- 2004-07-29 WO PCT/US2004/024901 patent/WO2005046575A2/en active Application Filing
- 2004-07-29 CA CA2534342A patent/CA2534342C/en not_active Expired - Fee Related
- 2004-07-29 SG SG2012005310A patent/SG178721A1/en unknown
- 2004-07-29 EP EP04816791A patent/EP1660017A4/de not_active Withdrawn
- 2004-07-29 NZ NZ545570A patent/NZ545570A/xx not_active IP Right Cessation
- 2004-07-29 NZ NZ601780A patent/NZ601780A/xx not_active IP Right Cessation
- 2004-07-29 CN CNA2004800282229A patent/CN101123878A/zh active Pending
- 2004-07-29 JP JP2006522125A patent/JP2007510621A/ja active Pending
- 2004-07-29 NZ NZ601772A patent/NZ601772A/xx not_active IP Right Cessation
- 2004-07-29 AU AU2004289174A patent/AU2004289174B2/en not_active Ceased
- 2004-07-29 KR KR1020067002214A patent/KR20060073584A/ko active Search and Examination
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2006
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SG178721A1 (en) | 2012-03-29 |
AU2004289174A2 (en) | 2005-05-26 |
NZ601780A (en) | 2012-10-26 |
WO2005046575A3 (en) | 2007-10-04 |
CA2534342C (en) | 2016-05-10 |
KR20130081319A (ko) | 2013-07-16 |
JP2013035863A (ja) | 2013-02-21 |
NZ545570A (en) | 2012-07-27 |
KR20120116991A (ko) | 2012-10-23 |
CN101123878A (zh) | 2008-02-13 |
JP2007510621A (ja) | 2007-04-26 |
NZ601772A (en) | 2012-10-26 |
EP1660017A4 (de) | 2011-03-09 |
EP1660017A2 (de) | 2006-05-31 |
ZA200600660B (en) | 2007-04-25 |
AU2004289174B2 (en) | 2011-05-19 |
KR20060073584A (ko) | 2006-06-28 |
SG145693A1 (en) | 2008-09-29 |
CA2534342A1 (en) | 2005-05-26 |
WO2005046575A2 (en) | 2005-05-26 |
AU2004289174A1 (en) | 2005-05-26 |
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