IL163803A0 - Heterocyclic amide derivatives as inhibitors of glycogen phosphorylase - Google Patents

Heterocyclic amide derivatives as inhibitors of glycogen phosphorylase

Info

Publication number
IL163803A0
IL163803A0 IL16380303A IL16380303A IL163803A0 IL 163803 A0 IL163803 A0 IL 163803A0 IL 16380303 A IL16380303 A IL 16380303A IL 16380303 A IL16380303 A IL 16380303A IL 163803 A0 IL163803 A0 IL 163803A0
Authority
IL
Israel
Prior art keywords
inhibitors
amide derivatives
glycogen phosphorylase
heterocyclic amide
heterocyclic
Prior art date
Application number
IL16380303A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IL163803A0 publication Critical patent/IL163803A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Indole Compounds (AREA)
IL16380303A 2002-03-06 2003-03-04 Heterocyclic amide derivatives as inhibitors of glycogen phosphorylase IL163803A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0205165.4A GB0205165D0 (en) 2002-03-06 2002-03-06 Chemical compounds
PCT/GB2003/000877 WO2003074532A1 (en) 2002-03-06 2003-03-04 Heterocyclic amide derivatives as inhibitors of glycogen phosphorylase

Publications (1)

Publication Number Publication Date
IL163803A0 true IL163803A0 (en) 2005-12-18

Family

ID=9932329

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16380303A IL163803A0 (en) 2002-03-06 2003-03-04 Heterocyclic amide derivatives as inhibitors of glycogen phosphorylase

Country Status (18)

Country Link
US (2) US7129249B2 (enExample)
EP (1) EP1483270A1 (enExample)
JP (1) JP2005526058A (enExample)
KR (1) KR20040096661A (enExample)
CN (1) CN100384852C (enExample)
AR (1) AR038888A1 (enExample)
AU (1) AU2003214377A1 (enExample)
BR (1) BR0308146A (enExample)
CA (1) CA2477667A1 (enExample)
GB (1) GB0205165D0 (enExample)
IL (1) IL163803A0 (enExample)
MX (1) MXPA04008614A (enExample)
NO (1) NO20043852L (enExample)
NZ (1) NZ534990A (enExample)
PL (1) PL372973A1 (enExample)
TW (1) TW200305412A (enExample)
WO (1) WO2003074532A1 (enExample)
ZA (1) ZA200406679B (enExample)

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GB0205166D0 (en) 2002-03-06 2002-04-17 Astrazeneca Ab Chemical compounds
GB0205176D0 (en) 2002-03-06 2002-04-17 Astrazeneca Ab Chemical compounds
GB0205175D0 (en) 2002-03-06 2002-04-17 Astrazeneca Ab Chemical compounds
CA2495943C (en) * 2002-08-29 2009-07-21 Merck & Co., Inc. Indoles having anti-diabetic activity
GB0222912D0 (en) 2002-10-03 2002-11-13 Astrazeneca Ab Novel process and intermediates
GB0222909D0 (en) 2002-10-03 2002-11-13 Astrazeneca Ab Novel process and intermediates
GB0320422D0 (en) * 2003-08-30 2003-10-01 Astrazeneca Ab Chemical compounds
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US7402674B2 (en) 2004-01-31 2008-07-22 Sanofi-Aventis Deutschland Gmbh, 7-Phenylamino-4-quinolone-3-carboxylic acid derivatives, process for their preparation and their use as medicaments
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JP6274723B2 (ja) 2009-10-16 2018-02-07 メリンタ セラピューティクス，インコーポレイテッド 抗微生物性化合物および抗微生物性化合物の製造方法および使用方法
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Also Published As

Publication number Publication date
US20050131015A1 (en) 2005-06-16
ZA200406679B (en) 2005-01-18
US7129249B2 (en) 2006-10-31
CN1653070A (zh) 2005-08-10
MXPA04008614A (es) 2004-12-06
US7276517B2 (en) 2007-10-02
GB0205165D0 (en) 2002-04-17
AR038888A1 (es) 2005-02-02
CN100384852C (zh) 2008-04-30
EP1483270A1 (en) 2004-12-08
KR20040096661A (ko) 2004-11-16
PL372973A1 (en) 2005-08-08
TW200305412A (en) 2003-11-01
US20070043069A1 (en) 2007-02-22
AU2003214377A1 (en) 2003-09-16
BR0308146A (pt) 2004-12-07
CA2477667A1 (en) 2003-09-12
NZ534990A (en) 2006-02-24
JP2005526058A (ja) 2005-09-02
WO2003074532A1 (en) 2003-09-12
NO20043852L (no) 2004-09-14

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