IL155992A0 - Pharmaceutical compositions for the oral delivery of pharmacologically active agents - Google Patents

Pharmaceutical compositions for the oral delivery of pharmacologically active agents

Info

Publication number
IL155992A0
IL155992A0 IL15599201A IL15599201A IL155992A0 IL 155992 A0 IL155992 A0 IL 155992A0 IL 15599201 A IL15599201 A IL 15599201A IL 15599201 A IL15599201 A IL 15599201A IL 155992 A0 IL155992 A0 IL 155992A0
Authority
IL
Israel
Prior art keywords
pharmacologically active
active agents
pharmaceutical compositions
oral delivery
delivery
Prior art date
Application number
IL15599201A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of IL155992A0 publication Critical patent/IL155992A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/18Drugs for disorders of the endocrine system of the parathyroid hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Rheumatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL15599201A 2000-12-06 2001-12-05 Pharmaceutical compositions for the oral delivery of pharmacologically active agents IL155992A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25172900P 2000-12-06 2000-12-06
PCT/EP2001/014294 WO2002045754A2 (en) 2000-12-06 2001-12-05 Pharmaceutical compositions for the oral delivery of pharmacologically active agents

Publications (1)

Publication Number Publication Date
IL155992A0 true IL155992A0 (en) 2003-12-23

Family

ID=22953160

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15599201A IL155992A0 (en) 2000-12-06 2001-12-05 Pharmaceutical compositions for the oral delivery of pharmacologically active agents
IL155992A IL155992A (en) 2000-12-06 2003-05-19 Pharmacological preparations of pharmacologically active substances for oral administration

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL155992A IL155992A (en) 2000-12-06 2003-05-19 Pharmacological preparations of pharmacologically active substances for oral administration

Country Status (26)

Country Link
US (1) US7049283B2 (de)
EP (1) EP1341526B1 (de)
JP (2) JP4898078B2 (de)
KR (1) KR100847695B1 (de)
CN (1) CN1304048C (de)
AT (1) ATE513541T1 (de)
AU (2) AU3454702A (de)
BR (2) BR0115965A (de)
CA (1) CA2436599C (de)
CY (1) CY1112562T1 (de)
CZ (1) CZ305418B6 (de)
DK (1) DK1341526T3 (de)
EC (1) ECSP034639A (de)
ES (1) ES2367009T3 (de)
HU (1) HU230632B1 (de)
IL (2) IL155992A0 (de)
MX (1) MXPA03005096A (de)
NO (1) NO332936B1 (de)
NZ (1) NZ526196A (de)
PL (1) PL209703B1 (de)
PT (1) PT1341526E (de)
RU (1) RU2287999C2 (de)
SI (1) SI1341526T1 (de)
SK (1) SK287613B6 (de)
WO (1) WO2002045754A2 (de)
ZA (1) ZA200304295B (de)

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US20050054557A1 (en) * 2002-05-09 2005-03-10 Goldberg Michael M. Compositions for delivering parathyroid hormone and calcitonin
TW200403052A (en) * 2002-07-17 2004-03-01 Novartis Ag Use of organic compounds
PE20040724A1 (es) * 2002-08-01 2004-12-06 Novartis Ag Composicion para la administracion oral de calcitonina
JP5546715B2 (ja) * 2003-03-17 2014-07-09 日本たばこ産業株式会社 Cetp阻害剤の医薬組成物
TWI494102B (zh) * 2003-05-02 2015-08-01 Japan Tobacco Inc 包含s-〔2(〔〔1-(2-乙基丁基)環己基〕羰基〕胺基)苯基〕2-甲基丙烷硫酯及hmg輔酶a還原酶抑制劑之組合
PT1651248E (pt) * 2003-07-11 2009-11-10 Novartis Ag Composições farmacêuticas para dose oral compreendendo um agente de administração na forma micronizada
MXPA06000807A (es) * 2003-07-23 2006-08-23 Novartis Ag Uso de calcitonina en osteoartritis.
PT1663182E (pt) * 2003-09-12 2013-03-14 Amgen Inc Formulação de dissolução rápida de cinacalcet hcl
MXPA06013384A (es) * 2004-05-19 2007-03-01 Emisphere Tech Inc Formulaciones topicas de cromolin.
GB0422644D0 (en) * 2004-10-12 2004-11-10 Novartis Ag Organic compounds
GB0427603D0 (en) 2004-12-16 2005-01-19 Novartis Ag Organic compounds
EP1843755B1 (de) * 2005-02-01 2015-04-01 Emisphere Technologies, Inc. System zur magenretention und zur gesteuerten freisetzung
US8030271B2 (en) * 2005-07-05 2011-10-04 Emisphere Technologies, Inc. Compositions and methods for buccal delivery of human growth hormone
KR20080049128A (ko) 2005-09-19 2008-06-03 에미스페어 테크놀로지스, 인코포레이티드 N-(5-클로로살리실로일)-8-아미노카프릴산 이나트륨염의결정형
GB0522566D0 (en) * 2005-11-04 2005-12-14 Novartis Ag Organic compounds
BRPI0618723A2 (pt) * 2005-11-17 2011-09-06 Novartis Ag composição farmacêutica oral na forma de um comprimido prensado
JP2009527504A (ja) * 2006-02-23 2009-07-30 イオメディックス スリープ インターナショナル エスアールエル 良質な睡眠の誘導および維持のための組成物および方法
WO2008021088A2 (en) * 2006-08-08 2008-02-21 The Regents Of The University Of Californina Salicylanilides enhance oral delivery of therapeutic peptides
US8323688B2 (en) * 2006-08-31 2012-12-04 Novartis Ag Pharmaceutical compositions comprising hGH for oral delivery
CA2572004A1 (en) * 2006-12-08 2008-06-08 Bernard Charles Sherman Tablets comprising entacapone and crospovidone
ATE507818T1 (de) * 2007-03-02 2011-05-15 Novartis Ag Orale verabreichung eines calcitonins
PL2215047T3 (pl) 2007-11-02 2014-05-30 Emisphere Tech Inc Sposób leczenia niedoborów witaminy b12
CA2734442C (en) 2008-08-18 2016-08-16 Oramed Ltd Methods and compositions for oral administration of proteins
KR101673042B1 (ko) * 2009-03-12 2016-11-04 키바이오사이언스 아게 당뇨병 및 대사 증후군의 치료
EA026713B1 (ru) * 2010-06-09 2017-05-31 Эмисфире Текнолоджис, Инк. Твердая пероральная лекарственная форма для лечения дефицита железа или анемии и ее применение
PL3326620T3 (pl) 2010-12-16 2020-08-24 Novo Nordisk A/S Kompozycje stałe zawierające agonistę glp-1 i sól kwasu n-(8-(2- hydroksybenzoilo)amino)kaprylowego
BR112013026195A2 (pt) 2011-04-12 2016-11-29 Novo Nordisk As derivados de glp-1 duplamente acilados
CN111494323B (zh) 2012-03-22 2023-03-28 诺和诺德股份有限公司 包含递送剂的组合物及其制备
DK2827845T3 (en) 2012-03-22 2019-04-01 Novo Nordisk As COMPOSITIONS INCLUDING A PROCEDURE AND PREPARING THEREOF
HUE062740T2 (hu) 2012-03-22 2023-12-28 Novo Nordisk As GLP-1 peptidek készítményei és elõállításuk
US9993430B2 (en) 2012-06-20 2018-06-12 Novo Nordisk A/S Tablet formulation comprising semaglutide and a delivery agent
PT2991671T (pt) 2013-05-02 2018-11-05 Novo Nordisk As Dosagem oral de compostos de glp-1
CN104961687B (zh) * 2015-06-03 2017-07-25 苏州维泰生物技术有限公司 1,2‑二嗪衍生物及其制剂、用途
MY189670A (en) * 2015-07-08 2022-02-24 Research & Business Found Sungkyunkwan Univ Pyrrolidine carboxamido derivatives and methods for preparing and using the same
EA036204B1 (ru) * 2015-10-16 2020-10-14 Нобел Илач Санайи Ве Тиджарет А.Ш. Фармацевтические композиции нилотиниба гидрохлорида
CN107080739A (zh) * 2017-04-17 2017-08-22 深圳市泛谷药业股份有限公司 一种用于口服给药的固体快速释放布南色林片及其制备方法
SG11202006595RA (en) 2018-02-02 2020-08-28 Novo Nordisk As Solid compositions comprising a glp-1 agonist, a salt of n-(8-(2-hydroxybenzoyl)amino)caprylic acid and a lubricant
JP2021054781A (ja) * 2019-09-26 2021-04-08 デボン エルエス,リミテッド 共結晶形エフィナコナゾール、及びその製造方法
KR102301743B1 (ko) * 2020-12-29 2021-09-13 대봉엘에스 주식회사 에피나코나졸 경구용 조성물

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Also Published As

Publication number Publication date
NZ526196A (en) 2005-01-28
SK287613B6 (sk) 2011-04-05
AU2002234547B2 (en) 2005-03-24
CZ305418B6 (cs) 2015-09-09
DK1341526T3 (da) 2011-10-03
PT1341526E (pt) 2011-09-01
ATE513541T1 (de) 2011-07-15
MXPA03005096A (es) 2003-09-05
IL155992A (en) 2008-04-13
ECSP034639A (es) 2003-07-25
HUP0302319A2 (hu) 2003-11-28
CA2436599A1 (en) 2002-06-13
WO2002045754A3 (en) 2003-01-03
CN1479612A (zh) 2004-03-03
BR0115965A (pt) 2003-10-28
AU3454702A (en) 2002-06-18
CZ20031566A3 (cs) 2003-09-17
JP2009185052A (ja) 2009-08-20
NO20032511L (no) 2003-06-03
JP2004515480A (ja) 2004-05-27
HUP0302319A3 (en) 2013-04-29
WO2002045754A2 (en) 2002-06-13
EP1341526A2 (de) 2003-09-10
US7049283B2 (en) 2006-05-23
NO20032511D0 (no) 2003-06-03
BRPI0115965B1 (pt) 2017-09-26
RU2287999C2 (ru) 2006-11-27
CN1304048C (zh) 2007-03-14
SK6882003A3 (en) 2004-01-08
SI1341526T1 (sl) 2011-10-28
ZA200304295B (en) 2004-05-10
EP1341526B1 (de) 2011-06-22
CY1112562T1 (el) 2016-02-10
NO332936B1 (no) 2013-02-04
PL362247A1 (en) 2004-10-18
HU230632B1 (hu) 2017-05-29
PL209703B1 (pl) 2011-10-31
ES2367009T3 (es) 2011-10-27
CA2436599C (en) 2011-01-25
HK1059565A1 (en) 2004-07-09
JP4898078B2 (ja) 2012-03-14
KR100847695B1 (ko) 2008-07-23
KR20040018309A (ko) 2004-03-03
US20020123459A1 (en) 2002-09-05

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