IL150742A0 - Pyridopyrimidinone derivatives for the treatment of neurodegenerative disease - Google Patents

Pyridopyrimidinone derivatives for the treatment of neurodegenerative disease

Info

Publication number
IL150742A0
IL150742A0 IL15074200A IL15074200A IL150742A0 IL 150742 A0 IL150742 A0 IL 150742A0 IL 15074200 A IL15074200 A IL 15074200A IL 15074200 A IL15074200 A IL 15074200A IL 150742 A0 IL150742 A0 IL 150742A0
Authority
IL
Israel
Prior art keywords
treatment
neurodegenerative disease
pyridopyrimidinone derivatives
pyridopyrimidinone
derivatives
Prior art date
Application number
IL15074200A
Other languages
English (en)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of IL150742A0 publication Critical patent/IL150742A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL15074200A 2000-01-27 2000-11-30 Pyridopyrimidinone derivatives for the treatment of neurodegenerative disease IL150742A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17840000P 2000-01-27 2000-01-27
PCT/US2000/032572 WO2001055148A1 (en) 2000-01-27 2000-11-30 Pyridopyrimidinone derivatives for treatment of neurodegenerative disease

Publications (1)

Publication Number Publication Date
IL150742A0 true IL150742A0 (en) 2003-02-12

Family

ID=22652409

Family Applications (1)

Application Number Title Priority Date Filing Date
IL15074200A IL150742A0 (en) 2000-01-27 2000-11-30 Pyridopyrimidinone derivatives for the treatment of neurodegenerative disease

Country Status (22)

Country Link
US (1) US20040224958A1 (hu)
EP (1) EP1255755A1 (hu)
JP (1) JP2003523358A (hu)
KR (1) KR20020070520A (hu)
CN (1) CN1433417A (hu)
AR (1) AR029437A1 (hu)
AU (1) AU1808601A (hu)
BR (1) BR0017075A (hu)
CA (1) CA2394525A1 (hu)
CO (1) CO5280216A1 (hu)
CZ (1) CZ20022521A3 (hu)
GT (1) GT200100005A (hu)
HN (1) HN2001000012A (hu)
HU (1) HUP0203803A3 (hu)
IL (1) IL150742A0 (hu)
PA (1) PA8510801A1 (hu)
PE (1) PE20011228A1 (hu)
PL (1) PL357634A1 (hu)
SK (1) SK10772002A3 (hu)
SV (1) SV2002000287A (hu)
TN (1) TNSN01018A1 (hu)
WO (1) WO2001055148A1 (hu)

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US7235551B2 (en) * 2000-03-02 2007-06-26 Smithkline Beecham Corporation 1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
EP1333833B1 (en) * 2000-10-23 2011-08-24 GlaxoSmithKline LLC Novel trisubstituted-8H-pyrido[2,3-d]pyrimidin-7-one compound for the treatment of CSBP/p38 kinase mediated diseases
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US7105667B2 (en) 2001-05-01 2006-09-12 Bristol-Myers Squibb Co. Fused heterocyclic compounds and use thereof
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EP1397142A4 (en) 2001-06-19 2004-11-03 Bristol Myers Squibb Co PYRIMIDINE PHOSPHODIESTERASE (PDE) INHIBITORS 7
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GEP20063909B (en) 2002-01-22 2006-08-25 Warner Lambert Co 2-(PYRIDIN-2-YLAMINO)-PYRIDO[2,3d] PYRIMIDIN-7-ONES
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EP1786817A1 (de) * 2004-08-26 2007-05-23 Boehringer Ingelheim International GmbH Pteridinone als plk (polo like kinase) inhibitoren
JP5111113B2 (ja) 2004-12-13 2012-12-26 サネシス ファーマシューティカルズ， インコーポレイテッド Ｒａｆキナーゼ阻害剤として有用なピリドピリミジノン、ジヒドロピリミドピリミジノンおよびプテリジノン
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Also Published As

Publication number Publication date
US20040224958A1 (en) 2004-11-11
CA2394525A1 (en) 2001-08-02
CN1433417A (zh) 2003-07-30
AU1808601A (en) 2001-08-07
PL357634A1 (en) 2004-07-26
AR029437A1 (es) 2003-06-25
JP2003523358A (ja) 2003-08-05
KR20020070520A (ko) 2002-09-09
WO2001055148A1 (en) 2001-08-02
HN2001000012A (es) 2001-07-09
CZ20022521A3 (cs) 2003-02-12
CO5280216A1 (es) 2003-05-30
SV2002000287A (es) 2002-01-08
SK10772002A3 (sk) 2004-01-08
GT200100005A (es) 2002-02-05
BR0017075A (pt) 2002-11-05
HUP0203803A3 (en) 2004-09-28
PE20011228A1 (es) 2002-01-18
EP1255755A1 (en) 2002-11-13
TNSN01018A1 (en) 2005-11-10
HUP0203803A2 (hu) 2003-02-28
PA8510801A1 (es) 2002-12-11

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