IL150313A0 - Pyrrolidine derivatives as cyclic amp -specific phosphodiesterase inhibitors - Google Patents

Pyrrolidine derivatives as cyclic amp -specific phosphodiesterase inhibitors

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Publication number
IL150313A0
IL150313A0 IL15031300A IL15031300A IL150313A0 IL 150313 A0 IL150313 A0 IL 150313A0 IL 15031300 A IL15031300 A IL 15031300A IL 15031300 A IL15031300 A IL 15031300A IL 150313 A0 IL150313 A0 IL 150313A0
Authority
IL
Israel
Prior art keywords
cyclic amp
phosphodiesterase inhibitors
pyrrolidine derivatives
specific phosphodiesterase
disclosed
Prior art date
Application number
IL15031300A
Other languages
English (en)
Original Assignee
Icos Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Icos Corp filed Critical Icos Corp
Publication of IL150313A0 publication Critical patent/IL150313A0/xx

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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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IL15031300A 1999-12-23 2000-11-28 Pyrrolidine derivatives as cyclic amp -specific phosphodiesterase inhibitors IL150313A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/471,846 US6258833B1 (en) 1999-12-23 1999-12-23 Cyclic AMP-specific phosphodiesterase inhibitors
PCT/US2000/032401 WO2001047905A1 (en) 1999-12-23 2000-11-28 Pyrrolidine derivatives as cyclic amp-specific phosphodiesterase inhibitors

Publications (1)

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IL150313A0 true IL150313A0 (en) 2002-12-01

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IL15031300A IL150313A0 (en) 1999-12-23 2000-11-28 Pyrrolidine derivatives as cyclic amp -specific phosphodiesterase inhibitors

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US (6) US6258833B1 (is)
EP (1) EP1242400B1 (is)
JP (1) JP4294903B2 (is)
KR (1) KR20020063600A (is)
CN (1) CN1434813A (is)
AT (1) ATE325108T1 (is)
AU (1) AU778543B2 (is)
BG (1) BG65892B1 (is)
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HK (1) HK1051359A1 (is)
HR (1) HRP20020541B1 (is)
HU (1) HUP0301113A3 (is)
IL (1) IL150313A0 (is)
IS (1) IS6436A (is)
MX (1) MXPA02006212A (is)
NO (1) NO20023008L (is)
PL (1) PL202227B1 (is)
RS (1) RS50841B (is)
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TR (1) TR200400702T4 (is)
UA (1) UA73964C2 (is)
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Families Citing this family (53)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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