IL140093A0 - Glycopeptide derivatives and pharmaceutical compositions containing the same - Google Patents

Glycopeptide derivatives and pharmaceutical compositions containing the same

Info

Publication number
IL140093A0
IL140093A0 IL14009399A IL14009399A IL140093A0 IL 140093 A0 IL140093 A0 IL 140093A0 IL 14009399 A IL14009399 A IL 14009399A IL 14009399 A IL14009399 A IL 14009399A IL 140093 A0 IL140093 A0 IL 140093A0
Authority
IL
Israel
Prior art keywords
pharmaceutical compositions
compositions containing
same
derivatives
glycopeptide derivatives
Prior art date
Application number
IL14009399A
Other languages
English (en)
Original Assignee
Advanced Medicine Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Advanced Medicine Inc filed Critical Advanced Medicine Inc
Publication of IL140093A0 publication Critical patent/IL140093A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL14009399A 1998-12-23 1999-12-22 Glycopeptide derivatives and pharmaceutical compositions containing the same IL140093A0 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US11372898P 1998-12-23 1998-12-23
US12931399P 1999-04-14 1999-04-14
US16402499P 1999-11-04 1999-11-04
US16997899P 1999-12-10 1999-12-10
PCT/US1999/030543 WO2000039156A1 (en) 1998-12-23 1999-12-22 Glycopeptide derivatives and pharmaceutical compositions containing the same

Publications (1)

Publication Number Publication Date
IL140093A0 true IL140093A0 (en) 2002-02-10

Family

ID=27493926

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14009399A IL140093A0 (en) 1998-12-23 1999-12-22 Glycopeptide derivatives and pharmaceutical compositions containing the same
IL140093A IL140093A (en) 1998-12-23 2000-12-05 History of glycopropeptide and pharmaceutical preparations containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL140093A IL140093A (en) 1998-12-23 2000-12-05 History of glycopropeptide and pharmaceutical preparations containing them

Country Status (23)

Country Link
US (9) US6392012B1 (ja)
EP (1) EP1140993B1 (ja)
JP (1) JP4362017B2 (ja)
KR (1) KR100665204B1 (ja)
CN (1) CN1249081C (ja)
AT (1) ATE242783T1 (ja)
AU (1) AU768204B2 (ja)
BR (1) BRPI9914221B8 (ja)
CA (1) CA2336445C (ja)
CZ (1) CZ301184B6 (ja)
DE (1) DE69908819T2 (ja)
DK (1) DK1140993T3 (ja)
ES (1) ES2201825T3 (ja)
HK (1) HK1040721B (ja)
HU (1) HU230190B1 (ja)
IL (2) IL140093A0 (ja)
NO (1) NO326066B1 (ja)
NZ (1) NZ508594A (ja)
PL (1) PL198311B1 (ja)
PT (1) PT1140993E (ja)
SI (1) SI1140993T1 (ja)
WO (1) WO2000039156A1 (ja)
ZA (1) ZA200007222B (ja)

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US6699836B2 (en) 1999-04-02 2004-03-02 The Trustees Of Princeton University Vancomycin analogs
AU4054900A (en) * 1999-04-02 2000-10-23 Advanced Medicine East, Inc. Desleucyl glycopeptide antibiotics and methods of making same
WO2001057071A2 (en) * 2000-02-04 2001-08-09 Advanced Medicine, Inc. Glycopeptide derivatives having antibiotic activity
EP1276759B1 (en) 2000-05-02 2008-07-30 Theravance, Inc. Reductive alkylation process on glycopeptides
WO2001083520A2 (en) * 2000-05-02 2001-11-08 Theravance,Inc Polyacid glycopeptide derivatives
BR0110530A (pt) 2000-05-02 2003-04-08 Theravance Inc Composições farmacêuticas contendo um antibiótico glicopeptìdico e uma ciclodextrina
UA75083C2 (uk) * 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
ES2302733T3 (es) * 2000-06-22 2008-08-01 Theravance, Inc. Derivados carboxi-sacaridos de glucopeptido.
AU2001259816A1 (en) 2000-06-22 2002-01-02 Advanced Medecine, Inc. Polyhydroxy glycopeptide derivatives
US6872804B2 (en) 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
US6905669B2 (en) * 2001-04-24 2005-06-14 Supergen, Inc. Compositions and methods for reestablishing gene transcription through inhibition of DNA methylation and histone deacetylase
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
EP1295711B1 (en) 2001-09-19 2006-04-12 The Procter & Gamble Company A color printed laminated structure, absorbent article comprising the same and process for manufacturing the same
TWI335332B (en) 2001-10-12 2011-01-01 Theravance Inc Cross-linked vancomycin-cephalosporin antibiotics
US7652039B2 (en) 2002-05-17 2010-01-26 Sequella, Inc. Methods of use and compositions for the diagnosis and treatment of infectious disease
US20040033986A1 (en) 2002-05-17 2004-02-19 Protopopova Marina Nikolaevna Anti tubercular drug: compositions and methods
EP1507796B1 (en) 2002-05-24 2012-05-02 Theravance, Inc. Cross-linked glycopeptide-cephalosporin antibiotics
US6951963B2 (en) 2002-06-17 2005-10-04 Theravance, Inc. Process for preparing N-protected β-amino aldehyde compounds
CA2491573A1 (en) * 2002-07-09 2004-01-15 Fasgen, Llc Methods of treating microbial infections in humans and animals
US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
AU2003294262B2 (en) * 2002-11-18 2007-08-23 Vicuron Pharmaceuticals Inc. Methods of administering dalbavancin for treatment of bacterial infections
ES2335013T3 (es) 2003-05-23 2010-03-18 Theravance, Inc. Antibioticos de glucopeptido-cefalosporina reticulados.
ATE388153T1 (de) * 2003-07-11 2008-03-15 Theravance Inc Quervernetzte glycopeptid-cephalosporin- antibiotika
DE102004055582A1 (de) * 2004-11-18 2006-05-24 Bayer Cropscience Ag N-Heterocyclyl-phthalsäurediamide
WO2006057303A1 (ja) 2004-11-29 2006-06-01 National University Corporation Nagoya University グリコペプチド抗生物質モノマー誘導体
US8304597B2 (en) 2004-12-15 2012-11-06 The Procter And Gamble Company Method of using an absorbent article having a functional enhancement indicator
US20070185015A1 (en) * 2005-02-28 2007-08-09 Chiron Corporation and North China Pharmaceutical Corporation Semi-synthetic desmethyl-vancomycin-based glycopeptides with antibiotic activity
US7632918B2 (en) * 2005-02-28 2009-12-15 Novartis Vaccines And Diagnostics, Inc. Semi-synthetic glycopeptides with antibiotic activity
US7368422B2 (en) * 2005-02-28 2008-05-06 Novartis Vaccines And Diagnostics Inc. Semi-synthetic rearranged vancomycin/desmethyl-vancomycin-based glycopeptides with antibiotic activity
WO2007038246A2 (en) 2005-09-22 2007-04-05 Medivas, Llc Solid polymer delivery compositions and methods for use thereof
EP1926780B1 (en) 2005-09-22 2013-08-14 Medivas, LLC Bis-( -amino)-diol-diester-containing poly(ester amide) and poly(ester urethane) compositions and methods of use
WO2007084507A2 (en) * 2006-01-13 2007-07-26 The Scripps Research Institute [ψ[CH2NH]PG4] GLYCOPEPTIDE ANTIBIOTIC ANALOGS
TW200808818A (en) * 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
WO2009081958A1 (ja) 2007-12-26 2009-07-02 Shionogi & Co., Ltd. グリコペプチド抗生物質配糖化誘導体
KR20100109936A (ko) * 2007-12-26 2010-10-11 리드 테라퓨틱스, 인크. 항박테리아제로서의 신규한 반(半)-합성 글리코펩티드
US8841440B2 (en) 2008-04-01 2014-09-23 Cornell University Organo-soluble chitosan salts and chitosan-derived biomaterials prepared thereof
GB2465863A (en) * 2008-12-05 2010-06-09 Lead Therapeutics Inc Semi-synthetic heptapeptidic glycopeptides for the treatment of bacterial infections
CN101928330B (zh) * 2009-06-26 2013-10-16 上海来益生物药物研究开发中心有限责任公司 一种新的化合物及其应用
EP2688580A4 (en) * 2011-03-24 2015-03-25 Seachaid Pharmaceuticals Inc DERIVATIVES OF VANCOMYCIN
AU2014322817A1 (en) * 2013-09-23 2016-04-21 Jawaharlal Nehru Centre for Advanced Scientific Research (JNCASR) Vancomycin-sugar conjugates and uses thereof
EP3240574A1 (en) * 2014-12-25 2017-11-08 Jawaharlal Nehru Centre For Advanced Scientific Research Glycopeptides and uses thereof
CN109072271A (zh) * 2016-01-15 2018-12-21 汉堡大学 用于制备鼠李糖基化类黄酮的方法
US10689407B2 (en) * 2016-01-28 2020-06-23 Envista Photo-cleavable primer compositions and methods of use
CN107325159A (zh) * 2016-04-29 2017-11-07 中国科学院上海药物研究所 一类万古霉素衍生物、其制备方法、药物组合物和用途
CA3062570A1 (en) * 2017-05-22 2018-11-29 Insmed Incorporated Lipo-glycopeptide cleavable derivatives and uses thereof
CN107987131B (zh) * 2017-11-16 2021-03-09 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的化合物、其制备方法和应用
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用
NL2023883B1 (en) * 2019-09-24 2021-04-26 Univ Leiden Antibiotic compounds
CN111620931B (zh) * 2020-06-12 2021-12-17 苏州博源医疗科技有限公司 万古霉素衍生物及其制备方法和应用
CN114213284B (zh) * 2022-01-04 2023-08-01 丽珠集团福州福兴医药有限公司 (9h-芴-9-基)-癸基(2-氧代乙基)氨基甲酸甲酯及其合成方法

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Also Published As

Publication number Publication date
CZ301184B6 (cs) 2009-12-02
US20030060598A1 (en) 2003-03-27
US6444786B1 (en) 2002-09-03
HK1040721B (zh) 2003-10-17
EP1140993B1 (en) 2003-06-11
HUP0400887A3 (en) 2012-09-28
CN1249081C (zh) 2006-04-05
BRPI9914221B8 (pt) 2021-05-25
IL140093A (en) 2006-06-11
CA2336445C (en) 2011-07-19
KR20010085857A (ko) 2001-09-07
DE69908819T2 (de) 2004-05-06
US6392012B1 (en) 2002-05-21
ES2201825T3 (es) 2004-03-16
NO20006323L (no) 2001-02-12
US20080103292A1 (en) 2008-05-01
KR100665204B1 (ko) 2007-01-04
CN1315961A (zh) 2001-10-03
US20060241024A1 (en) 2006-10-26
AU768204B2 (en) 2003-12-04
EP1140993A1 (en) 2001-10-10
NO20006323D0 (no) 2000-12-12
CZ200122A3 (en) 2001-06-13
JP2002533472A (ja) 2002-10-08
WO2000039156A1 (en) 2000-07-06
BR9914221B1 (pt) 2013-12-31
PT1140993E (pt) 2003-10-31
NO326066B1 (no) 2008-09-08
US7351791B2 (en) 2008-04-01
PL348451A1 (en) 2002-05-20
DE69908819D1 (de) 2003-07-17
HUP0400887A2 (hu) 2004-08-30
PL198311B1 (pl) 2008-06-30
US6455669B1 (en) 2002-09-24
US6949681B2 (en) 2005-09-27
NZ508594A (en) 2003-05-30
US20090215982A1 (en) 2009-08-27
AU3127300A (en) 2000-07-31
SI1140993T1 (en) 2003-12-31
US7101964B2 (en) 2006-09-05
ZA200007222B (en) 2002-03-06
US8030445B2 (en) 2011-10-04
ATE242783T1 (de) 2003-06-15
HU230190B1 (hu) 2015-09-28
US7723470B2 (en) 2010-05-25
BR9914221A (pt) 2001-06-26
US20040204346A1 (en) 2004-10-14
HK1040721A1 (en) 2002-06-21
DK1140993T3 (da) 2003-10-06
US6962970B2 (en) 2005-11-08
US20050239690A1 (en) 2005-10-27
JP4362017B2 (ja) 2009-11-11
CA2336445A1 (en) 2000-07-06

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