IL111002A - History of piperidine, their preparation and the pharmaceutical preparations containing them - Google Patents

History of piperidine, their preparation and the pharmaceutical preparations containing them

Info

Publication number
IL111002A
IL111002A IL11100294A IL11100294A IL111002A IL 111002 A IL111002 A IL 111002A IL 11100294 A IL11100294 A IL 11100294A IL 11100294 A IL11100294 A IL 11100294A IL 111002 A IL111002 A IL 111002A
Authority
IL
Israel
Prior art keywords
tetrazol
methoxy
phenyl
piperidin
title compound
Prior art date
Application number
IL11100294A
Other languages
English (en)
Hebrew (he)
Other versions
IL111002A0 (en
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939319606A external-priority patent/GB9319606D0/en
Priority claimed from GB9326583A external-priority patent/GB9326583D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of IL111002A0 publication Critical patent/IL111002A0/xx
Publication of IL111002A publication Critical patent/IL111002A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
IL11100294A 1993-09-22 1994-09-19 History of piperidine, their preparation and the pharmaceutical preparations containing them IL111002A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939319606A GB9319606D0 (en) 1993-09-22 1993-09-22 Chemical compounds
GB9326583A GB9326583D0 (en) 1993-12-31 1993-12-31 Chemical compounds

Publications (2)

Publication Number Publication Date
IL111002A0 IL111002A0 (en) 1994-11-28
IL111002A true IL111002A (en) 1998-09-24

Family

ID=26303560

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11100294A IL111002A (en) 1993-09-22 1994-09-19 History of piperidine, their preparation and the pharmaceutical preparations containing them

Country Status (30)

Country Link
US (2) US5703240A (da)
EP (1) EP0720609B1 (da)
JP (2) JP2865872B2 (da)
CN (1) CN1061041C (da)
AP (1) AP495A (da)
AT (1) ATE173255T1 (da)
AU (1) AU681190B2 (da)
BG (1) BG62169B1 (da)
CA (1) CA2172529A1 (da)
CO (1) CO4290298A1 (da)
CZ (1) CZ285479B6 (da)
DE (1) DE69414590T2 (da)
DK (1) DK0720609T3 (da)
ES (1) ES2123829T3 (da)
FI (1) FI961270A (da)
GR (1) GR3029354T3 (da)
HK (1) HK1004219A1 (da)
HR (1) HRP940575B1 (da)
HU (1) HU217428B (da)
IL (1) IL111002A (da)
IS (1) IS4208A (da)
NO (1) NO307830B1 (da)
NZ (1) NZ273614A (da)
OA (1) OA10576A (da)
PE (1) PE18295A1 (da)
PL (1) PL179585B1 (da)
SI (1) SI0720609T1 (da)
SK (1) SK280901B6 (da)
UA (1) UA44711C2 (da)
WO (1) WO1995008549A1 (da)

Families Citing this family (98)

* Cited by examiner, † Cited by third party
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US5922737A (en) * 1996-02-21 1999-07-13 Hoechst Marion Roussel, Inc. Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases
US5998439A (en) 1996-02-21 1999-12-07 Hoescht Marion Roussel, Inc. Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
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Family Cites Families (6)

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Publication number Priority date Publication date Assignee Title
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UA41251C2 (uk) * 1990-01-04 2001-09-17 Пфайзер, Інк. Гідровані азотвмісні гетероциклічні сполуки, похідні піперидину, фармацевтична композиція та спосіб пригнічення активності речовини р в організмі
US5332817A (en) * 1990-01-04 1994-07-26 Pfizer Inc. 3-aminopiperidine derivatives and related nitrogen containing heterocycles
UA39168C2 (uk) * 1991-06-20 2001-06-15 Пфайзер, Інк. Фторалкоксифенільні похідні піперидину або хінуклідину, що є антагоністами речовини p і фармацевтична композиція на їх основі
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IS4208A (is) * 1993-09-22 1995-03-23 Glaxo Group Limited 3-(tetrazólýl-benzyl)amínó-piperadidín afleiður

Also Published As

Publication number Publication date
FI961270A (fi) 1996-05-03
CO4290298A1 (es) 1996-04-17
GR3029354T3 (en) 1999-05-28
US5703240A (en) 1997-12-30
AU7697494A (en) 1995-04-10
ATE173255T1 (de) 1998-11-15
NO961156D0 (no) 1996-03-21
BG100487A (bg) 1996-12-31
CN1135218A (zh) 1996-11-06
EP0720609B1 (en) 1998-11-11
IS4208A (is) 1995-03-23
DE69414590D1 (de) 1998-12-17
WO1995008549A1 (en) 1995-03-30
PE18295A1 (es) 1995-07-27
UA44711C2 (uk) 2002-03-15
OA10576A (en) 2002-06-03
JPH09505275A (ja) 1997-05-27
HRP940575A2 (en) 1997-02-28
AP9400671A0 (en) 1994-10-31
HU217428B (hu) 2000-01-28
BG62169B1 (bg) 1999-04-30
AU681190B2 (en) 1997-08-21
PL179585B1 (pl) 2000-09-29
NO307830B1 (no) 2000-06-05
CA2172529A1 (en) 1995-03-30
SK280901B6 (sk) 2000-09-12
EP0720609A1 (en) 1996-07-10
NO961156L (no) 1996-05-21
NZ273614A (en) 1997-09-22
HUT75648A (en) 1997-05-28
CZ285479B6 (cs) 1999-08-11
CZ83096A3 (en) 1996-09-11
IL111002A0 (en) 1994-11-28
HK1004219A1 (en) 1998-11-20
HU9600722D0 (en) 1996-05-28
SI0720609T1 (en) 1999-02-28
DE69414590T2 (de) 1999-04-15
HRP940575B1 (en) 2000-06-30
JP2865872B2 (ja) 1999-03-08
PL313619A1 (en) 1996-07-08
FI961270A0 (fi) 1996-03-19
CN1061041C (zh) 2001-01-24
US5843966A (en) 1998-12-01
SK38396A3 (en) 1997-02-05
AP495A (en) 1996-05-28
JPH11106341A (ja) 1999-04-20
ES2123829T3 (es) 1999-01-16
DK0720609T3 (da) 1999-07-26

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