IL107133A - Piperidine derivatives, their preparation and pharmaceutical preparations containing them - Google Patents

Piperidine derivatives, their preparation and pharmaceutical preparations containing them

Info

Publication number
IL107133A
IL107133A IL107133A IL10713393A IL107133A IL 107133 A IL107133 A IL 107133A IL 107133 A IL107133 A IL 107133A IL 10713393 A IL10713393 A IL 10713393A IL 107133 A IL107133 A IL 107133A
Authority
IL
Israel
Prior art keywords
alkyl
disorder
compound
formula
optionally substituted
Prior art date
Application number
IL107133A
Other languages
English (en)
Hebrew (he)
Other versions
IL107133A0 (en
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of IL107133A0 publication Critical patent/IL107133A0/xx
Publication of IL107133A publication Critical patent/IL107133A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL107133A 1992-09-28 1993-09-27 Piperidine derivatives, their preparation and pharmaceutical preparations containing them IL107133A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9211551A FR2696177B1 (fr) 1992-09-28 1992-09-28 Dérivés de pipéridine, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
IL107133A0 IL107133A0 (en) 1993-12-28
IL107133A true IL107133A (en) 1998-03-10

Family

ID=9433967

Family Applications (1)

Application Number Title Priority Date Filing Date
IL107133A IL107133A (en) 1992-09-28 1993-09-27 Piperidine derivatives, their preparation and pharmaceutical preparations containing them

Country Status (24)

Country Link
US (1) US5434169A (ja)
EP (1) EP0591027A1 (ja)
JP (1) JPH06211838A (ja)
KR (1) KR940007020A (ja)
CN (1) CN1087339A (ja)
AP (1) AP424A (ja)
AU (1) AU658533B2 (ja)
CA (1) CA2107061A1 (ja)
CZ (1) CZ282080B6 (ja)
DZ (1) DZ1718A1 (ja)
FI (1) FI934221A (ja)
FR (1) FR2696177B1 (ja)
HU (2) HUT65303A (ja)
IL (1) IL107133A (ja)
MA (1) MA22981A1 (ja)
MX (1) MX9305932A (ja)
NO (1) NO933435L (ja)
NZ (1) NZ248776A (ja)
OA (1) OA09840A (ja)
PL (1) PL172860B1 (ja)
SK (1) SK103193A3 (ja)
TN (1) TNSN93107A1 (ja)
TW (1) TW272190B (ja)
ZA (1) ZA937156B (ja)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2191106T3 (es) * 1995-09-18 2003-09-01 Glaxo Group Ltd Uso de ondansetron en la fabricacion de un medicamento para el tratamiento del temblor.
EP0918518A4 (en) * 1996-04-19 2002-05-02 Univ California TREATMENT OF MIND AND MOOD DISEASES WITH GLUTAMATERGIC MODULATORS.
FR2765221B1 (fr) * 1997-06-25 1999-07-30 Synthelabo Derives de 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide, leur preparation et leur application en therapeutique
US6013654A (en) * 1997-08-14 2000-01-11 Pharmacia & Upjohn Company Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases
GB9918425D0 (en) * 1999-08-04 1999-10-06 Novartis Ag Organic compounds
US6887870B1 (en) * 1999-10-12 2005-05-03 Bristol-Myers Squibb Company Heterocyclic sodium/proton exchange inhibitors and method
US7183305B2 (en) 2003-11-11 2007-02-27 Allergan, Inc. Process for the synthesis of imidazoles
US7880017B2 (en) 2003-11-11 2011-02-01 Allergan, Inc. Process for the synthesis of imidazoles
WO2007014851A2 (en) * 2005-07-29 2007-02-08 F. Hoffmann-La Roche Ag Indol-3-yl-carbonyl-piperidin and piperazin derivatives
FR2925902B1 (fr) * 2008-01-02 2011-01-07 Sanofi Aventis DERIVES D'IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
WO2010080357A1 (en) * 2008-12-18 2010-07-15 Boehringer Ingelheim International Gmbh Serotonin 5-ht2b receptor inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61210080A (ja) * 1985-03-13 1986-09-18 Chisso Corp アルデヒドラクトンの製造法
FR2579596B1 (fr) * 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique
US5008390A (en) * 1985-05-23 1991-04-16 Smithkline Beckman Corporation Compounds for preparing 6-phenyl-2,3-dihydroimidazo[2,1-b]-thiazoles and corresponding thiazines
IT1230703B (it) * 1989-01-26 1991-10-29 Luso Farmaco Inst Derivati imidazolonici ad attivita' antiipertensiva, loro metodi di preparazione e composizioni farmaceutiche che li contengono.
US4925851A (en) * 1989-05-23 1990-05-15 Sandoz Pharmaceuticals Corp. 2- or 4-substituted-[2-(1H-imidazol-1-yl)ethyl]piperidines
FR2671083B1 (fr) * 1990-12-31 1994-12-23 Inst Nat Sante Rech Med Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques.

Also Published As

Publication number Publication date
NZ248776A (en) 1995-09-26
HUT65303A (en) 1994-05-02
MA22981A1 (fr) 1994-04-01
PL172860B1 (pl) 1997-12-31
OA09840A (fr) 1994-08-15
CN1087339A (zh) 1994-06-01
MX9305932A (es) 1994-04-29
NO933435D0 (no) 1993-09-27
NO933435L (no) 1994-03-29
PL300515A1 (en) 1994-04-05
HU9302727D0 (en) 1993-12-28
CZ282080B6 (cs) 1997-05-14
DZ1718A1 (fr) 2002-02-17
IL107133A0 (en) 1993-12-28
KR940007020A (ko) 1994-04-26
FI934221A (fi) 1994-03-29
FI934221A0 (fi) 1993-09-27
TNSN93107A1 (fr) 1994-03-17
CA2107061A1 (en) 1994-03-29
AP424A (en) 1995-11-04
HU211249A9 (en) 1995-11-28
JPH06211838A (ja) 1994-08-02
AU4860693A (en) 1994-04-14
SK103193A3 (en) 1994-08-10
CZ9302015A3 (en) 1994-04-13
US5434169A (en) 1995-07-18
FR2696177A1 (fr) 1994-04-01
EP0591027A1 (fr) 1994-04-06
FR2696177B1 (fr) 1995-05-12
AU658533B2 (en) 1995-04-13
ZA937156B (en) 1994-05-23
AP9300575A0 (en) 1993-10-31
TW272190B (ja) 1996-03-11

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Legal Events

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FF Patent granted
RH Patent void