NO933435L - Piperidinderivater, deres fremstilling og anvendelse - Google Patents

Piperidinderivater, deres fremstilling og anvendelse

Info

Publication number
NO933435L
NO933435L NO933435A NO933435A NO933435L NO 933435 L NO933435 L NO 933435L NO 933435 A NO933435 A NO 933435A NO 933435 A NO933435 A NO 933435A NO 933435 L NO933435 L NO 933435L
Authority
NO
Norway
Prior art keywords
group
alkoxy
preparation
hydrogen atom
piperidine derivatives
Prior art date
Application number
NO933435A
Other languages
English (en)
Other versions
NO933435D0 (no
Inventor
Samir Jegham
Itzchak Angel
Thomas Andrew Purcell
Johannes Schoemaker
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO933435D0 publication Critical patent/NO933435D0/no
Publication of NO933435L publication Critical patent/NO933435L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Forbindelser med formel (l) hvor R er et hydrogenatom.eller en rettkjedet eller forgrenet (Cj-CJalkylgruppe, og Ar er en fenylgruppe som eventuelt er substituert med et eller flere radikaler valgt blant halogen- atomene og aminogruppene, (Cj-Cj)alkoksy eller (C3-C6)syklo- alkyl(C!-C2)alkoksy eller en heteroarylgruppe, med unntak av de forbindelser hvor R er et hydrogenatom og Ar er en fenylgruppe eller en 4-klorfenylgruppe, og deres addisjonssalter av farmasøytiske tålbare syrer. Forbindelse har terapeutisk anvendelse.
NO933435A 1992-09-28 1993-09-27 Piperidinderivater, deres fremstilling og anvendelse NO933435L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9211551A FR2696177B1 (fr) 1992-09-28 1992-09-28 Dérivés de pipéridine, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
NO933435D0 NO933435D0 (no) 1993-09-27
NO933435L true NO933435L (no) 1994-03-29

Family

ID=9433967

Family Applications (1)

Application Number Title Priority Date Filing Date
NO933435A NO933435L (no) 1992-09-28 1993-09-27 Piperidinderivater, deres fremstilling og anvendelse

Country Status (24)

Country Link
US (1) US5434169A (no)
EP (1) EP0591027A1 (no)
JP (1) JPH06211838A (no)
KR (1) KR940007020A (no)
CN (1) CN1087339A (no)
AP (1) AP424A (no)
AU (1) AU658533B2 (no)
CA (1) CA2107061A1 (no)
CZ (1) CZ282080B6 (no)
DZ (1) DZ1718A1 (no)
FI (1) FI934221A (no)
FR (1) FR2696177B1 (no)
HU (2) HUT65303A (no)
IL (1) IL107133A (no)
MA (1) MA22981A1 (no)
MX (1) MX9305932A (no)
NO (1) NO933435L (no)
NZ (1) NZ248776A (no)
OA (1) OA09840A (no)
PL (1) PL172860B1 (no)
SK (1) SK103193A3 (no)
TN (1) TNSN93107A1 (no)
TW (1) TW272190B (no)
ZA (1) ZA937156B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR199800488T1 (xx) * 1995-09-18 1998-05-21 Glaxo Group Limited Diskinezi i�in 5-HT3 resept�r antagonistleri.
EP0918518A4 (en) * 1996-04-19 2002-05-02 Univ California TREATMENT OF MIND AND MOOD DISEASES WITH GLUTAMATERGIC MODULATORS.
FR2765221B1 (fr) * 1997-06-25 1999-07-30 Synthelabo Derives de 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide, leur preparation et leur application en therapeutique
US6013654A (en) * 1997-08-14 2000-01-11 Pharmacia & Upjohn Company Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases
GB9918425D0 (en) * 1999-08-04 1999-10-06 Novartis Ag Organic compounds
US6887870B1 (en) * 1999-10-12 2005-05-03 Bristol-Myers Squibb Company Heterocyclic sodium/proton exchange inhibitors and method
US7880017B2 (en) 2003-11-11 2011-02-01 Allergan, Inc. Process for the synthesis of imidazoles
US7183305B2 (en) 2003-11-11 2007-02-27 Allergan, Inc. Process for the synthesis of imidazoles
RU2422442C2 (ru) * 2005-07-29 2011-06-27 Ф. Хоффманн-Ля Рош Аг Производные индол-3-ил-карбонил-пиперидина и пиперазина
FR2925902B1 (fr) * 2008-01-02 2011-01-07 Sanofi Aventis DERIVES D'IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
US8609696B2 (en) 2008-12-18 2013-12-17 Boehringer Ingelheim International Gmbh Serotonin 5-HT2B receptor inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61210080A (ja) * 1985-03-13 1986-09-18 Chisso Corp アルデヒドラクトンの製造法
FR2579596B1 (fr) * 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique
US5008390A (en) * 1985-05-23 1991-04-16 Smithkline Beckman Corporation Compounds for preparing 6-phenyl-2,3-dihydroimidazo[2,1-b]-thiazoles and corresponding thiazines
IT1230703B (it) * 1989-01-26 1991-10-29 Luso Farmaco Inst Derivati imidazolonici ad attivita' antiipertensiva, loro metodi di preparazione e composizioni farmaceutiche che li contengono.
US4925851A (en) * 1989-05-23 1990-05-15 Sandoz Pharmaceuticals Corp. 2- or 4-substituted-[2-(1H-imidazol-1-yl)ethyl]piperidines
FR2671083B1 (fr) * 1990-12-31 1994-12-23 Inst Nat Sante Rech Med Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques.

Also Published As

Publication number Publication date
OA09840A (fr) 1994-08-15
AP424A (en) 1995-11-04
EP0591027A1 (fr) 1994-04-06
HUT65303A (en) 1994-05-02
FR2696177B1 (fr) 1995-05-12
CN1087339A (zh) 1994-06-01
MA22981A1 (fr) 1994-04-01
AU658533B2 (en) 1995-04-13
SK103193A3 (en) 1994-08-10
IL107133A (en) 1998-03-10
HU9302727D0 (en) 1993-12-28
AP9300575A0 (en) 1993-10-31
PL172860B1 (pl) 1997-12-31
ZA937156B (en) 1994-05-23
TW272190B (no) 1996-03-11
NZ248776A (en) 1995-09-26
TNSN93107A1 (fr) 1994-03-17
IL107133A0 (en) 1993-12-28
PL300515A1 (en) 1994-04-05
HU211249A9 (en) 1995-11-28
CA2107061A1 (en) 1994-03-29
US5434169A (en) 1995-07-18
DZ1718A1 (fr) 2002-02-17
KR940007020A (ko) 1994-04-26
MX9305932A (es) 1994-04-29
NO933435D0 (no) 1993-09-27
FI934221A0 (fi) 1993-09-27
CZ9302015A3 (en) 1994-04-13
CZ282080B6 (cs) 1997-05-14
FI934221A (fi) 1994-03-29
FR2696177A1 (fr) 1994-04-01
JPH06211838A (ja) 1994-08-02
AU4860693A (en) 1994-04-14

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