ZA937156B - Piperidine derivatives their preparation and theirapplication in therapy - Google Patents

Piperidine derivatives their preparation and theirapplication in therapy

Info

Publication number
ZA937156B
ZA937156B ZA937156A ZA937156A ZA937156B ZA 937156 B ZA937156 B ZA 937156B ZA 937156 A ZA937156 A ZA 937156A ZA 937156 A ZA937156 A ZA 937156A ZA 937156 B ZA937156 B ZA 937156B
Authority
ZA
South Africa
Prior art keywords
theirapplication
therapy
preparation
piperidine derivatives
piperidine
Prior art date
Application number
ZA937156A
Other languages
English (en)
Inventor
Samir Jegham
Thomas Purcell
Itzchak Angel
Johannes Schoemaker
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of ZA937156B publication Critical patent/ZA937156B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ZA937156A 1992-09-28 1993-09-27 Piperidine derivatives their preparation and theirapplication in therapy ZA937156B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9211551A FR2696177B1 (fr) 1992-09-28 1992-09-28 Dérivés de pipéridine, leur préparation et leur application en thérapeutique.

Publications (1)

Publication Number Publication Date
ZA937156B true ZA937156B (en) 1994-05-23

Family

ID=9433967

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA937156A ZA937156B (en) 1992-09-28 1993-09-27 Piperidine derivatives their preparation and theirapplication in therapy

Country Status (24)

Country Link
US (1) US5434169A (no)
EP (1) EP0591027A1 (no)
JP (1) JPH06211838A (no)
KR (1) KR940007020A (no)
CN (1) CN1087339A (no)
AP (1) AP424A (no)
AU (1) AU658533B2 (no)
CA (1) CA2107061A1 (no)
CZ (1) CZ282080B6 (no)
DZ (1) DZ1718A1 (no)
FI (1) FI934221A (no)
FR (1) FR2696177B1 (no)
HU (2) HUT65303A (no)
IL (1) IL107133A (no)
MA (1) MA22981A1 (no)
MX (1) MX9305932A (no)
NO (1) NO933435L (no)
NZ (1) NZ248776A (no)
OA (1) OA09840A (no)
PL (1) PL172860B1 (no)
SK (1) SK103193A3 (no)
TN (1) TNSN93107A1 (no)
TW (1) TW272190B (no)
ZA (1) ZA937156B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR199800488T1 (xx) * 1995-09-18 1998-05-21 Glaxo Group Limited Diskinezi i�in 5-HT3 resept�r antagonistleri.
EP0918518A4 (en) * 1996-04-19 2002-05-02 Univ California TREATMENT OF MIND AND MOOD DISEASES WITH GLUTAMATERGIC MODULATORS.
FR2765221B1 (fr) * 1997-06-25 1999-07-30 Synthelabo Derives de 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide, leur preparation et leur application en therapeutique
US6013654A (en) * 1997-08-14 2000-01-11 Pharmacia & Upjohn Company Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases
GB9918425D0 (en) * 1999-08-04 1999-10-06 Novartis Ag Organic compounds
US6887870B1 (en) * 1999-10-12 2005-05-03 Bristol-Myers Squibb Company Heterocyclic sodium/proton exchange inhibitors and method
US7880017B2 (en) 2003-11-11 2011-02-01 Allergan, Inc. Process for the synthesis of imidazoles
US7183305B2 (en) 2003-11-11 2007-02-27 Allergan, Inc. Process for the synthesis of imidazoles
RU2422442C2 (ru) * 2005-07-29 2011-06-27 Ф. Хоффманн-Ля Рош Аг Производные индол-3-ил-карбонил-пиперидина и пиперазина
FR2925902B1 (fr) * 2008-01-02 2011-01-07 Sanofi Aventis DERIVES D'IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
US8609696B2 (en) 2008-12-18 2013-12-17 Boehringer Ingelheim International Gmbh Serotonin 5-HT2B receptor inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61210080A (ja) * 1985-03-13 1986-09-18 Chisso Corp アルデヒドラクトンの製造法
FR2579596B1 (fr) * 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique
US5008390A (en) * 1985-05-23 1991-04-16 Smithkline Beckman Corporation Compounds for preparing 6-phenyl-2,3-dihydroimidazo[2,1-b]-thiazoles and corresponding thiazines
IT1230703B (it) * 1989-01-26 1991-10-29 Luso Farmaco Inst Derivati imidazolonici ad attivita' antiipertensiva, loro metodi di preparazione e composizioni farmaceutiche che li contengono.
US4925851A (en) * 1989-05-23 1990-05-15 Sandoz Pharmaceuticals Corp. 2- or 4-substituted-[2-(1H-imidazol-1-yl)ethyl]piperidines
FR2671083B1 (fr) * 1990-12-31 1994-12-23 Inst Nat Sante Rech Med Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques.

Also Published As

Publication number Publication date
OA09840A (fr) 1994-08-15
AP424A (en) 1995-11-04
EP0591027A1 (fr) 1994-04-06
HUT65303A (en) 1994-05-02
FR2696177B1 (fr) 1995-05-12
CN1087339A (zh) 1994-06-01
MA22981A1 (fr) 1994-04-01
AU658533B2 (en) 1995-04-13
SK103193A3 (en) 1994-08-10
IL107133A (en) 1998-03-10
HU9302727D0 (en) 1993-12-28
AP9300575A0 (en) 1993-10-31
PL172860B1 (pl) 1997-12-31
TW272190B (no) 1996-03-11
NZ248776A (en) 1995-09-26
TNSN93107A1 (fr) 1994-03-17
NO933435L (no) 1994-03-29
IL107133A0 (en) 1993-12-28
PL300515A1 (en) 1994-04-05
HU211249A9 (en) 1995-11-28
CA2107061A1 (en) 1994-03-29
US5434169A (en) 1995-07-18
DZ1718A1 (fr) 2002-02-17
KR940007020A (ko) 1994-04-26
MX9305932A (es) 1994-04-29
NO933435D0 (no) 1993-09-27
FI934221A0 (fi) 1993-09-27
CZ9302015A3 (en) 1994-04-13
CZ282080B6 (cs) 1997-05-14
FI934221A (fi) 1994-03-29
FR2696177A1 (fr) 1994-04-01
JPH06211838A (ja) 1994-08-02
AU4860693A (en) 1994-04-14

Similar Documents

Publication Publication Date Title
ZA937155B (en) Piperidine derivatives their preparation and theirapplication in therapeutics
ZA93958B (en) Piperazine and piperidine derivatives and their use in therapy
IL101865A0 (en) Thiopyranopyrrole derivatives and their preparation
GB2221390B (en) Niacin-containing composition and its therapeutic use
HU9400190D0 (en) Therapeutic compositions and methods
IL99612A0 (en) 2-aminopyrimidine-4-carboxamide derivatives,their preparation and their use in therapy
ZA885150B (en) N-aminobutyl-n-phenylarylamide derivatives,their preparation and their application in therapy
IL118119A0 (en) Azacycloalkane derivatives their preparation and their application in therapy
ZA937156B (en) Piperidine derivatives their preparation and theirapplication in therapy
ZA943649B (en) Piperidine derivatives their preparation and use
IL92682A0 (en) Piperidinedione derivatives and their reduction to 4-phenylpiperidines
ZA964563B (en) Isoindole derivatives their preparation and their application in therapy
IL101617A0 (en) 2-aminopyrimidine-4-carboxamide derivatives,their preparation and their application in therapy
GB9413090D0 (en) Benzazepine derivatives compositions containing them and their use in therapy
IL107726A0 (en) Pyrrole derivatives their preparation and their therapeutic use
GB2221464B (en) Oxaza heterocycles and their use in pharmaceutical compositions
ZA892841B (en) Benzothiazepin-4-one derivative,their preparation and their application in therapy
GB9621419D0 (en) 3-3-disubstituted piperidine derivatives and their use as therapeutic agents
ZA904290B (en) 1-phenyl-1,4-dihydro-3-amino-4-oxopyridazine derivatives,their preparation and their application in therapy
NZ230921A (en) 3-phenyloxymethyl-cephalosporin derivatives and medicaments
AU1745092A (en) Thiazolidine derivatives and their use in therapy
GB9112545D0 (en) Improvements in and relating to hinges
HK1003571A1 (en) Alkenyltetrazole derivatives their preparation and use
ZA939333B (en) 3-(6-quinolylmethyl)-4H-imidazol-4-one derivatives their preparation and their application in therapy
NZ248041A (en) Aminoalkyl- tetrahydrofuran derivatives and medicaments