HU229800B1 - Stabilized aqueous suspensions for parenteral use containing steroids - Google Patents
Stabilized aqueous suspensions for parenteral use containing steroids Download PDFInfo
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- HU229800B1 HU229800B1 HU0302021A HUP0302021A HU229800B1 HU 229800 B1 HU229800 B1 HU 229800B1 HU 0302021 A HU0302021 A HU 0302021A HU P0302021 A HUP0302021 A HU P0302021A HU 229800 B1 HU229800 B1 HU 229800B1
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- pharmaceutical formulation
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- methionine
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- 239000007900 aqueous suspension Substances 0.000 title claims description 30
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- PSGAAPLEWMOORI-PEINSRQWSA-N medroxyprogesterone acetate Chemical compound C([C@@]12C)CC(=O)C=C1[C@@H](C)C[C@@H]1[C@@H]2CC[C@]2(C)[C@@](OC(C)=O)(C(C)=O)CC[C@H]21 PSGAAPLEWMOORI-PEINSRQWSA-N 0.000 claims description 25
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Classifications
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- A61K9/0012—Galenical forms characterised by the site of application
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- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Dispersion Chemistry (AREA)
- Dermatology (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Oncology (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| US09/571,395 US6495534B2 (en) | 2000-05-15 | 2000-05-15 | Stabilized aqueous suspensions for parenteral use |
| PCT/EP2001/004643 WO2001087266A1 (en) | 2000-05-15 | 2001-04-25 | Stabilized aqueous suspensions for parenteral use |
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| HUP0302021A3 HUP0302021A3 (en) | 2011-03-28 |
| HU229800B1 true HU229800B1 (en) | 2014-07-28 |
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| WO2004043375A2 (en) * | 2002-11-08 | 2004-05-27 | Bristol-Myers Squibb Company | Pharmaceutical compositions and methods of using taxane derivatives |
| DE602004015755D1 (de) * | 2003-03-31 | 2008-09-25 | Alza Corp | Nicht wässrige einphasige visköse vehikel und formulierungen die diese vehikel verwenden |
| KR101288265B1 (ko) * | 2003-09-03 | 2013-07-26 | 미스콘 트레이딩 에스.에이. | 자궁 내막증의 치료 방법 |
| US20050171167A1 (en) * | 2003-11-04 | 2005-08-04 | Haby Thomas A. | Process and formulation containing epothilones and analogs thereof |
| US20050106214A1 (en) * | 2003-11-14 | 2005-05-19 | Guohua Chen | Excipients in drug delivery vehicles |
| CA2581076A1 (en) * | 2004-09-14 | 2006-03-23 | Molecular Therapeutics, Inc. | D-methionine formulation with improved biopharmaceutical properties |
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| US10806740B2 (en) | 2012-06-18 | 2020-10-20 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
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| US9649353B2 (en) | 2013-09-17 | 2017-05-16 | Terapio Corporation | Methods of preventing or treating mucositis by administering RLIP76 |
| CN104706578B (zh) * | 2013-12-14 | 2019-04-23 | 天津金耀集团有限公司 | 一种醋酸甲泼尼龙混悬注射液组合物的制备方法 |
| MX2016014281A (es) | 2014-05-22 | 2017-02-22 | Therapeuticsmd Inc | Formulaciones y terapias de reemplazo de combinación de hormonas naturales. |
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| US2861920A (en) * | 1954-05-04 | 1958-11-25 | Upjohn Co | Therapeutic suspensions of steroids containing pvp and/or pva |
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| US4154820A (en) * | 1976-02-23 | 1979-05-15 | Akzona Incorporated | Compositions containing alkali metal sulfate salts of conjugated estrogens and antioxidants as stabilizers |
| JP2577744B2 (ja) | 1986-07-18 | 1997-02-05 | 中外製薬株式会社 | 安定な顆粒球コロニ−刺激因子含有製剤 |
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-
2000
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2001
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- 2001-04-25 JP JP2001583735A patent/JP4205341B2/ja not_active Expired - Lifetime
- 2001-04-25 WO PCT/EP2001/004643 patent/WO2001087266A1/en not_active Ceased
- 2001-04-25 DK DK01945040T patent/DK1282402T3/da active
- 2001-04-25 BR BR0110841-7A patent/BR0110841A/pt not_active Application Discontinuation
- 2001-04-25 CA CA002409059A patent/CA2409059C/en not_active Expired - Lifetime
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- 2001-04-25 HU HU0302021A patent/HU229800B1/hu unknown
- 2001-04-25 PL PL365793A patent/PL203075B1/pl unknown
- 2001-04-25 AU AU2001267371A patent/AU2001267371B2/en not_active Expired
- 2001-04-25 EE EEP200200631A patent/EE05376B1/xx unknown
- 2001-04-25 HK HK03106493.6A patent/HK1054194B/zh not_active IP Right Cessation
- 2001-04-25 EA EA200201208A patent/EA007682B1/ru not_active IP Right Cessation
- 2001-04-25 SI SI200130485T patent/SI1282402T1/sl unknown
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- 2001-04-25 EP EP01945040A patent/EP1282402B1/en not_active Expired - Lifetime
- 2001-04-25 AT AT01945040T patent/ATE313316T1/de active
- 2001-04-25 CZ CZ20023750A patent/CZ303872B6/cs not_active IP Right Cessation
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- 2001-04-25 CN CNB018095895A patent/CN100473376C/zh not_active Expired - Lifetime
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- 2001-04-25 SK SK1598-2002A patent/SK287641B6/sk not_active IP Right Cessation
- 2001-04-25 AU AU6737101A patent/AU6737101A/xx active Pending
- 2001-04-25 KR KR1020027015431A patent/KR100828957B1/ko not_active Expired - Lifetime
- 2001-05-09 TW TW090111029A patent/TWI256310B/zh not_active IP Right Cessation
- 2001-05-14 AR ARP010102268A patent/AR029924A1/es not_active Application Discontinuation
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2002
- 2002-08-21 US US10/225,320 patent/US20030114430A1/en not_active Abandoned
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Owner name: PFIZER ITALIA S.R.L., IT Free format text: FORMER OWNER(S): PHARMACIA & UPJOHN CO., US; PHARMACIA ITALIA S.P.A., IT |