HU180273B - Process for producing 1,5-disubstituted-2-pyrrolidone derivatives - Google Patents

Process for producing 1,5-disubstituted-2-pyrrolidone derivatives Download PDF

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Publication number
HU180273B
HU180273B HU77PI587A HUPI000587A HU180273B HU 180273 B HU180273 B HU 180273B HU 77PI587 A HU77PI587 A HU 77PI587A HU PI000587 A HUPI000587 A HU PI000587A HU 180273 B HU180273 B HU 180273B
Authority
HU
Hungary
Prior art keywords
pyrrolidone
group
formula
reaction
prepared
Prior art date
Application number
HU77PI587A
Other languages
German (de)
English (en)
Hungarian (hu)
Inventor
Albin J Nelson
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of HU180273B publication Critical patent/HU180273B/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms
    • C07D207/262-Pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU77PI587A 1976-08-06 1977-08-05 Process for producing 1,5-disubstituted-2-pyrrolidone derivatives HU180273B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US71236276A 1976-08-06 1976-08-06

Publications (1)

Publication Number Publication Date
HU180273B true HU180273B (en) 1983-02-28

Family

ID=24861795

Family Applications (1)

Application Number Title Priority Date Filing Date
HU77PI587A HU180273B (en) 1976-08-06 1977-08-05 Process for producing 1,5-disubstituted-2-pyrrolidone derivatives

Country Status (31)

Country Link
JP (2) JPS5321159A (xx)
AR (1) AR217080A1 (xx)
AT (1) AT362887B (xx)
AU (1) AU508007B2 (xx)
BE (1) BE857506A (xx)
BG (1) BG31073A3 (xx)
CA (1) CA1077948A (xx)
CH (1) CH624934A5 (xx)
CS (1) CS221269B2 (xx)
DD (2) DD136135A5 (xx)
DE (1) DE2735904A1 (xx)
DK (1) DK352077A (xx)
ES (2) ES461388A1 (xx)
FI (1) FI70009C (xx)
FR (1) FR2369260A1 (xx)
GB (2) GB1556570A (xx)
GR (1) GR68688B (xx)
HU (1) HU180273B (xx)
IE (1) IE45505B1 (xx)
IL (1) IL52615A (xx)
LU (1) LU77936A1 (xx)
NL (1) NL7708637A (xx)
NO (1) NO772752L (xx)
NZ (1) NZ184806A (xx)
PH (1) PH17398A (xx)
PL (2) PL112931B1 (xx)
PT (1) PT66891B (xx)
SE (1) SE423813B (xx)
SU (3) SU703016A3 (xx)
YU (1) YU192577A (xx)
ZA (1) ZA774704B (xx)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5695569A (en) * 1979-12-27 1981-08-03 Canon Inc Forming method for bar lens sphere face
US4321201A (en) * 1980-09-22 1982-03-23 E. I. Du Pont De Nemours And Company Optically active tert-alkyl 7-(2-oxo-5-carbonyloxypyrrolidinyl) heptanoates
JPS59137224A (ja) * 1983-01-25 1984-08-07 Mitsubishi Electric Corp 電気鉄道用き電電圧補償装置
PT1132086E (pt) * 2000-01-31 2006-09-29 Pfizer Prod Inc Utilizacao de agonistas selectivos para o receptor da prostaglandina (pge2) 4 (ep4) para o tratamento de falha renal aguda e cronica
AU2001290250A1 (en) * 2000-09-21 2002-04-02 Ono Pharmaceutical Co. Ltd. Ep4 receptor agonists containing 8-azaprostaglandin derivatives as the active ingredient
DK1339678T3 (da) * 2000-11-27 2008-02-04 Pfizer Prod Inc Selektive agonister til EP4-receptor til behandling af osteoporose
CA2454584C (en) * 2001-07-23 2009-09-22 Ono Pharmaceutical Co., Ltd. Pharmaceutical composition for treatment of diseases associated with decrease in bone mass comprising ep4 agonist as active ingredient
DE60307607T2 (de) * 2002-03-18 2007-08-09 Pfizer Products Inc., Groton Verwendung von selektiven ep4 rezeptor agonisten zur behandlung von krankheiten
US6573294B1 (en) * 2002-05-14 2003-06-03 Allergan, Inc. 8-azaprostaglandin analogs as agents for lowering intraocular pressure
US7256211B1 (en) * 2003-01-21 2007-08-14 Ono Pharmaceutical Co., Ltd. 8-azaprostaglandin derivatives and medical use thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1386146A (en) * 1972-05-03 1975-03-05 Ici Ltd Cyclopentane derivatives
JPS511460A (en) * 1974-06-24 1976-01-08 Tanabe Seiyaku Co 22 piroridonjudotaino seiho
JPS514166A (ja) * 1974-06-28 1976-01-14 Tanabe Seiyaku Co 22piroridonjudotaino seiho
US3975399A (en) * 1974-08-06 1976-08-17 E. I. Du Pont De Nemours And Company 1,5-Disubstituted-2-pyrrolidinones, -3-pyrrolin-2-ones, and -4-pyrrolin-2-ones
DE2528664A1 (de) * 1975-06-27 1977-01-13 Hoechst Ag Pyrrolidone und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
IE45505B1 (en) 1982-09-08
CS221269B2 (en) 1983-04-29
FI772376A (xx) 1978-02-07
CA1077948A (en) 1980-05-20
IL52615A (en) 1981-09-13
DD143768A5 (de) 1980-09-10
PH17398A (en) 1984-08-08
PT66891A (en) 1977-09-01
YU192577A (en) 1983-04-30
SU818480A3 (ru) 1981-03-30
FI70009C (fi) 1986-09-12
PT66891B (en) 1979-01-26
AU508007B2 (en) 1980-03-06
AR217080A1 (es) 1980-02-29
GB1556570A (en) 1979-11-28
FI70009B (fi) 1986-01-31
AU2751577A (en) 1979-02-08
ES471349A1 (es) 1979-09-16
IL52615A0 (en) 1977-10-31
BE857506A (fr) 1978-02-06
DK352077A (da) 1978-02-07
AT362887B (de) 1981-06-25
DD136135A5 (de) 1979-06-20
PL200124A1 (pl) 1978-05-22
CH624934A5 (xx) 1981-08-31
BG31073A3 (en) 1981-10-15
IE45505L (en) 1978-02-06
JPS5321159A (en) 1978-02-27
JPS5531147B2 (xx) 1980-08-15
ZA774704B (en) 1978-06-28
SE423813B (sv) 1982-06-07
LU77936A1 (xx) 1978-04-27
JPS5555161A (en) 1980-04-22
PL112931B1 (en) 1980-11-29
GB1556569A (en) 1979-11-28
SU850000A3 (ru) 1981-07-23
ES461388A1 (es) 1978-12-01
FR2369260A1 (fr) 1978-05-26
ATA579477A (de) 1980-11-15
NL7708637A (nl) 1978-02-08
NZ184806A (en) 1980-04-28
GR68688B (xx) 1982-02-01
NO772752L (no) 1978-02-07
JPS585196B2 (ja) 1983-01-29
SU703016A3 (ru) 1979-12-05
DE2735904A1 (de) 1978-02-09
SE7708642L (sv) 1978-02-07
FR2369260B1 (xx) 1982-02-12

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