HRP20100017T1 - Derivati heteroaril-alkilkarbamata, postupak njihovog dobivanja i njihova upotreba kao inhibitora enzima faah - Google Patents
Derivati heteroaril-alkilkarbamata, postupak njihovog dobivanja i njihova upotreba kao inhibitora enzima faah Download PDFInfo
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- HRP20100017T1 HRP20100017T1 HR20100017T HRP20100017T HRP20100017T1 HR P20100017 T1 HRP20100017 T1 HR P20100017T1 HR 20100017 T HR20100017 T HR 20100017T HR P20100017 T HRP20100017 T HR P20100017T HR P20100017 T1 HRP20100017 T1 HR P20100017T1
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- ethyl
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- oxazolidinedione
- pyridyl
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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
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- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/12—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
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- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/04—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
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- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
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- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
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- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
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- C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
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- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
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- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
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- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/26—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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- C07D471/04—Ortho-condensed systems
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0401949A FR2866886B1 (fr) | 2004-02-26 | 2004-02-26 | Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique |
| PCT/FR2005/000451 WO2005090292A1 (fr) | 2004-02-26 | 2005-02-25 | Derives d’heteroaryl-alkylcarbamates, leur preparation et leur application comme inhibiteurs de l’enzyme faah |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20100017T1 true HRP20100017T1 (hr) | 2010-02-28 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20100017T HRP20100017T1 (hr) | 2004-02-26 | 2005-02-25 | Derivati heteroaril-alkilkarbamata, postupak njihovog dobivanja i njihova upotreba kao inhibitora enzima faah |
Country Status (28)
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|---|---|
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| EP (2) | EP1720829B1 (enExample) |
| JP (1) | JP4824668B2 (enExample) |
| KR (1) | KR20070011297A (enExample) |
| CN (1) | CN1926097B (enExample) |
| AR (1) | AR047973A1 (enExample) |
| AT (1) | ATE445592T1 (enExample) |
| AU (1) | AU2005223423B2 (enExample) |
| BR (1) | BRPI0508193A (enExample) |
| CA (1) | CA2554609A1 (enExample) |
| CY (1) | CY1109716T1 (enExample) |
| DE (1) | DE602005017122D1 (enExample) |
| DK (1) | DK1720829T3 (enExample) |
| ES (1) | ES2334449T3 (enExample) |
| FR (1) | FR2866886B1 (enExample) |
| HR (1) | HRP20100017T1 (enExample) |
| IL (1) | IL177329A (enExample) |
| MA (1) | MA28367A1 (enExample) |
| NO (1) | NO20064329L (enExample) |
| NZ (1) | NZ550008A (enExample) |
| PL (1) | PL1720829T3 (enExample) |
| PT (1) | PT1720829E (enExample) |
| RS (1) | RS51246B (enExample) |
| RU (1) | RU2364586C2 (enExample) |
| SI (1) | SI1720829T1 (enExample) |
| TW (1) | TW200533637A (enExample) |
| WO (1) | WO2005090292A1 (enExample) |
| ZA (1) | ZA200606724B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2866884B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives d'aryl-et d'heteroaryl-piperidinecarboxylates, leur preparation et leur application en therapeutique |
| FR2866885B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique |
| EP2141150B1 (en) | 2007-04-26 | 2013-12-11 | Takeda Pharmaceutical Company Limited | Bicyclic compound and pharmaceutical use thereof |
| WO2009070497A1 (en) * | 2007-11-28 | 2009-06-04 | Smithkline Beecham Corporation | SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE |
| KR101799429B1 (ko) * | 2010-05-03 | 2017-11-21 | 에스케이바이오팜 주식회사 | 신경 세포 사멸 또는 신경 퇴화를 억제하기 위한 약학적 조성물 |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2866734A (en) * | 1956-12-05 | 1958-12-30 | Us Vitamin Corp | 3-pyridylethyl 2, 4-oxazolidinediones and process |
| US3054794A (en) * | 1958-01-17 | 1962-09-18 | Us Vitamin Pharm Corp | Process for preparing 3-(aminoalkyl)-oxazolidine-2, 4-diones |
| US3742022A (en) * | 1967-05-08 | 1973-06-26 | A Verbiscar | Carbamate esters of physiologically active ph enenthylamines |
| US3876661A (en) * | 1971-03-02 | 1975-04-08 | Anthony J Verbiscar | Carbamate esters of serotonin and analogs |
| DE19647382A1 (de) * | 1996-11-15 | 1998-05-20 | Hoechst Ag | Heterocyclen als Inhibitoren der Leukozytenadhäsion und VLA-4-Antagonisten |
| CA2308850C (en) * | 1997-11-24 | 2007-07-10 | The Scripps Research Institute | Inhibitors of gap junction communication |
| AU2001229580A1 (en) * | 2000-01-18 | 2001-08-14 | Nuerogen Corporation | Substituted imidazoles as selective modulators of bradykinin b2 receptors |
| WO2002087569A1 (en) * | 2001-04-27 | 2002-11-07 | Bristol-Myers Squibb Company | Bisarylimidazolyl fatty acid amide hydrolase inhibitors |
| AU2003226755A1 (en) * | 2002-04-27 | 2003-11-17 | Merck Patent Gmbh | Carboxylic acid amides |
| FR2843964B1 (fr) * | 2002-08-29 | 2004-10-01 | Sanofi Synthelabo | Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique |
| CN100408556C (zh) * | 2002-10-07 | 2008-08-06 | 加利福尼亚大学董事会 | 通过阻断花生四烯酰乙醇酰胺的水解调节焦虑 |
| US7662971B2 (en) * | 2002-10-08 | 2010-02-16 | The Scripps Research Institute | Inhibitors of fatty acid amide hydrolase |
| US7309701B2 (en) * | 2002-11-19 | 2007-12-18 | Sanofi-Aventis Deutschland Gmbh | Pyridazinone derivatives as pharmaceuticals and pharmaceutical compositions containing them |
| FR2850377B1 (fr) * | 2003-01-23 | 2009-02-20 | Sanofi Synthelabo | Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique |
| FR2854633B1 (fr) * | 2003-05-07 | 2005-06-24 | Sanofi Synthelabo | Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique |
| UA82695C2 (uk) * | 2003-06-06 | 2008-05-12 | Нисан Кемикал Индастриз, Лтд. | Гетероароматичні сполуки як активатори рецептора тромбопоетину |
| US20050032747A1 (en) * | 2003-07-01 | 2005-02-10 | Wilmin Bartolini | COX-2 and FAAH inhibitors |
| EP1680411A2 (en) * | 2003-10-08 | 2006-07-19 | Vertex Pharmaceuticals Incorporated | Modulators of atp-binding cassette transporters containing cycloalkyl or pyranyl groups |
| FR2866885B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique |
| EP1574511A1 (en) * | 2004-03-03 | 2005-09-14 | Bayer CropScience S.A. | 2-Pyridinylethylcarboxamide derivatives and their use as fungicides |
| US20100152188A1 (en) * | 2005-08-05 | 2010-06-17 | Akella Satya Surya Visweswara Srinivas | Novel Heterocyclic Compounds |
| BRPI0616150A2 (pt) * | 2005-09-22 | 2011-06-07 | Sanofi Aventis | derivados de amino-alquil-amida como lìquidos receptores de ccr3 |
| FR2894578B1 (fr) * | 2005-12-12 | 2008-02-01 | Sanofi Aventis Sa | Derives heterocycliques, leur preparation et leur application en therapeutique. |
| US8741960B2 (en) * | 2006-01-25 | 2014-06-03 | Synta Pharmaceuticals Corp. | Substituted aromatic compounds for inflammation and immune-related uses |
| JO2754B1 (en) * | 2006-12-21 | 2014-03-15 | استرازينكا ايه بي | Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders |
| US9549982B2 (en) * | 2009-11-23 | 2017-01-24 | Foundational Biosystems, Llc | Ultra low dose nutraceutical compositions for enhancing sleep quality and treating sleep disorders |
-
2004
- 2004-02-26 FR FR0401949A patent/FR2866886B1/fr not_active Expired - Fee Related
-
2005
- 2005-02-25 WO PCT/FR2005/000451 patent/WO2005090292A1/fr not_active Ceased
- 2005-02-25 KR KR1020067017250A patent/KR20070011297A/ko not_active Abandoned
- 2005-02-25 PT PT05732902T patent/PT1720829E/pt unknown
- 2005-02-25 BR BRPI0508193-9A patent/BRPI0508193A/pt not_active IP Right Cessation
- 2005-02-25 SI SI200530882T patent/SI1720829T1/sl unknown
- 2005-02-25 ES ES05732902T patent/ES2334449T3/es not_active Expired - Lifetime
- 2005-02-25 HR HR20100017T patent/HRP20100017T1/hr unknown
- 2005-02-25 JP JP2007500260A patent/JP4824668B2/ja not_active Expired - Fee Related
- 2005-02-25 RS RSP-2010/0011A patent/RS51246B/sr unknown
- 2005-02-25 PL PL05732902T patent/PL1720829T3/pl unknown
- 2005-02-25 AT AT05732902T patent/ATE445592T1/de active
- 2005-02-25 DK DK05732902.1T patent/DK1720829T3/da active
- 2005-02-25 RU RU2006134026/04A patent/RU2364586C2/ru not_active IP Right Cessation
- 2005-02-25 NZ NZ550008A patent/NZ550008A/en unknown
- 2005-02-25 EP EP05732902A patent/EP1720829B1/fr not_active Expired - Lifetime
- 2005-02-25 TW TW094105874A patent/TW200533637A/zh unknown
- 2005-02-25 DE DE602005017122T patent/DE602005017122D1/de not_active Expired - Lifetime
- 2005-02-25 CN CN2005800058656A patent/CN1926097B/zh not_active Expired - Fee Related
- 2005-02-25 ZA ZA200606724A patent/ZA200606724B/xx unknown
- 2005-02-25 CA CA002554609A patent/CA2554609A1/fr not_active Abandoned
- 2005-02-25 AU AU2005223423A patent/AU2005223423B2/en not_active Ceased
- 2005-02-25 EP EP09172706A patent/EP2251324A1/fr not_active Withdrawn
- 2005-05-24 AR ARP050100666A patent/AR047973A1/es unknown
-
2006
- 2006-08-07 IL IL177329A patent/IL177329A/en not_active IP Right Cessation
- 2006-08-14 US US11/464,355 patent/US7645757B2/en not_active Expired - Fee Related
- 2006-08-22 MA MA29285A patent/MA28367A1/fr unknown
- 2006-09-25 NO NO20064329A patent/NO20064329L/no not_active Application Discontinuation
-
2009
- 2009-11-24 US US12/625,125 patent/US20100069405A1/en not_active Abandoned
-
2010
- 2010-01-11 CY CY20101100030T patent/CY1109716T1/el unknown
-
2011
- 2011-06-09 US US13/156,551 patent/US20110237595A1/en not_active Abandoned
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