HK1212217A1 - Methods of treating alzheimers disease and pharmaceutical compositions thereof - Google Patents

Methods of treating alzheimers disease and pharmaceutical compositions thereof

Info

Publication number
HK1212217A1
HK1212217A1 HK16100112.5A HK16100112A HK1212217A1 HK 1212217 A1 HK1212217 A1 HK 1212217A1 HK 16100112 A HK16100112 A HK 16100112A HK 1212217 A1 HK1212217 A1 HK 1212217A1
Authority
HK
Hong Kong
Prior art keywords
methods
pharmaceutical compositions
alzheimers disease
treating alzheimers
treating
Prior art date
Application number
HK16100112.5A
Other languages
English (en)
Chinese (zh)
Inventor
.施密特
.阿伯格
Original Assignee
Lundbeck As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49118521&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1212217(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck As filed Critical Lundbeck As
Publication of HK1212217A1 publication Critical patent/HK1212217A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/4045Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HK16100112.5A 2012-09-09 2016-01-07 Methods of treating alzheimers disease and pharmaceutical compositions thereof HK1212217A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261698664P 2012-09-09 2012-09-09
US201361782084P 2013-03-14 2013-03-14
PCT/EP2013/068516 WO2014037532A1 (en) 2012-09-09 2013-09-06 Methods of treating alzheimer's disease and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
HK1212217A1 true HK1212217A1 (en) 2016-06-10

Family

ID=49118521

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16100112.5A HK1212217A1 (en) 2012-09-09 2016-01-07 Methods of treating alzheimers disease and pharmaceutical compositions thereof

Country Status (33)

Country Link
US (4) US9375418B2 (pt)
EP (1) EP2892563B1 (pt)
JP (2) JP6693744B2 (pt)
KR (2) KR102342127B1 (pt)
CN (1) CN104619344A (pt)
AP (1) AP2015008306A0 (pt)
AU (1) AU2013311573B2 (pt)
BR (1) BR112015005117B1 (pt)
CA (1) CA2883751C (pt)
CL (1) CL2015000578A1 (pt)
CY (1) CY1121062T1 (pt)
DK (1) DK2892563T3 (pt)
EA (1) EA030448B1 (pt)
ES (1) ES2703630T3 (pt)
GE (1) GEP201706776B (pt)
HK (1) HK1212217A1 (pt)
HR (1) HRP20182069T1 (pt)
IL (1) IL237369B (pt)
JO (1) JO3459B1 (pt)
LT (1) LT2892563T (pt)
MX (1) MX368305B (pt)
MY (1) MY182539A (pt)
NI (1) NI201500031A (pt)
NZ (1) NZ630589A (pt)
PL (1) PL2892563T3 (pt)
PT (1) PT2892563T (pt)
RS (1) RS58104B1 (pt)
RU (1) RU2675786C2 (pt)
SG (1) SG11201501774QA (pt)
SI (1) SI2892563T1 (pt)
TN (1) TN2015000076A1 (pt)
TW (1) TWI632909B (pt)
WO (1) WO2014037532A1 (pt)

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JO3459B1 (ar) 2012-09-09 2020-07-05 H Lundbeck As تركيبات صيدلانية لعلاج مرض الزهايمر
TWI627174B (zh) 2013-03-14 2018-06-21 比利時商健生藥品公司 P2x7調控劑
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JO3639B1 (ar) * 2014-07-04 2020-08-27 H Lundbeck As صورة متعددة الشكل جديدة لـ n-[2-(6-فلورو-1h-إندول-3-يل)إيثيل]-3-(2،2،3،3-تترا فلورو بروبوكسي)بنزيل أمين هيدروكلوريد
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CN109562085A (zh) 2015-06-12 2019-04-02 阿速万科学有限责任公司 用于预防和治疗rem睡眠行为障碍的二芳基和芳基杂芳基脲衍生物
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PT3484467T (pt) 2016-05-18 2020-06-16 Suven Life Sciences Ltd Combinação de antagonistas puros do recetor 5-ht6 com inibidores de acetilcolinesterase
CN106309436A (zh) * 2016-07-25 2017-01-11 宁波大学 可用作乙酰胆碱酯酶抑制剂的色胺衍生物及其用途
CN107118146B (zh) * 2017-04-13 2019-09-03 宁波大学 一种6-溴色胺衍生物及其制备方法和用途
HUE053636T2 (hu) * 2017-05-24 2021-07-28 H Lundbeck As 5-HT6 receptor antagonista és acetilkolin-észteráz inhibitor kombinációja Alzheimer-kór kezelésében történõ alkalmazásra ApoE4 alléleket hordozó betegek szubpopulációjában
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KR20210069080A (ko) 2018-09-28 2021-06-10 얀센 파마슈티카 엔.브이. 모노아실글리세롤 리파아제 조절제
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JP2023518511A (ja) 2020-03-26 2023-05-01 ヤンセン ファーマシューティカ エヌ.ベー. モノアシルグリセロールリパーゼ調節因子

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Also Published As

Publication number Publication date
TN2015000076A1 (en) 2016-06-29
WO2014037532A1 (en) 2014-03-13
LT2892563T (lt) 2019-01-10
US20180071254A1 (en) 2018-03-15
US20160354343A1 (en) 2016-12-08
US10660878B2 (en) 2020-05-26
KR20150065680A (ko) 2015-06-15
US9789085B2 (en) 2017-10-17
CL2015000578A1 (es) 2015-05-15
CY1121062T1 (el) 2019-12-11
MX2015002879A (es) 2015-07-06
KR20200137028A (ko) 2020-12-08
AP2015008306A0 (en) 2015-03-31
TWI632909B (zh) 2018-08-21
JP2015528471A (ja) 2015-09-28
DK2892563T3 (en) 2019-01-21
RU2675786C2 (ru) 2018-12-25
TW201414474A (zh) 2014-04-16
JP2019059760A (ja) 2019-04-18
PL2892563T3 (pl) 2019-04-30
KR102342127B1 (ko) 2021-12-21
AU2013311573B2 (en) 2017-10-12
EP2892563A1 (en) 2015-07-15
MX368305B (es) 2019-09-27
IL237369A0 (en) 2015-04-30
RS58104B1 (sr) 2019-02-28
JP6693744B2 (ja) 2020-05-13
AU2013311573A1 (en) 2015-03-12
ES2703630T3 (es) 2019-03-11
RU2015107877A (ru) 2016-10-27
HRP20182069T1 (hr) 2019-02-08
AU2013311573A8 (en) 2015-03-19
NI201500031A (es) 2016-02-15
CN104619344A (zh) 2015-05-13
BR112015005117A2 (pt) 2017-07-04
SG11201501774QA (en) 2015-05-28
CA2883751C (en) 2020-11-24
US20160256437A1 (en) 2016-09-08
MY182539A (en) 2021-01-25
SI2892563T1 (sl) 2019-02-28
US9375418B2 (en) 2016-06-28
EA030448B1 (ru) 2018-08-31
GEP201706776B (en) 2017-11-27
IL237369B (en) 2018-11-29
PT2892563T (pt) 2019-01-10
EA201590353A1 (ru) 2016-03-31
CA2883751A1 (en) 2014-03-13
US20140073681A1 (en) 2014-03-13
NZ630589A (en) 2015-12-24
US9687473B2 (en) 2017-06-27
EP2892563B1 (en) 2018-11-14
JO3459B1 (ar) 2020-07-05
BR112015005117B1 (pt) 2022-06-21

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