HK1198165A1 - 氟化雌激素受體調節劑及其用途 - Google Patents

氟化雌激素受體調節劑及其用途

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Publication number
HK1198165A1
HK1198165A1 HK14111641.4A HK14111641A HK1198165A1 HK 1198165 A1 HK1198165 A1 HK 1198165A1 HK 14111641 A HK14111641 A HK 14111641A HK 1198165 A1 HK1198165 A1 HK 1198165A1
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HK
Hong Kong
Prior art keywords
fluorinated
estrogen receptor
receptor modulators
modulators
estrogen
Prior art date
Application number
HK14111641.4A
Other languages
English (en)
Inventor
尼古拉斯．
．史密斯
史蒂文．
．加維克
梅米特．卡爾曼
約翰尼．
．長澤
安迪利耶．
．萊
賽琳．博納富斯
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Publication date
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Publication of HK1198165A1 publication Critical patent/HK1198165A1/zh

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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
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    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
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    • C07D311/60—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with aryl radicals attached in position 2
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    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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    • C07D311/70—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with two hydrocarbon radicals attached in position 2 and elements other than carbon and hydrogen in position 6
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Psychology (AREA)
HK14111641.4A 2011-12-14 2014-11-18 氟化雌激素受體調節劑及其用途 HK1198165A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161570756P 2011-12-14 2011-12-14
PCT/US2012/069933 WO2013090836A1 (en) 2011-12-14 2012-12-14 Fluorinated estrogen receptor modulators and uses thereof

Publications (1)

Publication Number Publication Date
HK1198165A1 true HK1198165A1 (zh) 2015-03-13

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HK14111641.4A HK1198165A1 (zh) 2011-12-14 2014-11-18 氟化雌激素受體調節劑及其用途

Country Status (15)

Country Link
US (2) US9193714B2 (zh)
EP (2) EP2791132A4 (zh)
JP (2) JP2015500346A (zh)
KR (1) KR20140101399A (zh)
CN (1) CN104114551B (zh)
AU (1) AU2012351942B2 (zh)
BR (1) BR112014014124A2 (zh)
CA (1) CA2857057A1 (zh)
EA (1) EA029559B1 (zh)
HK (1) HK1198165A1 (zh)
IL (1) IL232793A (zh)
MX (1) MX357496B (zh)
PH (1) PH12014501351B1 (zh)
SG (1) SG11201403002RA (zh)
WO (2) WO2013090829A1 (zh)

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