HK1177195A1 - Substituted 3-phenylpropionic acids and the use thereof 3- - Google Patents

Substituted 3-phenylpropionic acids and the use thereof 3-

Info

Publication number
HK1177195A1
HK1177195A1 HK13104154.9A HK13104154A HK1177195A1 HK 1177195 A1 HK1177195 A1 HK 1177195A1 HK 13104154 A HK13104154 A HK 13104154A HK 1177195 A1 HK1177195 A1 HK 1177195A1
Authority
HK
Hong Kong
Prior art keywords
substituted
phenylpropionic acids
phenylpropionic
acids
Prior art date
Application number
HK13104154.9A
Other languages
English (en)
Chinese (zh)
Inventor
Thomas Lampe
Michael Hahn
Johannes-Peter Stasch
Karl-Heinz Schlemmer
Frank Wunder
Sheikh Sherif El
Volkhart Min-Jian Li
Eva-Maria Becker
Friederike Stoll
Andreas Knorr
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of HK1177195A1 publication Critical patent/HK1177195A1/xx

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    • C07C233/88Carboxylic acid amides having nitrogen atoms of carboxamide groups bound to an acyclic carbon atom and to a carbon atom of a six-membered aromatic ring wherein at least one ortho-hydrogen atom has been replaced
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
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    • A61K31/655Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
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    • C07C205/36Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system
    • C07C205/38Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system the oxygen atom of at least one of the etherified hydroxy groups being further bound to a carbon atom of a six-membered aromatic ring, e.g. nitrodiphenyl ethers
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    • C07C233/55Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a carbon atom of an unsaturated carbon skeleton
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HK13104154.9A 2009-10-28 2013-04-03 Substituted 3-phenylpropionic acids and the use thereof 3- HK1177195A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102009046115A DE102009046115A1 (de) 2009-10-28 2009-10-28 Substituierte 3-Phenylpropansäuren und ihre Verwendung
PCT/EP2010/065910 WO2011051165A1 (fr) 2009-10-28 2010-10-21 Acides 3-phénylpropioniques substitués et leur utilisation

Publications (1)

Publication Number Publication Date
HK1177195A1 true HK1177195A1 (en) 2013-08-16

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HK13104154.9A HK1177195A1 (en) 2009-10-28 2013-04-03 Substituted 3-phenylpropionic acids and the use thereof 3-

Country Status (23)

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US (2) US20110130445A1 (fr)
EP (1) EP2493845B1 (fr)
JP (1) JP5801312B2 (fr)
KR (1) KR20120101411A (fr)
CN (1) CN102712577B (fr)
AR (1) AR079015A1 (fr)
AU (1) AU2010311678B2 (fr)
BR (1) BR112012010057A2 (fr)
CA (1) CA2777152C (fr)
DE (1) DE102009046115A1 (fr)
DK (1) DK2493845T3 (fr)
ES (1) ES2446970T3 (fr)
HK (1) HK1177195A1 (fr)
HR (1) HRP20140270T1 (fr)
IL (1) IL218989A (fr)
MX (1) MX2012004951A (fr)
PL (1) PL2493845T3 (fr)
PT (1) PT2493845E (fr)
RU (1) RU2553263C2 (fr)
TW (1) TWI487519B (fr)
UY (1) UY32970A (fr)
WO (1) WO2011051165A1 (fr)
ZA (1) ZA201202465B (fr)

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DE102008018675A1 (de) 2008-04-14 2009-10-15 Bayer Schering Pharma Aktiengesellschaft Oxo-heterocyclisch substituierte Carbonsäure-Derivate und ihre Verwendung
DE102009012314A1 (de) * 2009-03-09 2010-09-16 Bayer Schering Pharma Aktiengesellschaft Oxo-heterocyclisch substituierte Alkylcarbonsäuren und ihre Verwendung
DE102009046115A1 (de) 2009-10-28 2011-09-08 Bayer Schering Pharma Aktiengesellschaft Substituierte 3-Phenylpropansäuren und ihre Verwendung
EP2549875B1 (fr) 2010-03-25 2015-05-13 Merck Sharp & Dohme Corp. Activateurs de guanylate cyclase solubles
MA34330B1 (fr) 2010-05-27 2013-06-01 Merck Sharp & Dohme Activateurs de guanylate cyclase soluble
US8895583B2 (en) 2010-10-28 2014-11-25 Merck Sharp & Dohme Corp. Soluble guanylate cyclase activators
BR112013013663A2 (pt) 2010-12-07 2016-09-06 Bayer Ip Gmbh ácidos 1-benzilcicloalquilcarboxílicos substituídos e sua utilização
DE102011007272A1 (de) * 2011-04-13 2012-10-18 Bayer Pharma Aktiengesellschaft Verzweigte 3-Phenylpropionsäure-Derivate und ihre Verwendung
CN104144920A (zh) * 2012-02-28 2014-11-12 皮拉马尔企业有限公司 作为gpr促效剂的苯基烷酸衍生物
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ZA201202465B (en) 2013-08-28
CA2777152C (fr) 2017-09-19
US20110130445A1 (en) 2011-06-02
CN102712577A (zh) 2012-10-03
WO2011051165A1 (fr) 2011-05-05
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JP2013509369A (ja) 2013-03-14
CA2777152A1 (fr) 2011-05-05
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IL218989A (en) 2015-10-29
DK2493845T3 (en) 2014-03-24
EP2493845B1 (fr) 2013-12-25
BR112012010057A2 (pt) 2019-09-24
PT2493845E (pt) 2014-02-24
AU2010311678B2 (en) 2015-09-03
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TWI487519B (zh) 2015-06-11
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IL218989A0 (en) 2012-06-28
UY32970A (es) 2011-05-31
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US20140142069A1 (en) 2014-05-22
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