PL2247601T3 - Tiazopirymidynony i ich zastosowanie - Google Patents

Tiazopirymidynony i ich zastosowanie

Info

Publication number
PL2247601T3
PL2247601T3 PL09771847T PL09771847T PL2247601T3 PL 2247601 T3 PL2247601 T3 PL 2247601T3 PL 09771847 T PL09771847 T PL 09771847T PL 09771847 T PL09771847 T PL 09771847T PL 2247601 T3 PL2247601 T3 PL 2247601T3
Authority
PL
Poland
Prior art keywords
thiazopyrimidinones
Prior art date
Application number
PL09771847T
Other languages
English (en)
Inventor
John Joseph Deadman
Eric Dale Jones
Giang Thanh Le
David Ian Rhodes
Neeranat Thienthong
De Graff Nicholas Andrew Van
Lisa Jane Winfield
Original Assignee
Avexa Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2008903405A external-priority patent/AU2008903405A0/en
Application filed by Avexa Ltd filed Critical Avexa Ltd
Publication of PL2247601T3 publication Critical patent/PL2247601T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL09771847T 2008-07-02 2009-07-02 Tiazopirymidynony i ich zastosowanie PL2247601T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
AU2008903405A AU2008903405A0 (en) 2008-07-02 Thiazopyrimidinones and uses thereof
US16193109P 2009-03-20 2009-03-20
US16193109A 2009-03-20 2009-03-20
PCT/AU2009/000856 WO2010000030A1 (en) 2008-07-02 2009-07-02 Thiazopyrimidinones and uses thereof
EP09771847.2A EP2247601B1 (en) 2008-07-02 2009-07-02 Thiazopyrimidinones and uses thereof

Publications (1)

Publication Number Publication Date
PL2247601T3 true PL2247601T3 (pl) 2013-09-30

Family

ID=41465415

Family Applications (1)

Application Number Title Priority Date Filing Date
PL09771847T PL2247601T3 (pl) 2008-07-02 2009-07-02 Tiazopirymidynony i ich zastosowanie

Country Status (7)

Country Link
US (1) US8426405B2 (pl)
EP (1) EP2247601B1 (pl)
JP (1) JP5539978B2 (pl)
CA (1) CA2729649A1 (pl)
ES (1) ES2408654T3 (pl)
PL (1) PL2247601T3 (pl)
WO (1) WO2010000030A1 (pl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2005252685B2 (en) 2004-06-07 2010-12-16 THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES, CENTERS FOR DISEASE CONTROL AND PREVENTION Real-time PCR point mutation assays for detecting HIV-1 resistance to antiviral drugs
US8206929B2 (en) 2009-01-07 2012-06-26 Roche Molecular Systems, Inc. Nucleic acid amplification with allele-specific suppression of sequence variants
MX2012009869A (es) 2010-02-26 2012-09-12 Japan Tobacco Inc Derivado de 1, 3,4, 8-tetrahidro-2h-pirido[1, 2-a]pirazina y sus uso como inhibidor de la integrasa del vih.
US9879317B2 (en) 2011-02-17 2018-01-30 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services, Centers For Disease Control And Prevention Real-time PCR point mutation assays for detecting HIV-1 resistance to antiviral drugs
IL286328B1 (en) 2019-03-22 2026-04-01 Gilead Sciences Inc Tricyclic bridging compounds of carbamoylpyridone and their pharmaceutical use
CN115151540A (zh) 2019-12-02 2022-10-04 风暴治疗有限公司 作为mettl3抑制剂的多杂环化合物
CR20220418A (es) 2020-02-24 2022-10-10 Gilead Sciences Inc Compuestos tetracíclicos para el tratamiento de infecciones por vih
CA3192145A1 (en) 2020-09-30 2022-04-07 Gilead Sciences, Inc. Bridged tricyclic carbamoylpyridone compounds and uses thereof
JP7591155B2 (ja) 2021-01-19 2024-11-27 ギリアード サイエンシーズ， インコーポレイテッド 置換ピリドトリアジン化合物及びその使用
TWI856796B (zh) 2022-04-06 2024-09-21 美商基利科學股份有限公司 橋聯三環胺甲醯基吡啶酮化合物及其用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU551718B2 (en) * 1981-07-15 1986-05-08 Farmitalia Carlo Erba S.P.A. Substituted thiazolo(3,2-alpha)pyrimidines
ZA824797B (en) * 1981-07-15 1983-04-27 Erba Farmitalia Substituted thiazolo(3,2-a)pyrimidines and process for their preparation
DK3042894T1 (da) 2001-08-10 2016-11-07 Shionogi & Co Antiviralt middel
DE60209381T2 (de) * 2001-10-26 2006-10-05 Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. N-substituierte hydroxypyrimidinoncarboxamid-hemmer der hiv-integrase
TW200526635A (en) * 2003-12-22 2005-08-16 Shionogi & Co Hydroxypyrimidinone derivative having HIV integrase inhibitory activity
BRPI0720564A2 (pt) * 2006-12-22 2011-08-16 Avexa Ltd pirimidinonas biciclìcas e seus usos
EP2291377B1 (en) * 2008-07-02 2015-02-18 Avexa Limited Imidazopyrimidinones and uses thereof
BRPI0913934A2 (pt) * 2008-07-02 2015-10-20 Avexa Ltd compostos tendo propriedades antivirais

Also Published As

Publication number Publication date
WO2010000030A1 (en) 2010-01-07
US20110281861A1 (en) 2011-11-17
JP2011526246A (ja) 2011-10-06
US8426405B2 (en) 2013-04-23
EP2247601A4 (en) 2011-01-19
CA2729649A1 (en) 2010-01-07
ES2408654T3 (es) 2013-06-21
JP5539978B2 (ja) 2014-07-02
EP2247601B1 (en) 2013-04-10
EP2247601A1 (en) 2010-11-10

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