HK1135976A1 - Pyridin-3-yl derivatives as immunomodulating agents - Google Patents

Pyridin-3-yl derivatives as immunomodulating agents

Info

Publication number
HK1135976A1
HK1135976A1 HK10102256.3A HK10102256A HK1135976A1 HK 1135976 A1 HK1135976 A1 HK 1135976A1 HK 10102256 A HK10102256 A HK 10102256A HK 1135976 A1 HK1135976 A1 HK 1135976A1
Authority
HK
Hong Kong
Prior art keywords
pyridin
derivatives
immunomodulating agents
immunomodulating
agents
Prior art date
Application number
HK10102256.3A
Other languages
English (en)
Inventor
Martin Bolli
David Lehmann
Boris Mathys
Claus Mueller
Oliver Nayler
Beat Steiner
Joerg Velker
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of HK1135976A1 publication Critical patent/HK1135976A1/xx

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
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    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Transplantation (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK10102256.3A 2006-09-08 2010-03-02 Pyridin-3-yl derivatives as immunomodulating agents HK1135976A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IB2006053187 2006-09-08
PCT/IB2007/053593 WO2008029370A1 (en) 2006-09-08 2007-09-06 Pyridin-3-yl derivatives as immunomodulating agents

Publications (1)

Publication Number Publication Date
HK1135976A1 true HK1135976A1 (en) 2010-06-18

Family

ID=38982768

Family Applications (1)

Application Number Title Priority Date Filing Date
HK10102256.3A HK1135976A1 (en) 2006-09-08 2010-03-02 Pyridin-3-yl derivatives as immunomodulating agents

Country Status (27)

Country Link
US (1) US8288554B2 (da)
EP (1) EP2069335B1 (da)
JP (1) JP5253400B2 (da)
KR (1) KR101454937B1 (da)
CN (1) CN101522670B (da)
AR (1) AR062684A1 (da)
AU (1) AU2007292992B2 (da)
BR (1) BRPI0716633A2 (da)
CA (1) CA2661315C (da)
CL (1) CL2007002594A1 (da)
CY (1) CY1113858T1 (da)
DK (1) DK2069335T3 (da)
ES (1) ES2400163T3 (da)
HK (1) HK1135976A1 (da)
HR (1) HRP20130180T1 (da)
IL (1) IL197394A (da)
MA (1) MA30717B1 (da)
MX (1) MX2009002234A (da)
MY (1) MY150661A (da)
NO (1) NO20091409L (da)
NZ (1) NZ576059A (da)
PL (1) PL2069335T3 (da)
PT (1) PT2069335E (da)
RU (1) RU2454413C2 (da)
SI (1) SI2069335T1 (da)
TW (1) TWI399371B (da)
WO (1) WO2008029370A1 (da)

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NZ576059A (en) 2012-03-30
CN101522670B (zh) 2012-05-23
IL197394A0 (en) 2009-12-24
RU2454413C2 (ru) 2012-06-27
AU2007292992A1 (en) 2008-03-13
AR062684A1 (es) 2008-11-26
BRPI0716633A2 (pt) 2013-09-24
NO20091409L (no) 2009-04-07
ES2400163T3 (es) 2013-04-08
IL197394A (en) 2013-08-29
TW200817358A (en) 2008-04-16
CA2661315A1 (en) 2008-03-13
EP2069335A1 (en) 2009-06-17
KR20090060327A (ko) 2009-06-11
WO2008029370A1 (en) 2008-03-13
MY150661A (en) 2014-02-14
RU2009112726A (ru) 2010-10-20
SI2069335T1 (sl) 2013-04-30
US20100168005A1 (en) 2010-07-01
EP2069335B1 (en) 2012-12-26
TWI399371B (zh) 2013-06-21
MA30717B1 (fr) 2009-09-01
US8288554B2 (en) 2012-10-16
PT2069335E (pt) 2013-03-04
DK2069335T3 (da) 2013-02-18
CY1113858T1 (el) 2016-07-27
PL2069335T3 (pl) 2013-05-31
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HRP20130180T1 (hr) 2013-03-31
JP5253400B2 (ja) 2013-07-31
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CL2007002594A1 (es) 2008-06-06
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