GT200600078A - Derivados de indol, benzotiofeno, benzofurano e indeno cicloalquil condensados - Google Patents
Derivados de indol, benzotiofeno, benzofurano e indeno cicloalquil condensadosInfo
- Publication number
- GT200600078A GT200600078A GT200600078A GT200600078A GT200600078A GT 200600078 A GT200600078 A GT 200600078A GT 200600078 A GT200600078 A GT 200600078A GT 200600078 A GT200600078 A GT 200600078A GT 200600078 A GT200600078 A GT 200600078A
- Authority
- GT
- Guatemala
- Prior art keywords
- benzotiofen
- cyclalkyl
- inden
- indol
- benzofuran
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/82—Carbazoles; Hydrogenated carbazoles
- C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
- C07D233/76—Two oxygen atoms, e.g. hydantoin with substituted hydrocarbon radicals attached to the third ring carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
LA PRESENTE INVENCIÓN SE REFIERE A COMPUESTOS DE FÓRMULA GENERAL I EN LA QUE R1,R2,R3,R4,R5,W,Z,Y,X,Q,R15,R16,N,M, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS SON MODULADORES DE SEROTONINA POR LO QUE SON DE UTILIDAD ENTRE OTRAS COSAS PARA EJERCER UNA ACCIÓN ANTIDEPRESIVA.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US65366605P | 2005-02-17 | 2005-02-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
GT200600078A true GT200600078A (es) | 2007-04-12 |
Family
ID=36609274
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200600078A GT200600078A (es) | 2005-02-17 | 2006-02-16 | Derivados de indol, benzotiofeno, benzofurano e indeno cicloalquil condensados |
Country Status (13)
Country | Link |
---|---|
US (2) | US7297704B2 (es) |
EP (1) | EP1856126A2 (es) |
JP (1) | JP2008530229A (es) |
CN (1) | CN101120002A (es) |
AR (1) | AR052674A1 (es) |
AU (1) | AU2006214233A1 (es) |
BR (1) | BRPI0608353A2 (es) |
CA (1) | CA2597616A1 (es) |
GT (1) | GT200600078A (es) |
MX (1) | MX2007009783A (es) |
PA (1) | PA8663501A1 (es) |
TW (1) | TW200640931A (es) |
WO (1) | WO2006089053A2 (es) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102006016885A1 (de) * | 2006-04-11 | 2007-10-18 | Bayer Cropscience Ag | Mit bicyclischen Radikalen N-substituierte Diamino-1,3,5-triazine, Verfahren für ihre Herstellung, Zubereitungen davon und ihre Verwendung als Herbizide und Pflanzenwachstumsregulatoren |
UA98777C2 (en) | 2006-11-20 | 2012-06-25 | Эли Лилли Энд Компани | Tetrahydrocyclopenta[b]indole compounds as androgen receptor modulators |
JP5603327B2 (ja) * | 2008-05-16 | 2014-10-08 | イーライ リリー アンド カンパニー | テトラヒドロシクロペンタ[b]インドールアンドロゲン受容体調節物質 |
WO2010016584A1 (ja) | 2008-08-07 | 2010-02-11 | 杏林製薬株式会社 | ビシクロ[2.2.2]オクチルアミン誘導体の製造方法 |
CN102216267A (zh) * | 2008-09-16 | 2011-10-12 | 杏林制药株式会社 | 氨基乙酰基吡咯烷甲腈衍生物的纯化方法及其盐 |
GB0908394D0 (en) | 2009-05-15 | 2009-06-24 | Univ Leuven Kath | Novel viral replication inhibitors |
GB0913636D0 (en) | 2009-08-05 | 2009-09-16 | Univ Leuven Kath | Novel viral replication inhibitors |
CN102762575B (zh) | 2009-12-04 | 2015-04-15 | 桑诺维恩药品公司 | 多环化合物及其使用方法 |
US9132129B2 (en) | 2010-11-15 | 2015-09-15 | Katholieke Universiteit Leuven | Antiviral compounds |
AR088377A1 (es) * | 2011-10-20 | 2014-05-28 | Siena Biotech Spa | Proceso para la preparacion de 6-cloro-2,3,4,9-tetrahidro-1h-carbazol-1-carboxamida y compuestos intermedios de esta |
CN105125571B (zh) * | 2015-07-17 | 2018-11-06 | 四川大学 | Prmt1抑制剂在制备治疗可卡因成瘾的药物中的用途 |
JP2019523279A (ja) | 2016-07-29 | 2019-08-22 | サノビオン ファーマシューティカルズ インクSunovion Pharmaceuticals Inc. | 化合物および組成物ならびにそれらの使用 |
US10196403B2 (en) | 2016-07-29 | 2019-02-05 | Sunovion Pharmaceuticals Inc. | Compounds and compositions and uses thereof |
US11129807B2 (en) | 2017-02-16 | 2021-09-28 | Sunovion Pharmaceuticals Inc. | Methods of treating schizophrenia |
BR112020001433A2 (pt) | 2017-08-02 | 2020-07-28 | Sunovion Pharmaceuticals Inc. | compostos de isocromano e usos dos mesmos |
CA3091292A1 (en) | 2018-02-16 | 2019-08-22 | Sunovion Pharmaceuticals Inc. | Salts, crystal forms, and production methods thereof |
US11136304B2 (en) | 2019-03-14 | 2021-10-05 | Sunovion Pharmaceuticals Inc. | Salts of a heterocyclic compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof |
BR112022012758A2 (pt) | 2020-01-17 | 2022-09-06 | Daegu Gyeongbuk Medical Innovation Found | Composto, isômero do mesmo ou sal farmaceuticamente aceitável do mesmo, método de preparação e uso do dito composto, composição farmacêutica e alimento funcional saudável |
US11738002B2 (en) | 2020-04-14 | 2023-08-29 | Sunovion Pharmaceuticals Inc. | Methods of treating neurological and psychiatric disorders |
CN113512427B (zh) * | 2021-08-17 | 2023-04-28 | 烟台显华科技集团股份有限公司 | 具有负介电各向异性的液晶化合物、液晶组合物、液晶显示器件 |
CN113512430B (zh) * | 2021-08-17 | 2023-05-02 | 烟台显华科技集团股份有限公司 | 负介电各向异性液晶组合物及液晶显示器件 |
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-
2006
- 2006-02-16 WO PCT/US2006/005521 patent/WO2006089053A2/en active Application Filing
- 2006-02-16 EP EP06735272A patent/EP1856126A2/en not_active Withdrawn
- 2006-02-16 JP JP2007556296A patent/JP2008530229A/ja active Pending
- 2006-02-16 BR BRPI0608353-6A patent/BRPI0608353A2/pt not_active Application Discontinuation
- 2006-02-16 TW TW095105232A patent/TW200640931A/zh unknown
- 2006-02-16 AR ARP060100556A patent/AR052674A1/es not_active Application Discontinuation
- 2006-02-16 AU AU2006214233A patent/AU2006214233A1/en not_active Abandoned
- 2006-02-16 US US11/355,452 patent/US7297704B2/en not_active Expired - Fee Related
- 2006-02-16 PA PA20068663501A patent/PA8663501A1/es unknown
- 2006-02-16 CA CA002597616A patent/CA2597616A1/en not_active Abandoned
- 2006-02-16 MX MX2007009783A patent/MX2007009783A/es unknown
- 2006-02-16 CN CNA2006800053286A patent/CN101120002A/zh active Pending
- 2006-02-16 GT GT200600078A patent/GT200600078A/es unknown
-
2007
- 2007-10-11 US US11/870,660 patent/US20080081910A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US20060205759A1 (en) | 2006-09-14 |
WO2006089053A2 (en) | 2006-08-24 |
US20080081910A1 (en) | 2008-04-03 |
EP1856126A2 (en) | 2007-11-21 |
TW200640931A (en) | 2006-12-01 |
AU2006214233A1 (en) | 2006-08-24 |
WO2006089053A3 (en) | 2007-01-11 |
MX2007009783A (es) | 2007-08-22 |
JP2008530229A (ja) | 2008-08-07 |
BRPI0608353A2 (pt) | 2009-12-01 |
CA2597616A1 (en) | 2006-08-24 |
PA8663501A1 (es) | 2006-11-09 |
US7297704B2 (en) | 2007-11-20 |
CN101120002A (zh) | 2008-02-06 |
AR052674A1 (es) | 2007-03-28 |
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