GT200300075BA - Compuestos que modulan la actividad ppar y procedimientos para su preparacion (patente fraccionaria no. 2 de la solicitud no. pi-20030075) - Google Patents
Compuestos que modulan la actividad ppar y procedimientos para su preparacion (patente fraccionaria no. 2 de la solicitud no. pi-20030075)Info
- Publication number
- GT200300075BA GT200300075BA GT200300075BL GT200300075L GT200300075BA GT 200300075B A GT200300075B A GT 200300075BA GT 200300075B L GT200300075B L GT 200300075BL GT 200300075 L GT200300075 L GT 200300075L GT 200300075B A GT200300075B A GT 200300075BA
- Authority
- GT
- Guatemala
- Prior art keywords
- compounds
- therapy therapy
- procedures
- fractionary
- preparation
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 5
- 238000000034 method Methods 0.000 title abstract 4
- 102000003728 Peroxisome Proliferator-Activated Receptors Human genes 0.000 title abstract 2
- 108090000029 Peroxisome Proliferator-Activated Receptors Proteins 0.000 title abstract 2
- 230000000694 effects Effects 0.000 title abstract 2
- 238000002560 therapeutic procedure Methods 0.000 abstract 12
- 206010060378 Hyperinsulinaemia Diseases 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000003451 hyperinsulinaemic effect Effects 0.000 abstract 1
- 201000008980 hyperinsulinism Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
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- C07C323/10—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C323/18—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
- C07C323/20—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton with singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- C07C317/22—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
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- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Indole Compounds (AREA)
- Pyridine Compounds (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
- Peptides Or Proteins (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
LA INVENCIÓN SE REFIERE A COMPUESTOS QU ALTRAN LA ACTIVIDD DE PPAR. LA INVENCIÓN TAMBIÉN SE REFIERE A LAS SLAES FARAMECÉUTICAMENTE ACEPTABLES DE LOS COMPUESTOS, LAS COMPOSICIONES FARMACÉUTICAMENTE ACEPTABLES QUE COMPRENDEN LOS COMPUESTOS O SUS SALES, Y LOS PROCEDIMIENTOS DE UTILIZACIÓN DE ÉSTOS COMO AGENTES TERAPÉUTICOS PARA TRATAR O PREVENIR LA HIPERLIPIDEMIA, LA HIPERCOLESTEREMIA, LA OBESIDAD, LOS TRASTORNOS ALIMENTARIOS, LA HIPERGLUCEMIA, LA ATEROSCLEROSIS, LA HIPERTRIGLICERIDEMIA, LA HIPERINSULINEMIA Y LA DIABETES EN UN MAMÍFERO, ASÍ COM PROCEDIMIENTOS PARA SUPRIMIR EL APETITO Y MODULAR LOS NIVELES DE LEPTINA EN UN MAMÍFERO. LA PRESENTE INVENCIÓN SE REFIERE TAMBIÉN A PROCEDIMIENTOS PARA LA ELABORACIÓN DE LOS COMPUESTOS DESCRITOS.
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GT200300075AK GT200300075AA (es) | 2002-04-05 | 2003-04-01 | Compuestos que modulan la actividad ppar y procedimientos para su preparacion (patente fraccionaria no. 1 de la solicitud no. pi-20030075) |
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US (4) | US6875780B2 (es) |
EP (1) | EP1494989A2 (es) |
JP (2) | JP3816922B2 (es) |
KR (1) | KR100687166B1 (es) |
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BR (1) | BR0309169A (es) |
CA (1) | CA2481246C (es) |
CO (1) | CO5640080A2 (es) |
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EA (2) | EA009518B1 (es) |
GE (1) | GEP20074244B (es) |
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NO (1) | NO20044795L (es) |
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UA (1) | UA76838C2 (es) |
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- 2003-04-04 TW TW092107732A patent/TWI249522B/zh not_active IP Right Cessation
- 2003-04-04 HN HN2003000113A patent/HN2003000113A/es unknown
- 2003-04-04 PA PA20038570701A patent/PA8570701A1/es unknown
-
2004
- 2004-08-30 IS IS7429A patent/IS7429A/is unknown
- 2004-09-17 CO CO04092873A patent/CO5640080A2/es not_active Application Discontinuation
- 2004-09-28 MA MA27877A patent/MA27189A1/fr unknown
- 2004-10-04 TN TNP2004000191A patent/TNSN04191A1/fr unknown
- 2004-10-05 HR HRP20040916 patent/HRP20040916A2/hr not_active Application Discontinuation
- 2004-11-02 US US10/979,617 patent/US6939875B2/en not_active Ceased
- 2004-11-02 US US10/979,629 patent/US6964983B2/en not_active Expired - Fee Related
- 2004-11-04 NO NO20044795A patent/NO20044795L/no not_active Application Discontinuation
-
2005
- 2005-11-28 US US11/288,022 patent/USRE39916E1/en not_active Expired - Fee Related
- 2005-12-14 JP JP2005360431A patent/JP2006151985A/ja not_active Withdrawn
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