FI962487A - Rapamysiinijohdannaisia - Google Patents

Rapamysiinijohdannaisia Download PDF

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Publication number
FI962487A
FI962487A FI962487A FI962487A FI962487A FI 962487 A FI962487 A FI 962487A FI 962487 A FI962487 A FI 962487A FI 962487 A FI962487 A FI 962487A FI 962487 A FI962487 A FI 962487A
Authority
FI
Finland
Prior art keywords
pct
rapamycin derivatives
date jun
sec
rapamycin
Prior art date
Application number
FI962487A
Other languages
English (en)
Swedish (sv)
Other versions
FI962487A0 (fi
Inventor
Sylvain Cottens
Richard Sedrani
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939325800A external-priority patent/GB9325800D0/en
Priority claimed from GB939325802A external-priority patent/GB9325802D0/en
Priority claimed from GB9407138A external-priority patent/GB9407138D0/en
Priority claimed from GB9421982A external-priority patent/GB9421982D0/en
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of FI962487A publication Critical patent/FI962487A/fi
Publication of FI962487A0 publication Critical patent/FI962487A0/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Transplantation (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI962487A 1993-12-17 1996-06-14 Rapamysiinijohdannaisia FI962487A0 (fi)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB939325800A GB9325800D0 (en) 1993-12-17 1993-12-17 Organic compounds
GB939325802A GB9325802D0 (en) 1993-12-17 1993-12-17 Organic compounds
GB9407138A GB9407138D0 (en) 1994-04-11 1994-04-11 Organic compounds
GB9421982A GB9421982D0 (en) 1994-11-01 1994-11-01 Organic compounds
PCT/EP1994/004191 WO1995016691A1 (en) 1993-12-17 1994-12-16 Rapamycin derivatives useful as immunosuppressants

Publications (2)

Publication Number Publication Date
FI962487A true FI962487A (fi) 1996-06-14
FI962487A0 FI962487A0 (fi) 1996-06-14

Family

ID=27451097

Family Applications (1)

Application Number Title Priority Date Filing Date
FI962487A FI962487A0 (fi) 1993-12-17 1996-06-14 Rapamysiinijohdannaisia

Country Status (21)

Country Link
US (1) US5912253A (fi)
EP (1) EP0734389B1 (fi)
JP (1) JP3745772B2 (fi)
CN (1) CN1046944C (fi)
AT (1) ATE191218T1 (fi)
AU (1) AU687491B2 (fi)
BR (1) BR9408323A (fi)
CZ (1) CZ284650B6 (fi)
DE (1) DE69423781T2 (fi)
DK (1) DK0734389T3 (fi)
ES (1) ES2146741T3 (fi)
FI (1) FI962487A0 (fi)
GR (1) GR3033545T3 (fi)
HU (1) HUT74686A (fi)
NO (1) NO962540L (fi)
NZ (1) NZ277498A (fi)
PL (1) PL314238A1 (fi)
PT (1) PT734389E (fi)
SG (1) SG64372A1 (fi)
SK (1) SK78196A3 (fi)
WO (1) WO1995016691A1 (fi)

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ATE191218T1 (de) 2000-04-15
CN1046944C (zh) 1999-12-01
CN1137797A (zh) 1996-12-11
JPH09506604A (ja) 1997-06-30
NO962540L (no) 1996-06-14
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WO1995016691A1 (en) 1995-06-22
AU1273995A (en) 1995-07-03
US5912253A (en) 1999-06-15
PT734389E (pt) 2000-09-29
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SG64372A1 (en) 1999-04-27
FI962487A0 (fi) 1996-06-14
CZ284650B6 (cs) 1999-01-13
DK0734389T3 (da) 2000-08-21
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BR9408323A (pt) 1997-08-19
ES2146741T3 (es) 2000-08-16
NZ277498A (en) 1998-03-25
CZ175796A3 (en) 1996-09-11
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