FI935529A - Aminometylensubstituerade icke-aromatiska heterocykliska foereningar - Google Patents

Aminometylensubstituerade icke-aromatiska heterocykliska foereningar Download PDF

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Publication number
FI935529A
FI935529A FI935529A FI935529A FI935529A FI 935529 A FI935529 A FI 935529A FI 935529 A FI935529 A FI 935529A FI 935529 A FI935529 A FI 935529A FI 935529 A FI935529 A FI 935529A
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Finland
Prior art keywords
aminomethylsubstituted
aromatic heterocyclic
heterocyclic derivatives
compounds
formula
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FI935529A
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English (en)
Other versions
FI935529A0 (fi
Inventor
Harry R Howard
Brian T O'neill
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Pfizer
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Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI935529A0 publication Critical patent/FI935529A0/fi
Publication of FI935529A publication Critical patent/FI935529A/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI935529A 1992-12-10 1993-12-09 Aminometylensubstituerade icke-aromatiska heterocykliska foereningar FI935529A (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US98865392A 1992-12-10 1992-12-10

Publications (2)

Publication Number Publication Date
FI935529A0 FI935529A0 (fi) 1993-12-09
FI935529A true FI935529A (fi) 1994-06-11

Family

ID=25534364

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935529A FI935529A (fi) 1992-12-10 1993-12-09 Aminometylensubstituerade icke-aromatiska heterocykliska foereningar

Country Status (15)

Country Link
EP (2) EP0675886B1 (fi)
JP (2) JP2722279B2 (fi)
CN (1) CN1092771A (fi)
AT (1) ATE194340T1 (fi)
AU (1) AU5169693A (fi)
CA (1) CA2150123C (fi)
DE (1) DE69328975T2 (fi)
DK (1) DK0675886T3 (fi)
ES (1) ES2147759T3 (fi)
FI (1) FI935529A (fi)
GR (1) GR3034329T3 (fi)
IL (1) IL107843A0 (fi)
MX (1) MX9307810A (fi)
PT (1) PT675886E (fi)
WO (1) WO1994013663A1 (fi)

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US6288225B1 (en) 1996-05-09 2001-09-11 Pfizer Inc Substituted benzolactam compounds as substance P antagonists
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TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
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Also Published As

Publication number Publication date
JPH07509490A (ja) 1995-10-19
JPH1095780A (ja) 1998-04-14
FI935529A0 (fi) 1993-12-09
EP0675886B1 (en) 2000-07-05
CA2150123A1 (en) 1994-06-23
JP3165401B2 (ja) 2001-05-14
EP0675886A1 (en) 1995-10-11
WO1994013663A1 (en) 1994-06-23
JP2722279B2 (ja) 1998-03-04
EP0806423A1 (en) 1997-11-12
ATE194340T1 (de) 2000-07-15
CN1092771A (zh) 1994-09-28
ES2147759T3 (es) 2000-10-01
CA2150123C (en) 2004-12-07
PT675886E (pt) 2000-12-29
DE69328975T2 (de) 2000-11-09
DK0675886T3 (da) 2000-09-18
IL107843A0 (en) 1994-04-12
DE69328975D1 (de) 2000-08-10
MX9307810A (es) 1994-07-29
GR3034329T3 (en) 2000-12-29
AU5169693A (en) 1994-07-04

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