FI924353L - Foerfarande foer framstaellning av nya acylaler av imidazol-5-karboxylsyraderivat - Google Patents

Foerfarande foer framstaellning av nya acylaler av imidazol-5-karboxylsyraderivat Download PDF

Info

Publication number
FI924353L
FI924353L FI924353A FI924353A FI924353L FI 924353 L FI924353 L FI 924353L FI 924353 A FI924353 A FI 924353A FI 924353 A FI924353 A FI 924353A FI 924353 L FI924353 L FI 924353L
Authority
FI
Finland
Prior art keywords
acylaler
nya
imidazole
acid derivatives
carboxyl acid
Prior art date
Application number
FI924353A
Other languages
English (en)
Finnish (fi)
Other versions
FI924353A7 (fi
FI924353A0 (fi
Inventor
Dieter Binder
Josef Weinberger
Original Assignee
Chem Pharm Forsch Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chem Pharm Forsch Gmbh filed Critical Chem Pharm Forsch Gmbh
Publication of FI924353A0 publication Critical patent/FI924353A0/fi
Publication of FI924353A7 publication Critical patent/FI924353A7/fi
Publication of FI924353L publication Critical patent/FI924353L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI924353A 1991-10-04 1992-09-29 Foerfarande foer framstaellning av nya acylaler av imidazol-5-karboxylsyraderivat FI924353L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
AT0198791A AT398202B (de) 1991-10-04 1991-10-04 Neue imidazolderivate, verfahren zu ihrer herstellung und ihre verwendung

Publications (3)

Publication Number Publication Date
FI924353A0 FI924353A0 (fi) 1992-09-29
FI924353A7 FI924353A7 (fi) 1993-04-05
FI924353L true FI924353L (fi) 1993-04-05

Family

ID=3525398

Family Applications (1)

Application Number Title Priority Date Filing Date
FI924353A FI924353L (fi) 1991-10-04 1992-09-29 Foerfarande foer framstaellning av nya acylaler av imidazol-5-karboxylsyraderivat

Country Status (22)

Country Link
US (1) US5298519A (cs)
EP (1) EP0535420A1 (cs)
JP (1) JP2544565B2 (cs)
CN (1) CN1032856C (cs)
AT (1) AT398202B (cs)
AU (1) AU649357B2 (cs)
CA (1) CA2079735A1 (cs)
CZ (1) CZ301992A3 (cs)
FI (1) FI924353L (cs)
HR (1) HRP920817A2 (cs)
HU (1) HUT62291A (cs)
IL (1) IL103329A (cs)
LV (1) LV10256B (cs)
MY (1) MY108350A (cs)
NO (1) NO923798L (cs)
NZ (1) NZ244320A (cs)
RU (1) RU2105764C1 (cs)
SI (1) SI9200240A (cs)
SK (1) SK301992A3 (cs)
TW (1) TW223073B (cs)
YU (1) YU48290B (cs)
ZA (1) ZA927205B (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2105939B1 (es) * 1994-08-02 1998-07-01 Uriach & Cia Sa J Nuevos pirazoles con actividad antagonista de la angiotensina ii.
WO2005011646A2 (en) * 2003-07-31 2005-02-10 Nicox S.A. Nitrooxy derivatives of losartan, valsatan, candesartan, telmisartan, eprosartan and olmesartan as angiotensin-ii receptor blockers for the treatment of cardiovascular diseases
CN101024643A (zh) * 2006-02-20 2007-08-29 上海艾力斯医药科技有限公司 咪唑-5-羧酸类衍生物、制备方法及其应用
CN101195615B (zh) * 2006-12-06 2013-03-27 深圳市信立泰资产管理有限公司 咪唑-5-羧酸衍生物的盐、制备方法及其药物组合物
EP2103610B1 (en) * 2006-12-06 2011-09-21 Shanghai Allist Pharmaceutical., Inc. Salts of imidazol-5-carboxylic acid derivatives, preparation methods and use thereof
CN101214242A (zh) * 2007-01-05 2008-07-09 上海艾力斯医药科技有限公司 新的药用组合物
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
ES2559319T3 (es) 2007-06-04 2016-02-11 Synergy Pharmaceuticals Inc. Agonistas de guanilato cliclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros trastornos
CN101317842A (zh) * 2007-06-07 2008-12-10 上海艾力斯医药科技有限公司 一种咪唑-5-羧酸衍生物的治疗用途
CN101367795B (zh) * 2007-08-17 2012-05-02 上海艾力斯生物医药有限公司 一种咪唑-5-羧酸衍生物及其制备方法
CN101407511B (zh) * 2007-10-11 2013-01-09 上海艾力斯生物医药有限公司 一种结晶型的咪唑-5-羧酸衍生物
WO2009149279A2 (en) 2008-06-04 2009-12-10 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
EP2321341B1 (en) 2008-07-16 2017-02-22 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
CN103012377A (zh) * 2011-09-27 2013-04-03 江苏艾力斯生物医药有限公司 一种咪唑-5-羧酸酯的重结晶方法
HK1220611A1 (zh) 2013-03-15 2017-05-12 Bausch Health Ireland Limited 用於治疗胃肠道病症的组成物
WO2014151206A1 (en) 2013-03-15 2014-09-25 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase and their uses
SI3004138T1 (sl) 2013-06-05 2024-07-31 Bausch Health Ireland Limited Ultra čisti agonisti gvanilat ciklaze C, postopek za njihovo pripravo in uporabo

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1334092C (en) * 1986-07-11 1995-01-24 David John Carini Angiotensin ii receptor blocking imidazoles
US5064825A (en) * 1989-06-01 1991-11-12 Merck & Co., Inc. Angiotensin ii antagonists
HU215834B (hu) * 1989-06-30 1999-04-28 E. I. Du Pont De Nemours And Co. Eljárás aromás csoporttal szubsztituált imidazolszármazékok, valamint ezeket hatóanyagként tartalmazó gyógyszerkészítmények előállítására
EP0411507B1 (en) * 1989-08-02 1994-10-26 Takeda Chemical Industries, Ltd. Pyrazole derivatives, their production and use
DE4132632A1 (de) * 1991-10-01 1993-04-08 Bayer Ag Substituierte imidazolyl-propensaeurederivate
DE4132631A1 (de) * 1991-10-01 1993-04-08 Bayer Ag Imidazolyl-propensaeurederivate
DE69329982T2 (de) * 1992-06-02 2001-09-27 Sankyo Co., Ltd. 4-Carboxyimidazolderivate als Angiotensin-II-Antagonisten und ihre therapeutische Verwendung

Also Published As

Publication number Publication date
CN1032856C (zh) 1996-09-25
IL103329A0 (en) 1993-03-15
NO923798D0 (no) 1992-09-30
MY108350A (en) 1996-09-30
IL103329A (en) 1996-10-31
FI924353A7 (fi) 1993-04-05
RU2105764C1 (ru) 1998-02-27
ZA927205B (en) 1993-03-23
SI9200240A (en) 1993-06-30
CZ301992A3 (en) 1993-08-11
EP0535420A1 (de) 1993-04-07
YU87592A (sh) 1995-10-03
US5298519A (en) 1994-03-29
AU649357B2 (en) 1994-05-19
NZ244320A (en) 1995-01-27
LV10256A (lv) 1994-10-20
YU48290B (sh) 1998-05-15
SK301992A3 (en) 1995-10-11
JP2544565B2 (ja) 1996-10-16
CN1071426A (zh) 1993-04-28
NO923798L (no) 1993-04-05
FI924353A0 (fi) 1992-09-29
HUT62291A (en) 1993-04-28
AT398202B (de) 1994-10-25
TW223073B (cs) 1994-05-01
HRP920817A2 (en) 1996-08-31
CA2079735A1 (en) 1993-04-05
HU9203149D0 (en) 1992-12-28
AU2617692A (en) 1993-04-08
JPH05310731A (ja) 1993-11-22
LV10256B (en) 1995-04-20
ATA198791A (de) 1994-02-15

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Legal Events

Date Code Title Description
GB Transfer or assigment of application

Owner name: BINDER, DIETER

FD Application lapsed