FI875096A - Foerfarande foer framstaellning av nya substituerade alkandifosfonsyror. - Google Patents

Foerfarande foer framstaellning av nya substituerade alkandifosfonsyror. Download PDF

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Publication number
FI875096A
FI875096A FI875096A FI875096A FI875096A FI 875096 A FI875096 A FI 875096A FI 875096 A FI875096 A FI 875096A FI 875096 A FI875096 A FI 875096A FI 875096 A FI875096 A FI 875096A
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FI
Finland
Prior art keywords
halogen
substituted
phosphono group
atoms
alkandifosfonsyror
Prior art date
Application number
FI875096A
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English (en)
Other versions
FI87570C (fi
FI875096A0 (fi
FI87570B (fi
Inventor
Knut A Jaeggi
Leo Widler
Original Assignee
Ciba Geigy Ag
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Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of FI875096A0 publication Critical patent/FI875096A0/fi
Publication of FI875096A publication Critical patent/FI875096A/fi
Application granted granted Critical
Publication of FI87570B publication Critical patent/FI87570B/fi
Publication of FI87570C publication Critical patent/FI87570C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
    • C07F9/6539—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503—Five-membered rings
    • C07F9/65031—Five-membered rings having the nitrogen atoms in the positions 1 and 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503—Five-membered rings
    • C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
    • C07F9/6518—Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nutrition Science (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Control Of El Displays (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Glass Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI875096A 1986-11-21 1987-11-18 Foerfarande foer framstaellning av nya substituerade alkandifosfonsyror FI87570C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH466686 1986-11-21
CH466686 1986-11-21

Publications (4)

Publication Number Publication Date
FI875096A0 FI875096A0 (fi) 1987-11-18
FI875096A true FI875096A (fi) 1988-05-22
FI87570B FI87570B (fi) 1992-10-15
FI87570C FI87570C (fi) 1993-01-25

Family

ID=4280350

Family Applications (1)

Application Number Title Priority Date Filing Date
FI875096A FI87570C (fi) 1986-11-21 1987-11-18 Foerfarande foer framstaellning av nya substituerade alkandifosfonsyror

Country Status (27)

Country Link
US (1) US4939130A (fi)
EP (1) EP0275821B1 (fi)
JP (1) JP2744238B2 (fi)
KR (1) KR960010752B1 (fi)
AT (1) ATE72816T1 (fi)
AU (1) AU607722B2 (fi)
CA (1) CA1338937C (fi)
CY (1) CY1827A (fi)
DD (1) DD270533A5 (fi)
DE (2) DE3776880D1 (fi)
DK (1) DK174098B1 (fi)
ES (1) ES2038692T4 (fi)
FI (1) FI87570C (fi)
GR (1) GR3003895T3 (fi)
HK (1) HK114894A (fi)
HU (1) HU199150B (fi)
IE (1) IE59816B1 (fi)
IL (1) IL84497A (fi)
LU (1) LU90838I2 (fi)
MX (1) MX9427A (fi)
NL (1) NL300058I2 (fi)
NO (2) NO173446C (fi)
NZ (1) NZ222610A (fi)
PH (1) PH24345A (fi)
PT (1) PT86167B (fi)
SG (1) SG92194G (fi)
ZA (1) ZA878698B (fi)

Families Citing this family (148)

* Cited by examiner, † Cited by third party
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DE3626058A1 (de) * 1986-08-01 1988-02-11 Boehringer Mannheim Gmbh Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
DE3640938A1 (de) * 1986-11-29 1988-06-01 Boehringer Mannheim Gmbh Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindung enthaltende arzneimittel
MX21452A (es) * 1989-07-07 1994-01-31 Ciba Geigy Ag Preparaciones farmaceuticas que se administran en forma topica.
US5139786A (en) * 1989-07-07 1992-08-18 Ciba-Geigy Corporation Topical formulations
JPH06507156A (ja) * 1991-04-27 1994-08-11 日本チバガイギー株式会社 トリアゾール化合物
US5763611A (en) * 1992-05-29 1998-06-09 The Procter & Gamble Company Thio-substituted cyclic phosphonate compounds, pharmaceutical compositions, and methods for treating abnormal calcium and phosphate metabolism
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IL84497A (en) 1994-10-21
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HU199150B (en) 1990-01-29
NO2001015I2 (no) 2004-10-11
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SG92194G (en) 1995-04-28
IE873148L (en) 1988-05-21
IE59816B1 (en) 1994-04-06
CY1827A (en) 1995-12-01
PT86167B (pt) 1990-08-31
FI87570C (fi) 1993-01-25
HK114894A (en) 1994-10-27
PH24345A (en) 1990-06-13
AU8145387A (en) 1988-05-26
LU90838I2 (fr) 2001-11-19
FI875096A0 (fi) 1987-11-18
DK174098B1 (da) 2002-06-17
KR960010752B1 (ko) 1996-08-08
KR880006204A (ko) 1988-07-22
AU607722B2 (en) 1991-03-14
US4939130A (en) 1990-07-03
EP0275821B1 (de) 1992-02-26
ATE72816T1 (de) 1992-03-15
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EP0275821A1 (de) 1988-07-27
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DK609587D0 (da) 1987-11-20
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DE3776880D1 (de) 1992-04-02
NO874856L (no) 1988-05-24
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FI87570B (fi) 1992-10-15
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