FI76790C - Foerfarande foer framstaellning av 2,4-diamino-5-(3',4',5'-trimetoxibensyl)pyrimidin. - Google Patents

Foerfarande foer framstaellning av 2,4-diamino-5-(3',4',5'-trimetoxibensyl)pyrimidin. Download PDF

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Publication number
FI76790C
FI76790C FI822268A FI822268A FI76790C FI 76790 C FI76790 C FI 76790C FI 822268 A FI822268 A FI 822268A FI 822268 A FI822268 A FI 822268A FI 76790 C FI76790 C FI 76790C
Authority
FI
Finland
Prior art keywords
ch3o
general formula
formula
compound
guanidine
Prior art date
Application number
FI822268A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI76790B (fi
FI822268L (fi
FI822268A0 (fi
Inventor
Istvan Simonyi
Ivan Beck
Andras Dietz
Elemer Jakfalvi
Laszlo Ladanyi
Zoltan Takacs
Imre Biro
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of FI822268A0 publication Critical patent/FI822268A0/fi
Publication of FI822268L publication Critical patent/FI822268L/fi
Publication of FI76790B publication Critical patent/FI76790B/fi
Application granted granted Critical
Publication of FI76790C publication Critical patent/FI76790C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FI822268A 1981-06-26 1982-06-24 Foerfarande foer framstaellning av 2,4-diamino-5-(3',4',5'-trimetoxibensyl)pyrimidin. FI76790C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU811869A HU187370B (en) 1981-06-26 1981-06-26 Improved process for producing 2,4-diamino-5-bracket-3-comma above, 4-comma above,5-comma above-trimethoxy-benzyl-bracket closed-pyrimidine
HU186981 1981-06-26

Publications (4)

Publication Number Publication Date
FI822268A0 FI822268A0 (fi) 1982-06-24
FI822268L FI822268L (fi) 1982-12-27
FI76790B FI76790B (fi) 1988-08-31
FI76790C true FI76790C (fi) 1988-12-12

Family

ID=10956594

Family Applications (1)

Application Number Title Priority Date Filing Date
FI822268A FI76790C (fi) 1981-06-26 1982-06-24 Foerfarande foer framstaellning av 2,4-diamino-5-(3',4',5'-trimetoxibensyl)pyrimidin.

Country Status (21)

Country Link
JP (1) JPS5838266A (cs)
AT (1) AT387961B (cs)
AU (1) AU547823B2 (cs)
BE (1) BE893611A (cs)
CA (1) CA1174679A (cs)
CH (1) CH648834A5 (cs)
CS (1) CS244908B2 (cs)
DD (1) DD202703A5 (cs)
DK (1) DK155434C (cs)
ES (1) ES513482A0 (cs)
FI (1) FI76790C (cs)
FR (1) FR2508450B1 (cs)
GB (1) GB2104508B (cs)
GR (1) GR76159B (cs)
HU (1) HU187370B (cs)
IE (1) IE53466B1 (cs)
IL (1) IL66132A (cs)
IT (1) IT1190889B (cs)
SE (1) SE451133B (cs)
SU (1) SU1145929A3 (cs)
YU (1) YU42774B (cs)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2602507B1 (fr) * 1986-08-08 1989-06-09 Sanofi Pharma Procede de preparation de diamino-2,4 benzyl-5 pyrimidines

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB743221A (en) * 1953-05-26 1956-01-11 Wellcome Found Improvements in or relating to the manufacture of acrylonitriles
DE1303727B (de) * 1959-09-03 1976-02-05 Ausscheidung aus: 14 45 176 The Wellcome Foundation Ltd., London Alpha-Arylidensubstituierte Propioni-Irile
NL122146C (cs) * 1960-09-02
US4033962A (en) * 1975-06-26 1977-07-05 Hoffman-La Roche Inc. 2,4-Diamino-pyrimidine derivatives and processes
DE2635765C3 (de) * 1976-08-09 1979-02-08 Ludwig Heumann & Co Gmbh, 8500 Nuernberg Verfahren zur Herstellung von 2,4-EMamino-5-(3',4'r5'-trimethoxybenzyl)-pyrimidin
US4115650A (en) * 1976-11-17 1978-09-19 Hoffmann-La Roche Inc. Process for preparing 2,4-diamino-5-(substituted benzyl)-pyrimidines
DE2730467A1 (de) * 1977-07-06 1979-01-18 Basf Ag Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
IE53466B1 (en) 1988-11-23
IE821520L (en) 1982-12-26
DD202703A5 (de) 1983-09-28
SE8203914L (sv) 1982-12-27
CH648834A5 (de) 1985-04-15
CA1174679A (en) 1984-09-18
SU1145929A3 (ru) 1985-03-15
FI76790B (fi) 1988-08-31
SE8203914D0 (sv) 1982-06-23
ES8304949A1 (es) 1983-04-01
SE451133B (sv) 1987-09-07
GR76159B (cs) 1984-08-03
GB2104508A (en) 1983-03-09
IL66132A0 (en) 1982-09-30
FR2508450A1 (fr) 1982-12-31
ATA244982A (de) 1988-09-15
FR2508450B1 (fr) 1986-01-03
JPS5838266A (ja) 1983-03-05
ES513482A0 (es) 1983-04-01
DK288082A (da) 1982-12-27
AU547823B2 (en) 1985-11-07
HU187370B (en) 1985-12-28
BE893611A (fr) 1982-12-23
GB2104508B (en) 1985-01-16
IT1190889B (it) 1988-02-24
AT387961B (de) 1989-04-10
CS244908B2 (en) 1986-08-14
IL66132A (en) 1985-04-30
DK155434C (da) 1989-09-18
DK155434B (da) 1989-04-10
CS471782A2 (en) 1985-09-17
YU138582A (en) 1984-10-31
AU8534682A (en) 1983-01-06
FI822268L (fi) 1982-12-27
FI822268A0 (fi) 1982-06-24
YU42774B (en) 1988-12-31
IT8222035A0 (it) 1982-06-24

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Owner name: E GY T GYOGYSZERVEGYESZETI GYAR