FI70900C - Foerfarande foer framstaellning av terapeutiskt anvaendbara imdazotia- och imidazooxadiazolalkenkarboxylsyraamider - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara imdazotia- och imidazooxadiazolalkenkarboxylsyraamider Download PDF

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Publication number
FI70900C
FI70900C FI811630A FI811630A FI70900C FI 70900 C FI70900 C FI 70900C FI 811630 A FI811630 A FI 811630A FI 811630 A FI811630 A FI 811630A FI 70900 C FI70900 C FI 70900C
Authority
FI
Finland
Prior art keywords
alkyl
general formula
methyl
phenyl
hydroxyalkyl
Prior art date
Application number
FI811630A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI70900B (fi
FI811630L (fi
Inventor
Horst Meyer
Harald Horstmann
Eike Moeller
Bernward Garthoff
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19803020421 external-priority patent/DE3020421A1/de
Priority claimed from DE19803043158 external-priority patent/DE3043158A1/de
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of FI811630L publication Critical patent/FI811630L/fi
Priority to FI831950A priority Critical patent/FI71745C/fi
Publication of FI70900B publication Critical patent/FI70900B/fi
Application granted granted Critical
Publication of FI70900C publication Critical patent/FI70900C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
FI811630A 1980-05-29 1981-05-27 Foerfarande foer framstaellning av terapeutiskt anvaendbara imdazotia- och imidazooxadiazolalkenkarboxylsyraamider FI70900C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI831950A FI71745C (fi) 1980-05-29 1983-05-31 Foerfarande foer framstaellning av -(imidazo-/2,1-b/-1,3,4-tiadiazol-5-yl)-alkenkarboxylsyror, vilka aer mellanprodukter vid framstaellning av diuretiska imidazotiadiazolalken- karboxylsyraaminer.

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3020421 1980-05-29
DE19803020421 DE3020421A1 (de) 1980-05-29 1980-05-29 Imidazoazolalkensaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE19803043158 DE3043158A1 (de) 1980-11-15 1980-11-15 Imidazoazolalkensaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE3043158 1980-11-15

Publications (3)

Publication Number Publication Date
FI811630L FI811630L (fi) 1981-11-30
FI70900B FI70900B (fi) 1986-07-18
FI70900C true FI70900C (fi) 1986-10-27

Family

ID=25785736

Family Applications (1)

Application Number Title Priority Date Filing Date
FI811630A FI70900C (fi) 1980-05-29 1981-05-27 Foerfarande foer framstaellning av terapeutiskt anvaendbara imdazotia- och imidazooxadiazolalkenkarboxylsyraamider

Country Status (13)

Country Link
US (1) US4444770A (hu)
EP (1) EP0041215B1 (hu)
AU (1) AU543307B2 (hu)
CA (1) CA1188690A (hu)
DE (1) DE3173607D1 (hu)
DK (1) DK233281A (hu)
ES (1) ES8203897A1 (hu)
FI (1) FI70900C (hu)
GR (1) GR74557B (hu)
HU (1) HU186887B (hu)
IL (1) IL62960A (hu)
NO (2) NO811630L (hu)
PT (1) PT73058B (hu)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3208437A1 (de) * 1982-03-09 1983-09-15 Bayer Ag, 5090 Leverkusen Imidazothiadiazolalkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE3329621A1 (de) * 1983-08-17 1985-02-28 Bayer Ag, 5090 Leverkusen Aminoalkyl-imidazothiadiazol-alkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
IT1213175B (it) * 1984-06-06 1989-12-14 Mediolanum Farmaceutici Srl Derivati imidazotiazolmetilen-acetidrazidi, loro preparazione e composizioni farmaceutiche ad attivita'diuretica.
DE3542662A1 (de) * 1985-12-03 1987-06-04 Bayer Ag Imidazothiadiazinalkensaeureamide, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung und ihre verwendung zur behandlung von krankheiten
DE3542661A1 (de) * 1985-12-03 1987-06-04 Bayer Ag Imidazopyridazinalkensaeureamide, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung
TW438796B (en) * 1996-05-15 2001-06-07 Hoffmann La Roche 2,4-diaminopyrimidine derivatives, the manufacture process thereof, and the antibiotically-active pharmaceutical composition containing the same
US20060135571A1 (en) * 2003-06-13 2006-06-22 Jaquith James B Imidazo(2,1-b)-1,3,4-thiadiazole sulfoxides and sulfones
DE102005010215A1 (de) * 2005-03-05 2006-09-07 Bayer Cropscience Ag Heterobicyclische Acrylamide
JP5410431B2 (ja) 2007-09-27 2014-02-05 セントロ ナシオナル デ インベスティガシオネス オンコロヒカス（セエネイオ） イミダゾロチアジアゾール類のプロテインキナーゼ阻害剤としての使用
US8318928B2 (en) * 2008-12-15 2012-11-27 Glenmark Pharmaceuticals, S.A. Fused imidazole carboxamides as TRPV3 modulators
HUE027964T2 (hu) 2009-04-02 2016-11-28 Fund Centro Nac De Investig Oncologicas Carlos Iii Imidazol[2,1-B][1,3,4]tiadiazol-származékok
EP2488533B1 (en) * 2009-10-13 2014-07-23 Council of Scientific & Industrial Research Imidazothiazole-chalcone derivatives as potential anticancer agents and process for the preparation thereof
BR112012011528A2 (pt) 2009-11-16 2019-09-24 Univ California métodos para inibir uma proteína quinase e para tratar uma doença associada com atividade de quinase, e, composto
EP2847200B1 (en) 2012-04-26 2017-03-29 Bristol-Myers Squibb Company Imidazothiadiazole derivatives as protease activated receptor 4 (par4) inhibitors for treating platelet aggregation
EP2855489B1 (en) 2012-04-26 2017-01-04 Bristol-Myers Squibb Company Imidazothiadiazole and imidazopyridazine derivatives as protease activated receptor 4 (par4) inhibitors for treating platelet aggregation
PL2841437T3 (pl) 2012-04-26 2017-12-29 Bristol-Myers Squibb Company Pochodne imidazotiadiazolu i imidazopirazyny jako inhibitory receptora 4 (par4) aktywowanego proteazą do leczenia agregacji płytek
EA039493B1 (ru) 2016-06-29 2022-02-02 Университе Де Монреаль Биарилметильные гетероциклы
WO2021078120A1 (en) 2019-10-21 2021-04-29 Novartis Ag Compounds and compositions for the treatment of parasitic diseases

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3615639A (en) * 1967-10-23 1971-10-26 Eastman Kodak Co Direct positive silver halide emulsions containing dyes as electron acceptors and spectral sensitizers
US3804823A (en) * 1972-02-15 1974-04-16 Eastman Kodak Co Heterocyclic containing monoazo compounds
US4042583A (en) * 1973-09-20 1977-08-16 Pfizer Inc. Imidazo[2,1-b]thiazole and thiazolo[3,2-a]-benzimidazole quaternary salts as hypoglycemic agents and growth promotants
OA04806A (fr) * 1973-12-10 1980-08-31 Bayer Ag Nouveaux esters triazolothiazolyliques d'acide (thiono)-phosphorique (phosphonique), leur procédé de préparation et leur application comme insecticides et acaricides.
AT340414B (de) * 1975-02-18 1977-12-12 Plantex Ltd Verfahren zur herstellung von neuen imidazo(2,1-b)thiazolderivaten und ihren salzen
US4263311A (en) * 1976-09-27 1981-04-21 Smithkline Corporation 5,6-Phenyl-2,3-dihydroimidazo [2,1-b] thiazoles
DE2823686A1 (de) * 1978-05-31 1979-12-06 Bayer Ag Imidazo eckige klammer auf 2.1-b eckige klammer zu eckige klammer auf 1.3.4 eckige klammer zu -thiadiazole
DE2902763A1 (de) * 1979-01-25 1980-08-07 Basf Ag Basische farbstoffe

Also Published As

Publication number Publication date
NO811630L (no) 1981-11-30
PT73058A (en) 1981-06-01
US4444770A (en) 1984-04-24
AU7090081A (en) 1981-12-03
ES502573A0 (es) 1982-04-01
PT73058B (en) 1982-07-01
IL62960A0 (en) 1981-07-31
FI70900B (fi) 1986-07-18
EP0041215A3 (en) 1982-04-14
HU186887B (en) 1985-10-28
EP0041215B1 (de) 1986-01-29
GR74557B (hu) 1984-06-29
IL62960A (en) 1986-04-29
ES8203897A1 (es) 1982-04-01
EP0041215A2 (de) 1981-12-09
FI811630L (fi) 1981-11-30
AU543307B2 (en) 1985-04-18
DK233281A (da) 1981-11-30
CA1188690A (en) 1985-06-11
DE3173607D1 (en) 1986-03-13
NO854688L (no) 1981-11-30

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Owner name: BAYER AKTIENGESELLSCHAFT