ES8203897A1 - Procedimiento para la obtencion de imidazoazoalquenamidas - Google Patents

Procedimiento para la obtencion de imidazoazoalquenamidas

Info

Publication number
ES8203897A1
ES8203897A1 ES502573A ES502573A ES8203897A1 ES 8203897 A1 ES8203897 A1 ES 8203897A1 ES 502573 A ES502573 A ES 502573A ES 502573 A ES502573 A ES 502573A ES 8203897 A1 ES8203897 A1 ES 8203897A1
Authority
ES
Spain
Prior art keywords
preparation
imidazoazolalkenyl
carboxamides
medicaments
intermediates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES502573A
Other languages
English (en)
Other versions
ES502573A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19803020421 external-priority patent/DE3020421A1/de
Priority claimed from DE19803043158 external-priority patent/DE3043158A1/de
Application filed by Bayer AG filed Critical Bayer AG
Publication of ES502573A0 publication Critical patent/ES502573A0/es
Publication of ES8203897A1 publication Critical patent/ES8203897A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE IMIDAZOAZOALQUENAMIDAS. CONSITE EN HACER REACCIONAR COMPUESTOS DE FORMULA GENERAL (I) CON DERIVADOS DE FOSFONATO (II) EN PRESENCIA DE BASES FUERTES Y DISOLVENTES ORGANICOS INERTES A TEMPERATURAS COMPRENDIDAS ENTRE -20 Y 40 GRADOS C. OPCIONALMENTE, SE PUEDE HACER REACCIONAR COMPUESTOS DE CARBONILO CON DERIVADOS DE ACETAMIDA EN PRESENCIA DE CATALIZADORES Y, EN CASO DADO, DE DISOLVENTES ORGANICOS INERTES A TEMPERATURAS DE 20 A 200 GRADOS C, O SE HACE REACCIONAR ACIDOS ALQUENICOS CON AMIDAS EN PRESENCIA DE DISOLVENTE ORGANICOS INERTES A TEMPERATURA DE 20 Y 150 GRADOS C.
ES502573A 1980-05-29 1981-05-28 Procedimiento para la obtencion de imidazoazoalquenamidas Expired ES8203897A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19803020421 DE3020421A1 (de) 1980-05-29 1980-05-29 Imidazoazolalkensaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE19803043158 DE3043158A1 (de) 1980-11-15 1980-11-15 Imidazoazolalkensaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln

Publications (2)

Publication Number Publication Date
ES502573A0 ES502573A0 (es) 1982-04-01
ES8203897A1 true ES8203897A1 (es) 1982-04-01

Family

ID=25785736

Family Applications (1)

Application Number Title Priority Date Filing Date
ES502573A Expired ES8203897A1 (es) 1980-05-29 1981-05-28 Procedimiento para la obtencion de imidazoazoalquenamidas

Country Status (13)

Country Link
US (1) US4444770A (es)
EP (1) EP0041215B1 (es)
AU (1) AU543307B2 (es)
CA (1) CA1188690A (es)
DE (1) DE3173607D1 (es)
DK (1) DK233281A (es)
ES (1) ES8203897A1 (es)
FI (1) FI70900C (es)
GR (1) GR74557B (es)
HU (1) HU186887B (es)
IL (1) IL62960A (es)
NO (2) NO811630L (es)
PT (1) PT73058B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3208437A1 (de) * 1982-03-09 1983-09-15 Bayer Ag, 5090 Leverkusen Imidazothiadiazolalkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE3329621A1 (de) * 1983-08-17 1985-02-28 Bayer Ag, 5090 Leverkusen Aminoalkyl-imidazothiadiazol-alkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
IT1213175B (it) * 1984-06-06 1989-12-14 Mediolanum Farmaceutici Srl Derivati imidazotiazolmetilen-acetidrazidi, loro preparazione e composizioni farmaceutiche ad attivita'diuretica.
DE3542661A1 (de) * 1985-12-03 1987-06-04 Bayer Ag Imidazopyridazinalkensaeureamide, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung
DE3542662A1 (de) * 1985-12-03 1987-06-04 Bayer Ag Imidazothiadiazinalkensaeureamide, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung und ihre verwendung zur behandlung von krankheiten
TW438796B (en) * 1996-05-15 2001-06-07 Hoffmann La Roche 2,4-diaminopyrimidine derivatives, the manufacture process thereof, and the antibiotically-active pharmaceutical composition containing the same
US20060135571A1 (en) * 2003-06-13 2006-06-22 Jaquith James B Imidazo(2,1-b)-1,3,4-thiadiazole sulfoxides and sulfones
DE102005010215A1 (de) * 2005-03-05 2006-09-07 Bayer Cropscience Ag Heterobicyclische Acrylamide
CN101878219B (zh) 2007-09-27 2014-04-02 西班牙国家癌症研究中心 用于作为蛋白激酶抑制剂使用的咪唑并噻二唑类
US8318928B2 (en) * 2008-12-15 2012-11-27 Glenmark Pharmaceuticals, S.A. Fused imidazole carboxamides as TRPV3 modulators
EP2414369B1 (en) 2009-04-02 2015-08-12 Fundación Centro Nacional de Investigaciones Oncológicas Carlos III Imidazo[2,1-b][1,3,4]thiadiazole derivatives
EP2488533B1 (en) * 2009-10-13 2014-07-23 Council of Scientific & Industrial Research Imidazothiazole-chalcone derivatives as potential anticancer agents and process for the preparation thereof
US20130035325A1 (en) * 2009-11-16 2013-02-07 The Regents Of The University Of California Kinase inhibitors
JP6101343B2 (ja) 2012-04-26 2017-03-22 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 血小板凝集を治療するためのプロテアーゼ活性化受容体4(par4)阻害剤としてのイミダゾチアジアゾールおよびイミダゾピリダジン誘導体
KR20200127273A (ko) 2012-04-26 2020-11-10 브리스톨-마이어스 스큅 컴퍼니 혈소판 응집을 치료하기 위한 프로테아제 활성화 수용체 4 (par4) 억제제로서의 이미다조티아디아졸 및 이미다조피라진 유도체
CA2871637A1 (en) 2012-04-26 2013-10-31 Bristol-Myers Squibb Company Imidazothiadiazole derivatives as protease activated receptor 4 (par4) inhibitors for treating platelet aggregation
WO2018005591A1 (en) 2016-06-29 2018-01-04 Universite De Montreal Biarylmethyl heterocycles
CA3158333A1 (en) 2019-10-21 2021-04-29 Novartis Ag Compounds and compositions for the treatment of parasitic diseases

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3615639A (en) * 1967-10-23 1971-10-26 Eastman Kodak Co Direct positive silver halide emulsions containing dyes as electron acceptors and spectral sensitizers
US3804823A (en) * 1972-02-15 1974-04-16 Eastman Kodak Co Heterocyclic containing monoazo compounds
US4042583A (en) * 1973-09-20 1977-08-16 Pfizer Inc. Imidazo[2,1-b]thiazole and thiazolo[3,2-a]-benzimidazole quaternary salts as hypoglycemic agents and growth promotants
OA04806A (fr) * 1973-12-10 1980-08-31 Bayer Ag Nouveaux esters triazolothiazolyliques d'acide (thiono)-phosphorique (phosphonique), leur procédé de préparation et leur application comme insecticides et acaricides.
AT340414B (de) * 1975-02-18 1977-12-12 Plantex Ltd Verfahren zur herstellung von neuen imidazo(2,1-b)thiazolderivaten und ihren salzen
US4263311A (en) * 1976-09-27 1981-04-21 Smithkline Corporation 5,6-Phenyl-2,3-dihydroimidazo [2,1-b] thiazoles
DE2823686A1 (de) * 1978-05-31 1979-12-06 Bayer Ag Imidazo eckige klammer auf 2.1-b eckige klammer zu eckige klammer auf 1.3.4 eckige klammer zu -thiadiazole
DE2902763A1 (de) * 1979-01-25 1980-08-07 Basf Ag Basische farbstoffe

Also Published As

Publication number Publication date
IL62960A0 (en) 1981-07-31
ES502573A0 (es) 1982-04-01
NO811630L (no) 1981-11-30
FI811630L (fi) 1981-11-30
HU186887B (en) 1985-10-28
DE3173607D1 (en) 1986-03-13
US4444770A (en) 1984-04-24
PT73058B (en) 1982-07-01
IL62960A (en) 1986-04-29
EP0041215A3 (en) 1982-04-14
CA1188690A (en) 1985-06-11
DK233281A (da) 1981-11-30
EP0041215A2 (de) 1981-12-09
AU7090081A (en) 1981-12-03
EP0041215B1 (de) 1986-01-29
PT73058A (en) 1981-06-01
GR74557B (es) 1984-06-29
FI70900B (fi) 1986-07-18
AU543307B2 (en) 1985-04-18
NO854688L (no) 1981-11-30
FI70900C (fi) 1986-10-27

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