FI811630L - Imidazoazolalkensyraamider nya mellanprodukter foer deras framstaellning samt framstaellning och anvaendning av dem i laekemedel - Google Patents

Imidazoazolalkensyraamider nya mellanprodukter foer deras framstaellning samt framstaellning och anvaendning av dem i laekemedel

Info

Publication number
FI811630L
FI811630L FI811630A FI811630A FI811630L FI 811630 L FI811630 L FI 811630L FI 811630 A FI811630 A FI 811630A FI 811630 A FI811630 A FI 811630A FI 811630 L FI811630 L FI 811630L
Authority
FI
Finland
Prior art keywords
framstaellning
imidazoazolalkensyraamider
laekemedel
dem
samt
Prior art date
Application number
FI811630A
Other languages
English (en)
Other versions
FI70900C (fi
FI70900B (fi
Inventor
Horst Meyer
Harald Horstmann
Eike Moeller
Bernward Garthoff
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19803020421 external-priority patent/DE3020421A1/de
Priority claimed from DE19803043158 external-priority patent/DE3043158A1/de
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of FI811630L publication Critical patent/FI811630L/fi
Priority to FI831950A priority Critical patent/FI71745C/fi
Application granted granted Critical
Publication of FI70900B publication Critical patent/FI70900B/fi
Publication of FI70900C publication Critical patent/FI70900C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
FI811630A 1980-05-29 1981-05-27 Foerfarande foer framstaellning av terapeutiskt anvaendbara imdazotia- och imidazooxadiazolalkenkarboxylsyraamider FI70900C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI831950A FI71745C (fi) 1980-05-29 1983-05-31 Foerfarande foer framstaellning av -(imidazo-/2,1-b/-1,3,4-tiadiazol-5-yl)-alkenkarboxylsyror, vilka aer mellanprodukter vid framstaellning av diuretiska imidazotiadiazolalken- karboxylsyraaminer.

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3020421 1980-05-29
DE19803020421 DE3020421A1 (de) 1980-05-29 1980-05-29 Imidazoazolalkensaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE3043158 1980-11-15
DE19803043158 DE3043158A1 (de) 1980-11-15 1980-11-15 Imidazoazolalkensaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln

Publications (3)

Publication Number Publication Date
FI811630L true FI811630L (fi) 1981-11-30
FI70900B FI70900B (fi) 1986-07-18
FI70900C FI70900C (fi) 1986-10-27

Family

ID=25785736

Family Applications (1)

Application Number Title Priority Date Filing Date
FI811630A FI70900C (fi) 1980-05-29 1981-05-27 Foerfarande foer framstaellning av terapeutiskt anvaendbara imdazotia- och imidazooxadiazolalkenkarboxylsyraamider

Country Status (13)

Country Link
US (1) US4444770A (fi)
EP (1) EP0041215B1 (fi)
AU (1) AU543307B2 (fi)
CA (1) CA1188690A (fi)
DE (1) DE3173607D1 (fi)
DK (1) DK233281A (fi)
ES (1) ES8203897A1 (fi)
FI (1) FI70900C (fi)
GR (1) GR74557B (fi)
HU (1) HU186887B (fi)
IL (1) IL62960A (fi)
NO (2) NO811630L (fi)
PT (1) PT73058B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3208437A1 (de) * 1982-03-09 1983-09-15 Bayer Ag, 5090 Leverkusen Imidazothiadiazolalkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
DE3329621A1 (de) * 1983-08-17 1985-02-28 Bayer Ag, 5090 Leverkusen Aminoalkyl-imidazothiadiazol-alkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln
IT1213175B (it) * 1984-06-06 1989-12-14 Mediolanum Farmaceutici Srl Derivati imidazotiazolmetilen-acetidrazidi, loro preparazione e composizioni farmaceutiche ad attivita'diuretica.
DE3542661A1 (de) * 1985-12-03 1987-06-04 Bayer Ag Imidazopyridazinalkensaeureamide, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung
DE3542662A1 (de) * 1985-12-03 1987-06-04 Bayer Ag Imidazothiadiazinalkensaeureamide, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung und ihre verwendung zur behandlung von krankheiten
TW438796B (en) * 1996-05-15 2001-06-07 Hoffmann La Roche 2,4-diaminopyrimidine derivatives, the manufacture process thereof, and the antibiotically-active pharmaceutical composition containing the same
WO2004111060A1 (en) * 2003-06-13 2004-12-23 Aegera Therapeutics Inc. IMIDAZO[2,1-b]-1,3,4-THIADIAZOLE SULFOXIDES AND SULFONES
DE102005010215A1 (de) * 2005-03-05 2006-09-07 Bayer Cropscience Ag Heterobicyclische Acrylamide
CN101878219B (zh) 2007-09-27 2014-04-02 西班牙国家癌症研究中心 用于作为蛋白激酶抑制剂使用的咪唑并噻二唑类
US8318928B2 (en) * 2008-12-15 2012-11-27 Glenmark Pharmaceuticals, S.A. Fused imidazole carboxamides as TRPV3 modulators
NZ595674A (en) 2009-04-02 2012-12-21 Ct Nac Investigaciones Oncologicas Cnio Imidazo[2,1-b][1,3,4]thiadiazole derivatives
US8916711B2 (en) * 2009-10-13 2014-12-23 Council Of Scientific And Industrial Research Imidazothiazole-chalcone derivatives as potential anticancer agents and process for the preparation thereof
US20130035325A1 (en) * 2009-11-16 2013-02-07 The Regents Of The University Of California Kinase inhibitors
MX2014012741A (es) 2012-04-26 2015-04-13 Bristol Myers Squibb Co Derivados de imidazotiadiazol e imidazopirazina como inhibidores del receptor 4 activado de proteasa (par4) para tratamiento de agregacion plaquetaria.
DK3243826T3 (da) 2012-04-26 2020-02-03 Bristol Myers Squibb Co Imidazothiadiazol-og imidazopyrazinderivater som proteaseaktiverede receptor 4- (par4) hæmmere til behandling af blodpladeaggregation
EA201491967A1 (ru) 2012-04-26 2015-03-31 Бристол-Майерс Сквибб Компани Производные имидазотиадиазола в качестве ингибиторов активируемых протеазой рецепторов 4 (par4) для лечения агрегации тромбоцитов
EA039493B1 (ru) 2016-06-29 2022-02-02 Университе Де Монреаль Биарилметильные гетероциклы
KR20220086619A (ko) 2019-10-21 2022-06-23 노파르티스 아게 기생충 질환 치료용 화합물 및 조성물

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3615639A (en) * 1967-10-23 1971-10-26 Eastman Kodak Co Direct positive silver halide emulsions containing dyes as electron acceptors and spectral sensitizers
US3804823A (en) * 1972-02-15 1974-04-16 Eastman Kodak Co Heterocyclic containing monoazo compounds
US4042583A (en) * 1973-09-20 1977-08-16 Pfizer Inc. Imidazo[2,1-b]thiazole and thiazolo[3,2-a]-benzimidazole quaternary salts as hypoglycemic agents and growth promotants
OA04806A (fr) * 1973-12-10 1980-08-31 Bayer Ag Nouveaux esters triazolothiazolyliques d'acide (thiono)-phosphorique (phosphonique), leur procédé de préparation et leur application comme insecticides et acaricides.
AT340414B (de) * 1975-02-18 1977-12-12 Plantex Ltd Verfahren zur herstellung von neuen imidazo(2,1-b)thiazolderivaten und ihren salzen
US4263311A (en) * 1976-09-27 1981-04-21 Smithkline Corporation 5,6-Phenyl-2,3-dihydroimidazo [2,1-b] thiazoles
DE2823686A1 (de) * 1978-05-31 1979-12-06 Bayer Ag Imidazo eckige klammer auf 2.1-b eckige klammer zu eckige klammer auf 1.3.4 eckige klammer zu -thiadiazole
DE2902763A1 (de) * 1979-01-25 1980-08-07 Basf Ag Basische farbstoffe

Also Published As

Publication number Publication date
PT73058A (en) 1981-06-01
AU7090081A (en) 1981-12-03
DE3173607D1 (en) 1986-03-13
CA1188690A (en) 1985-06-11
NO811630L (no) 1981-11-30
EP0041215A2 (de) 1981-12-09
NO854688L (no) 1981-11-30
EP0041215A3 (en) 1982-04-14
US4444770A (en) 1984-04-24
GR74557B (fi) 1984-06-29
AU543307B2 (en) 1985-04-18
ES502573A0 (es) 1982-04-01
DK233281A (da) 1981-11-30
EP0041215B1 (de) 1986-01-29
PT73058B (en) 1982-07-01
IL62960A0 (en) 1981-07-31
IL62960A (en) 1986-04-29
ES8203897A1 (es) 1982-04-01
FI70900C (fi) 1986-10-27
HU186887B (en) 1985-10-28
FI70900B (fi) 1986-07-18

Similar Documents

Publication Publication Date Title
FI810948L (fi) Nytt foerfarande foer framstaellning av kefalosporinantibiotika och i detta foerfarande anvaendbara nya mellanprodukter och framstaellning av dem
FI904527A0 (fi) Formkropp och kompositmaterial samt foerfarande foer framstaellning av formkroppen.
FI812980L (fi) Nya kefalosporiner foerfarande foer framstaellning av dessa mellanprodukter daerav samt foerfarande foer framstaellning av mellanprodukter
FI810058L (fi) Nya dipyridamol-retardationsformer och foerfarande foer deras framstaellning
FI814103L (fi) Foerfarande foer framstaellning av fiber- samt granulatmaterial anordning foer genomfoerande av foerfarandet foerfarande foer anvaendning av anordningen samt anvaendningen av fiber- samt granulatmaterialet
FI813971L (fi) Nya pyrimidoner deras framstaellning och deras anvaendning saosom laekemedel
FI811630L (fi) Imidazoazolalkensyraamider nya mellanprodukter foer deras framstaellning samt framstaellning och anvaendning av dem i laekemedel
FI811323L (fi) Foerfarande och anordning foer returnering av koepvagnar i en butik
FI813794L (fi) Nya imidazolylfenylaminer deras framstaellningsfoerfarande ochderas farmaceutiskt anvaendning samt mellanprodukter av f rastaellning
FI811540L (fi) Foerfarande foer styrning av linjetryckets foerdelning i en valsanordning och motsvarande valsanordning
FI810315L (fi) Foerfarande foer inmatning av virkesbitar i en virkesbearbetningsmaskin och anordning foer genomfoerande av foerfarandet
FI813934L (fi) Nya fenylalkylaminer deras framstaellning och deras anvaendning saosom laekemedel
FI811059L (fi) Foerfarande foer framstaellning av nya tricykliska etrar
FI811703L (fi) Nya kinoxalin-2-yl-etenylketoner och foerfarande foer deras framstaellning
FI822786L (fi) Foerfarande foer aotervinning av aedelmetaller och elektrolysanordning foer anvaendning i foerfaran
FI812969L (fi) Foerfarande foer montering och demontering av bjaelklagsformer vid betoneringsarbeten samt bjaelklagsform foer genomfoerande av foerfarandet
FI813561L (fi) Nya indolinoner deras framstaellning och deras anvaendning saosom laekemedel
FI810633L (fi) Nya kopplingsfaergkomponenter foer oxidationshaorfaerger deras framstaellning och haorfaergningspreparat innehaollande dem
FI820482L (fi) Isoleringspanel foer bruk i yttertak och vaeggar i byggnader samt yttertak och vaeggar innehaollande isoleringspanelerna
FI820957L (fi) Foerfarande foer tillvaratagande av monosackarider samt och anlaeggning foer genomfoerande av foerfarandet
FI812329L (fi) Foerfarande foer avlaegsnande av ytdefekter samt foer utfoerande av foerfarandet avsedd flerdelad braennare
FI811862L (fi) Foerfarande foer omformning av signalavsnitt foer kodad oeverfoering uppdelade talsignaler samt anordning foer genomfoerande av foerfarandet
FI810120L (fi) Nya tioler och foerfarande foer deras framstaellning
FI813441L (fi) Foerfarande foer framstaellning av polyolblandningar och nya polyolblandningar
FI802819A (fi) Sulfonerad lignindispergeringsmedel och faergaemne innehaollande detsamma samt foerfarande foer anvaendning daerav

Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: BAYER AKTIENGESELLSCHAFT