FI58129C - Foerfarande foer framstaellning av terapeutiskt anvaendbara tieno(3,2-f)-s-triazolo(4,3-a)(1,4)diazepinderivat - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara tieno(3,2-f)-s-triazolo(4,3-a)(1,4)diazepinderivat Download PDF

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Publication number
FI58129C
FI58129C FI357/74A FI35774A FI58129C FI 58129 C FI58129 C FI 58129C FI 357/74 A FI357/74 A FI 357/74A FI 35774 A FI35774 A FI 35774A FI 58129 C FI58129 C FI 58129C
Authority
FI
Finland
Prior art keywords
formula
compound
alkyl
chlorophenyl
thieno
Prior art date
Application number
FI357/74A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI58129B (fi
Inventor
Joseph Hellerbach
Paul Zeller
Dieter Binder
Otto Hromatka
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of FI58129B publication Critical patent/FI58129B/fi
Publication of FI58129C publication Critical patent/FI58129C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
FI357/74A 1973-02-08 1974-02-08 Foerfarande foer framstaellning av terapeutiskt anvaendbara tieno(3,2-f)-s-triazolo(4,3-a)(1,4)diazepinderivat FI58129C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH179973A CH584223A5 (da) 1973-02-08 1973-02-08
CH179973 1973-02-08

Publications (2)

Publication Number Publication Date
FI58129B FI58129B (fi) 1980-08-29
FI58129C true FI58129C (fi) 1980-12-10

Family

ID=4218866

Family Applications (1)

Application Number Title Priority Date Filing Date
FI357/74A FI58129C (fi) 1973-02-08 1974-02-08 Foerfarande foer framstaellning av terapeutiskt anvaendbara tieno(3,2-f)-s-triazolo(4,3-a)(1,4)diazepinderivat

Country Status (24)

Country Link
JP (1) JPS5833234B2 (da)
AR (2) AR203188A1 (da)
AT (1) AT343118B (da)
BE (1) BE810705A (da)
CA (1) CA1049009A (da)
CH (1) CH584223A5 (da)
DD (1) DD112454A5 (da)
DE (1) DE2405682C3 (da)
DK (1) DK137679B (da)
FI (1) FI58129C (da)
FR (1) FR2217007B1 (da)
GB (2) GB1456161A (da)
HU (2) HU170423B (da)
IE (1) IE38883B1 (da)
IL (1) IL44095A (da)
LU (1) LU69338A1 (da)
NL (1) NL174045C (da)
NO (1) NO142260C (da)
PH (1) PH12303A (da)
PL (3) PL97304B1 (da)
SE (1) SE416399B (da)
SU (3) SU715028A3 (da)
YU (1) YU39716B (da)
ZA (1) ZA74472B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT338799B (de) * 1974-03-02 1977-09-12 Boehringer Sohn Ingelheim Verfahren zur herstellung neuer substituierter 6-aryl-4h-s-triazolo-(3,4c)-thieno-(2,3e)-1,4-diazepine und ihrer salze
DE2533924C3 (de) * 1975-07-30 1979-05-03 C.H. Boehringer Sohn, 6507 Ingelheim Verfahren zur Herstellung von 6- Aryl-4H-striazolo [3,4-c] thieno [2,3-e] 1,4-diazepinen
DE2531678C3 (de) * 1975-07-16 1979-06-28 C.H. Boehringer Sohn, 6507 Ingelheim Thieno [2,3e] triazole [3,4c] 5,6-dihydro-l,4diazepine und Verfahren zu ihrer Herstellung
DE2708121A1 (de) * 1977-02-25 1978-09-07 Boehringer Sohn Ingelheim Triazolo-thieno-diazepin-l-one, verfahren zu ihrer herstellung und arzneimittel
FI63033C (fi) * 1977-07-21 1983-04-11 Boehringer Sohn Ingelheim Foerfarande foer framstaellning av anxiolytiska tranquilliserande sedativa och/eller neuroleptiska substituerade 1-piperazinyl-4h-s-triazolo(3,4-c)tieno(2,3-e)-1,4-diazepiner
DE3502392A1 (de) * 1985-01-25 1986-07-31 Boehringer Ingelheim KG, 6507 Ingelheim Neue thieno-triazolo-1,4-diazepino-2- carbonsaeureamide, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen
DE3778559D1 (de) * 1986-01-21 1992-06-04 Boehringer Ingelheim Kg Thieno-1,4-diazepine.
JP2582225B2 (ja) * 1994-04-15 1997-02-19 ナショナル住宅産業株式会社 建 具
WO1995032963A1 (fr) * 1994-06-01 1995-12-07 Yoshitomi Pharmaceutical Industries, Ltd. Compose de thienylazole et compose de thienotriazolodiazepine
CN1101680C (zh) * 1995-09-09 2003-02-19 弗·哈夫曼-拉罗切有限公司 噻吩并三唑并二氮杂䓬增加载脂蛋白a-1含量的用途

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904641A (en) * 1971-06-18 1975-09-09 Yoshitomi Pharmaceutical Triazolothienodiazepine compounds

Also Published As

Publication number Publication date
PL97275B1 (pl) 1978-02-28
BE810705A (fr) 1974-08-07
PL97304B1 (pl) 1978-02-28
DK137679C (da) 1978-09-25
AR203188A1 (es) 1975-08-22
SE416399B (sv) 1980-12-22
AR217034A1 (es) 1980-02-29
GB1456162A (en) 1976-11-17
IL44095A0 (en) 1974-05-16
NL7401117A (da) 1974-08-12
YU39716B (en) 1985-04-30
NO142260C (no) 1980-07-23
FR2217007A1 (da) 1974-09-06
NL174045B (nl) 1983-11-16
ZA74472B (en) 1974-11-27
GB1456161A (en) 1976-11-17
CA1049009A (en) 1979-02-20
DE2405682B2 (de) 1980-07-17
PH12303A (en) 1979-01-16
DE2405682C3 (de) 1981-03-12
HU173741B (hu) 1979-08-28
YU22874A (en) 1982-06-30
FR2217007B1 (da) 1978-02-03
DD112454A5 (da) 1975-04-12
DK137679B (da) 1978-04-17
ATA96474A (de) 1977-09-15
LU69338A1 (da) 1975-12-09
JPS49102698A (da) 1974-09-27
AU6485574A (en) 1975-07-24
SU747429A4 (ru) 1980-07-23
PL96107B1 (pl) 1977-12-31
IE38883B1 (en) 1978-06-21
DE2405682A1 (de) 1974-08-15
FI58129B (fi) 1980-08-29
JPS5833234B2 (ja) 1983-07-18
SU715028A3 (ru) 1980-02-05
HU170423B (da) 1977-06-28
NL174045C (nl) 1984-04-16
CH584223A5 (da) 1977-01-31
NO740405L (no) 1974-08-09
NO142260B (no) 1980-04-14
SU1060115A3 (ru) 1983-12-07
AT343118B (de) 1978-05-10
IE38883L (en) 1974-08-08
IL44095A (en) 1979-03-12

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