FI114709B - Menetelmä farmakologisesti aktiivisen N-t-butyyli-androst-3,5-dieeni-17b-karboksamidi-3-karboksyylihapon polymorfin A valmistamiseksi - Google Patents

Menetelmä farmakologisesti aktiivisen N-t-butyyli-androst-3,5-dieeni-17b-karboksamidi-3-karboksyylihapon polymorfin A valmistamiseksi Download PDF

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Publication number
FI114709B
FI114709B FI944414A FI944414A FI114709B FI 114709 B FI114709 B FI 114709B FI 944414 A FI944414 A FI 944414A FI 944414 A FI944414 A FI 944414A FI 114709 B FI114709 B FI 114709B
Authority
FI
Finland
Prior art keywords
polymorph
carboxamide
diene
butyl
carboxylic acid
Prior art date
Application number
FI944414A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI944414A (fi
FI944414A0 (fi
Inventor
Neil Howard Baine
Neville Lewis Holder
Donald Nathaniel Klein
Robert Lee Webb
Gary Edward Zuber
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of FI944414A publication Critical patent/FI944414A/fi
Publication of FI944414A0 publication Critical patent/FI944414A0/fi
Application granted granted Critical
Publication of FI114709B publication Critical patent/FI114709B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI944414A 1992-03-24 1994-09-23 Menetelmä farmakologisesti aktiivisen N-t-butyyli-androst-3,5-dieeni-17b-karboksamidi-3-karboksyylihapon polymorfin A valmistamiseksi FI114709B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB9206413 1992-03-24
GB929206413A GB9206413D0 (en) 1992-03-24 1992-03-24 N-t-butyl-androst-3,5-diene-17b-carboxamide-3-carboxylic acid polymorph a
US9302974 1993-03-24
PCT/US1993/002974 WO1993019081A1 (en) 1992-03-24 1993-03-24 N-T-BUTYL-ANDROST-3,5-DIENE-17β-CARBOXAMIDE-3-CARBOXYLIC ACID POLYMORPH A

Publications (3)

Publication Number Publication Date
FI944414A FI944414A (fi) 1994-09-23
FI944414A0 FI944414A0 (fi) 1994-09-23
FI114709B true FI114709B (fi) 2004-12-15

Family

ID=10712749

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944414A FI114709B (fi) 1992-03-24 1994-09-23 Menetelmä farmakologisesti aktiivisen N-t-butyyli-androst-3,5-dieeni-17b-karboksamidi-3-karboksyylihapon polymorfin A valmistamiseksi

Country Status (29)

Country Link
EP (1) EP0633892B1 (xx)
JP (1) JP2736169B2 (xx)
CN (1) CN1078723A (xx)
AP (1) AP403A (xx)
AT (1) ATE180490T1 (xx)
AU (1) AU669522B2 (xx)
BG (1) BG99062A (xx)
BR (1) BR9306139A (xx)
CA (1) CA2132535A1 (xx)
CZ (1) CZ286266B6 (xx)
DE (1) DE69325094T2 (xx)
DK (1) DK0633892T3 (xx)
ES (1) ES2134260T3 (xx)
FI (1) FI114709B (xx)
GB (1) GB9206413D0 (xx)
GR (1) GR3030779T3 (xx)
HU (1) HUT68120A (xx)
IL (1) IL105102A (xx)
MA (1) MA22841A1 (xx)
MX (1) MX9301656A (xx)
NO (1) NO943547D0 (xx)
NZ (1) NZ252008A (xx)
OA (1) OA10100A (xx)
PL (1) PL172523B1 (xx)
RU (1) RU94041839A (xx)
SI (1) SI9300140A (xx)
SK (1) SK113894A3 (xx)
WO (1) WO1993019081A1 (xx)
ZA (1) ZA932014B (xx)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4910226A (en) * 1987-04-29 1990-03-20 Smithkline Beckman Corporation Steroid 5-alpha-reductase inhibitors
IL104602A (en) * 1992-02-07 1997-07-13 Smithkline Beecham Corp Process for the preparation of 3-carbonylandrostadiene- 17-carboxamides and intermediates for this process

Also Published As

Publication number Publication date
CA2132535A1 (en) 1993-09-30
PL172523B1 (pl) 1997-10-31
JPH07505370A (ja) 1995-06-15
NZ252008A (en) 1996-06-25
ES2134260T3 (es) 1999-10-01
GR3030779T3 (en) 1999-11-30
ATE180490T1 (de) 1999-06-15
ZA932014B (en) 1994-09-22
BG99062A (en) 1995-08-28
AP403A (en) 1995-08-24
FI944414A (fi) 1994-09-23
SK113894A3 (en) 1995-04-12
MA22841A1 (fr) 1993-10-01
MX9301656A (es) 1994-02-28
NO943547L (no) 1994-09-23
GB9206413D0 (en) 1992-05-06
JP2736169B2 (ja) 1998-04-02
AU4044893A (en) 1993-10-21
IL105102A (en) 1997-02-18
FI944414A0 (fi) 1994-09-23
AP9300497A0 (en) 1993-04-30
EP0633892B1 (en) 1999-05-26
SI9300140A (en) 1993-09-30
NO943547D0 (no) 1994-09-23
IL105102A0 (en) 1994-08-26
AU669522B2 (en) 1996-06-13
HUT68120A (en) 1995-05-29
CZ231994A3 (en) 1995-01-18
BR9306139A (pt) 1998-06-23
EP0633892A4 (en) 1995-05-17
WO1993019081A1 (en) 1993-09-30
HU9402740D0 (en) 1994-12-28
DE69325094T2 (de) 1999-11-18
RU94041839A (ru) 1996-08-10
DK0633892T3 (da) 2000-04-10
CN1078723A (zh) 1993-11-24
CZ286266B6 (cs) 2000-03-15
EP0633892A1 (en) 1995-01-18
OA10100A (en) 1996-12-18
DE69325094D1 (de) 1999-07-01

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