MX9301656A - Polimorfo a de acido n-t-butil-androsta-3,5-dien-17(beta)-carboxiamido-3-carboxilico y procedimientos para su preparacion. - Google Patents

Polimorfo a de acido n-t-butil-androsta-3,5-dien-17(beta)-carboxiamido-3-carboxilico y procedimientos para su preparacion.

Info

Publication number
MX9301656A
MX9301656A MX9301656A MX9301656A MX9301656A MX 9301656 A MX9301656 A MX 9301656A MX 9301656 A MX9301656 A MX 9301656A MX 9301656 A MX9301656 A MX 9301656A MX 9301656 A MX9301656 A MX 9301656A
Authority
MX
Mexico
Prior art keywords
beta
butyl
carboxylic acid
procedures
androsta
Prior art date
Application number
MX9301656A
Other languages
English (en)
Inventor
Robert Lee Webb
Gary Edward Zuber
Neil Howard Baine
Neville Lewis Holder
Donald Nathaniel Kline
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of MX9301656A publication Critical patent/MX9301656A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Una forma polifórmica nueva Polimorfo 'A' de ácido N-t-butil-androst-3,5-dieno-17(beta)-carboxiamido- 3-carboxílico. También se describen procedimientos nuevos para preparar polimorfo 'A'.
MX9301656A 1992-03-24 1993-03-24 Polimorfo a de acido n-t-butil-androsta-3,5-dien-17(beta)-carboxiamido-3-carboxilico y procedimientos para su preparacion. MX9301656A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929206413A GB9206413D0 (en) 1992-03-24 1992-03-24 N-t-butyl-androst-3,5-diene-17b-carboxamide-3-carboxylic acid polymorph a

Publications (1)

Publication Number Publication Date
MX9301656A true MX9301656A (es) 1994-02-28

Family

ID=10712749

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9301656A MX9301656A (es) 1992-03-24 1993-03-24 Polimorfo a de acido n-t-butil-androsta-3,5-dien-17(beta)-carboxiamido-3-carboxilico y procedimientos para su preparacion.

Country Status (29)

Country Link
EP (1) EP0633892B1 (es)
JP (1) JP2736169B2 (es)
CN (1) CN1078723A (es)
AP (1) AP403A (es)
AT (1) ATE180490T1 (es)
AU (1) AU669522B2 (es)
BG (1) BG99062A (es)
BR (1) BR9306139A (es)
CA (1) CA2132535A1 (es)
CZ (1) CZ286266B6 (es)
DE (1) DE69325094T2 (es)
DK (1) DK0633892T3 (es)
ES (1) ES2134260T3 (es)
FI (1) FI114709B (es)
GB (1) GB9206413D0 (es)
GR (1) GR3030779T3 (es)
HU (1) HUT68120A (es)
IL (1) IL105102A (es)
MA (1) MA22841A1 (es)
MX (1) MX9301656A (es)
NO (1) NO943547L (es)
NZ (1) NZ252008A (es)
OA (1) OA10100A (es)
PL (1) PL172523B1 (es)
RU (1) RU94041839A (es)
SI (1) SI9300140A (es)
SK (1) SK113894A3 (es)
WO (1) WO1993019081A1 (es)
ZA (1) ZA932014B (es)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4910226A (en) * 1987-04-29 1990-03-20 Smithkline Beckman Corporation Steroid 5-alpha-reductase inhibitors
IL104602A (en) * 1992-02-07 1997-07-13 Smithkline Beecham Corp Process for the preparation of 3-carbonylandrostadiene- 17-carboxamides and intermediates for this process

Also Published As

Publication number Publication date
ATE180490T1 (de) 1999-06-15
ZA932014B (en) 1994-09-22
AU4044893A (en) 1993-10-21
DE69325094D1 (de) 1999-07-01
IL105102A (en) 1997-02-18
NZ252008A (en) 1996-06-25
CN1078723A (zh) 1993-11-24
HUT68120A (en) 1995-05-29
BR9306139A (pt) 1998-06-23
JPH07505370A (ja) 1995-06-15
MA22841A1 (fr) 1993-10-01
GB9206413D0 (en) 1992-05-06
AP9300497A0 (en) 1993-04-30
NO943547D0 (no) 1994-09-23
AU669522B2 (en) 1996-06-13
FI944414A (fi) 1994-09-23
OA10100A (en) 1996-12-18
IL105102A0 (en) 1994-08-26
EP0633892A1 (en) 1995-01-18
NO943547L (no) 1994-09-23
EP0633892B1 (en) 1999-05-26
RU94041839A (ru) 1996-08-10
CZ231994A3 (en) 1995-01-18
BG99062A (en) 1995-08-28
CA2132535A1 (en) 1993-09-30
EP0633892A4 (en) 1995-05-17
ES2134260T3 (es) 1999-10-01
FI944414A0 (fi) 1994-09-23
HU9402740D0 (en) 1994-12-28
JP2736169B2 (ja) 1998-04-02
SK113894A3 (en) 1995-04-12
DE69325094T2 (de) 1999-11-18
PL172523B1 (pl) 1997-10-31
CZ286266B6 (cs) 2000-03-15
SI9300140A (en) 1993-09-30
AP403A (en) 1995-08-24
WO1993019081A1 (en) 1993-09-30
GR3030779T3 (en) 1999-11-30
DK0633892T3 (da) 2000-04-10
FI114709B (fi) 2004-12-15

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