ES8503351A1 - Un procedimiento para preparar nuevos derivados de imidazo (4,5-c) piridina (como divisional de la solicitud de patente de invencion num. 517.193, presentada el 8 de noviembre de 1982) - Google Patents

Un procedimiento para preparar nuevos derivados de imidazo (4,5-c) piridina (como divisional de la solicitud de patente de invencion num. 517.193, presentada el 8 de noviembre de 1982)

Info

Publication number
ES8503351A1
ES8503351A1 ES523083A ES523083A ES8503351A1 ES 8503351 A1 ES8503351 A1 ES 8503351A1 ES 523083 A ES523083 A ES 523083A ES 523083 A ES523083 A ES 523083A ES 8503351 A1 ES8503351 A1 ES 8503351A1
Authority
ES
Spain
Prior art keywords
4alkyl
group
amino
compounds
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES523083A
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English (en)
Other versions
ES523083A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wellcome Foundation Ltd
Original Assignee
Wellcome Foundation Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Foundation Ltd filed Critical Wellcome Foundation Ltd
Publication of ES523083A0 publication Critical patent/ES523083A0/es
Publication of ES8503351A1 publication Critical patent/ES8503351A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE IMIDAZO 4,5-C PIRIDINA, DE FORMULA GENERAL (I), Y SUS SALES DE ADICION DE ACIDO FARMACEUTICAMENTE ACEPTABLES.CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA (II), A TEMPERATURA AMBIENTE O MEDIANTE CALENTAMIENTO, CON UN AGENTE OXIDANTE SELECCIONADO ENTRE PEROXIDO DE HIDROGENO, PERACIDOS ORGANICOS O BROMO.DE APLICACION COMO AGENTES CARDIOTONICOS, ESPECIALMENTE PARA EL TRATAMIENTO DE FALLOS CARDIACOS.
ES523083A 1981-11-10 1983-06-08 Un procedimiento para preparar nuevos derivados de imidazo (4,5-c) piridina (como divisional de la solicitud de patente de invencion num. 517.193, presentada el 8 de noviembre de 1982) Expired ES8503351A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB8133930 1981-11-10
GB8133942 1981-11-10
GB8213846 1982-05-12

Publications (2)

Publication Number Publication Date
ES523083A0 ES523083A0 (es) 1985-02-16
ES8503351A1 true ES8503351A1 (es) 1985-02-16

Family

ID=27261362

Family Applications (2)

Application Number Title Priority Date Filing Date
ES517193A Expired ES8401486A1 (es) 1981-11-10 1982-11-08 Un procedimiento para la preparacion de nuevos derivados de imidazo (4,5-c)piridina.
ES523083A Expired ES8503351A1 (es) 1981-11-10 1983-06-08 Un procedimiento para preparar nuevos derivados de imidazo (4,5-c) piridina (como divisional de la solicitud de patente de invencion num. 517.193, presentada el 8 de noviembre de 1982)

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES517193A Expired ES8401486A1 (es) 1981-11-10 1982-11-08 Un procedimiento para la preparacion de nuevos derivados de imidazo (4,5-c)piridina.

Country Status (17)

Country Link
US (1) US4603139A (es)
EP (1) EP0079083B1 (es)
KR (1) KR890000022B1 (es)
AR (1) AR241247A1 (es)
AU (1) AU9030682A (es)
DD (1) DD205904A5 (es)
DK (1) DK161325C (es)
ES (2) ES8401486A1 (es)
FI (1) FI79312C (es)
GB (1) GB2113675B (es)
GR (1) GR76746B (es)
IE (1) IE56478B1 (es)
IL (1) IL67206A0 (es)
MC (1) MC1491A1 (es)
NO (1) NO158100C (es)
PH (1) PH22764A (es)
PT (1) PT75820B (es)

Families Citing this family (78)

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DE3224512A1 (de) * 1982-07-01 1984-01-05 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazolderivate, ihre herstellung und diese verbindungen enthaltende arzneimittel
DE3324115A1 (de) * 1983-07-05 1985-01-17 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel
US4515796A (en) * 1983-09-08 1985-05-07 Eli Lilly And Company Certain naphthalenyl imidazo compounds and their pharmaceutical use
US4533734A (en) * 1983-11-10 1985-08-06 Eli Lilly And Company Inotropic agents
DE3346602A1 (de) * 1983-12-23 1985-07-11 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazo(4,5-c)pyridin-one, deren herstellung und diese verbindungen enthaltende arzneimittel
DE3347290A1 (de) * 1983-12-28 1985-07-11 Dr. Karl Thomae Gmbh, 7950 Biberach Neue 2-phenyl-imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel
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US4578387A (en) * 1984-03-05 1986-03-25 Eli Lilly And Company Inotropic agents
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US4740599A (en) * 1986-10-03 1988-04-26 Eli Lilly And Company Synthesis of alkylsulfinyl substituted 2-phenylimidazo(4,5-c)pyridines
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Also Published As

Publication number Publication date
GB2113675A (en) 1983-08-10
EP0079083A1 (en) 1983-05-18
ES523083A0 (es) 1985-02-16
FI823846A0 (fi) 1982-11-09
DK499582A (da) 1983-05-11
FI79312B (fi) 1989-08-31
DK161325B (da) 1991-06-24
IE56478B1 (en) 1991-08-14
ES517193A0 (es) 1983-12-01
AU9030682A (en) 1983-05-19
US4603139A (en) 1986-07-29
NO823732L (no) 1983-05-11
IE822667L (en) 1983-05-10
GR76746B (es) 1984-08-30
NO158100B (no) 1988-04-05
KR840002398A (ko) 1984-07-02
DD205904A5 (de) 1984-01-11
EP0079083B1 (en) 1991-02-27
NO158100C (no) 1988-07-13
PH22764A (en) 1988-12-12
MC1491A1 (fr) 1983-09-12
ES8401486A1 (es) 1983-12-01
FI79312C (fi) 1989-12-11
AR241247A1 (es) 1992-03-31
GB2113675B (en) 1985-10-30
FI823846L (fi) 1983-05-11
DK161325C (da) 1991-12-02
KR890000022B1 (ko) 1989-03-06
PT75820B (en) 1986-06-11
PT75820A (en) 1982-12-01
IL67206A0 (en) 1983-03-31

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