ES2927228T3 - Métodos de tratamiento del cáncer con inhibidores de farnesil transferasa - Google Patents
Métodos de tratamiento del cáncer con inhibidores de farnesil transferasa Download PDFInfo
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- ES2927228T3 ES2927228T3 ES19172562T ES19172562T ES2927228T3 ES 2927228 T3 ES2927228 T3 ES 2927228T3 ES 19172562 T ES19172562 T ES 19172562T ES 19172562 T ES19172562 T ES 19172562T ES 2927228 T3 ES2927228 T3 ES 2927228T3
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- UGGWPQSBPIFKDZ-KOTLKJBCSA-N vindesine Chemical compound C([C@@H](C[C@]1(C(=O)OC)C=2C(=CC3=C([C@]45[C@H]([C@@]([C@H](O)[C@]6(CC)C=CCN([C@H]56)CC4)(O)C(N)=O)N3C)C=2)OC)C[C@@](C2)(O)CC)N2CCC2=C1N=C1[C]2C=CC=C1 UGGWPQSBPIFKDZ-KOTLKJBCSA-N 0.000 description 1
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US201762507749P | 2017-05-17 | 2017-05-17 | |
| US201762519819P | 2017-06-14 | 2017-06-14 | |
| US15/820,157 US9956215B1 (en) | 2017-02-21 | 2017-11-21 | Methods of treating cancer with farnesyltransferase inhibitors |
| US15/820,012 US10137121B2 (en) | 2017-02-21 | 2017-11-21 | Methods of treating cancer with farnesyltransferase inhibitors |
| US201762596653P | 2017-12-08 | 2017-12-08 |
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| ES2927228T3 true ES2927228T3 (es) | 2022-11-03 |
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| ES18708563T Active ES2892157T3 (es) | 2017-02-21 | 2018-02-21 | Métodos de tratamiento del cáncer con inhibidores de farnesil transferasa |
Country Status (14)
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| EP (3) | EP3432883B1 (enExample) |
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| KR (3) | KR20200090982A (enExample) |
| CN (4) | CN109475550A (enExample) |
| AU (3) | AU2018225566B2 (enExample) |
| BR (1) | BR112019017375A2 (enExample) |
| CA (1) | CA3053795A1 (enExample) |
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| US9956215B1 (en) | 2017-02-21 | 2018-05-01 | Kura Oncology, Inc. | Methods of treating cancer with farnesyltransferase inhibitors |
| KR20200051601A (ko) * | 2017-08-07 | 2020-05-13 | 쿠라 온콜로지, 인크. | 파르네실전달효소 억제제를 이용하여 암을 치료하는 방법 |
| TW202108170A (zh) * | 2019-03-15 | 2021-03-01 | 美商庫拉腫瘤技術股份有限公司 | 以法呢基轉移酶(farnesyltransferase)抑制劑治療癌症患者之方法 |
| WO2025224720A1 (en) * | 2024-04-24 | 2025-10-30 | Biolinerx Ltd. | Methods of selecting treatment regimen against solid tumors |
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-
2018
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- 2018-02-21 CN CN201910346412.3A patent/CN109999037A/zh active Pending
- 2018-02-21 WO PCT/US2018/018989 patent/WO2018156609A1/en not_active Ceased
- 2018-02-21 CN CN202210399518.1A patent/CN114712354A/zh active Pending
- 2018-02-21 ES ES18708563T patent/ES2892157T3/es active Active
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2019
- 2019-05-21 AU AU2019203548A patent/AU2019203548C1/en active Active
- 2019-08-15 IL IL26872219A patent/IL268722A/en unknown
- 2019-08-16 MX MX2022008843A patent/MX2022008843A/es unknown
- 2019-08-19 PH PH12019501918A patent/PH12019501918A1/en unknown
- 2019-10-11 AU AU2019246922A patent/AU2019246922A1/en not_active Abandoned
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