ES2574927T3 - Piridinas bicíclicas y análogos como moduladores de sirtuina - Google Patents
Piridinas bicíclicas y análogos como moduladores de sirtuina Download PDFInfo
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- ES2574927T3 ES2574927T3 ES10830519.4T ES10830519T ES2574927T3 ES 2574927 T3 ES2574927 T3 ES 2574927T3 ES 10830519 T ES10830519 T ES 10830519T ES 2574927 T3 ES2574927 T3 ES 2574927T3
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- fluorine
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| PCT/US2010/054880 WO2011059839A1 (en) | 2009-10-29 | 2010-10-29 | Bicyclic pyridines and analogs as sirtuin modulators |
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| AU2009314631B2 (en) | 2008-11-12 | 2014-07-31 | Takeda Pharmaceutical Company Limited | Pyrazinopyrazines and derivatives as kinase inhibitors |
| KR20110098789A (ko) | 2008-12-08 | 2011-09-01 | 서트리스 파마슈티컬즈, 인코포레이티드 | 시르투인 조절제로서의 이소인돌리논 및 관련 유사체 |
| AU2009333251A1 (en) | 2008-12-16 | 2011-07-07 | Sirtris Pharmaceuticals, Inc. | Phthalazinone and related analogs as sirtuin modulators |
| CA2747715A1 (en) | 2008-12-19 | 2010-06-24 | Sirtris Pharmaceuticals, Inc. | Thiazolopyridine sirtuin modulating compounds |
| WO2010088574A1 (en) | 2009-01-30 | 2010-08-05 | Sirtris Pharmaceuticals, Inc. | Azabenzimidazoles and related analogs as sirtuin modulators |
| MX2011009213A (es) | 2009-03-02 | 2011-12-14 | Sirtris Pharmaceuticals Inc | Quinolinas 8-sustituidas y analogos relacionados como moduladores de sirtuina. |
| KR101820541B1 (ko) * | 2009-09-09 | 2018-02-28 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 8-옥소디히드로퓨린 유도체 |
| WO2011116176A1 (en) | 2010-03-17 | 2011-09-22 | Sirtris Pharmaceuticals Inc. | 3-substitued imidazo (4, 5-b) pyridines and analogs as sirtuin modulators |
-
2010
- 2010-10-29 WO PCT/US2010/054880 patent/WO2011059839A1/en not_active Ceased
- 2010-10-29 IN IN3799DEN2012 patent/IN2012DN03799A/en unknown
- 2010-10-29 MX MX2012004995A patent/MX2012004995A/es not_active Application Discontinuation
- 2010-10-29 AU AU2010319842A patent/AU2010319842A1/en not_active Abandoned
- 2010-10-29 CN CN201080060180.2A patent/CN102725291B/zh not_active Expired - Fee Related
- 2010-10-29 RU RU2012122065/04A patent/RU2550821C2/ru not_active IP Right Cessation
- 2010-10-29 JP JP2012537157A patent/JP2013509442A/ja not_active Ceased
- 2010-10-29 ES ES10830519.4T patent/ES2574927T3/es active Active
- 2010-10-29 CA CA2779303A patent/CA2779303A1/en not_active Abandoned
- 2010-10-29 KR KR1020127013635A patent/KR20120092141A/ko not_active Ceased
- 2010-10-29 BR BR112012010010A patent/BR112012010010A2/pt not_active IP Right Cessation
- 2010-10-29 US US13/504,134 patent/US9556201B2/en not_active Expired - Fee Related
- 2010-10-29 EP EP10830519.4A patent/EP2493888B1/en active Active
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2012
- 2012-04-23 IL IL219372A patent/IL219372A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2493888A1 (en) | 2012-09-05 |
| KR20120092141A (ko) | 2012-08-20 |
| AU2010319842A1 (en) | 2012-05-17 |
| CN102725291B (zh) | 2016-12-21 |
| RU2012122065A (ru) | 2013-12-10 |
| RU2550821C2 (ru) | 2015-05-20 |
| IL219372A0 (en) | 2012-06-28 |
| CA2779303A1 (en) | 2011-05-19 |
| MX2012004995A (es) | 2012-10-03 |
| EP2493888A4 (en) | 2013-05-01 |
| JP2013509442A (ja) | 2013-03-14 |
| BR112012010010A2 (pt) | 2018-03-20 |
| CN102725291A (zh) | 2012-10-10 |
| US20120252780A1 (en) | 2012-10-04 |
| IN2012DN03799A (Direct) | 2015-08-28 |
| WO2011059839A1 (en) | 2011-05-19 |
| EP2493888B1 (en) | 2016-04-06 |
| US9556201B2 (en) | 2017-01-31 |
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