ES2546671T3 - Pirazoles fungicidas - Google Patents
Pirazoles fungicidas Download PDFInfo
- Publication number
- ES2546671T3 ES2546671T3 ES11757463.2T ES11757463T ES2546671T3 ES 2546671 T3 ES2546671 T3 ES 2546671T3 ES 11757463 T ES11757463 T ES 11757463T ES 2546671 T3 ES2546671 T3 ES 2546671T3
- Authority
- ES
- Spain
- Prior art keywords
- alkyl
- formula
- meo
- independently
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US37915910P | 2010-09-01 | 2010-09-01 | |
| US379159P | 2010-09-01 | ||
| PCT/US2011/049908 WO2012030922A1 (en) | 2010-09-01 | 2011-08-31 | Fungicidal pyrazoles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2546671T3 true ES2546671T3 (es) | 2015-09-25 |
Family
ID=44651972
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES11757463.2T Active ES2546671T3 (es) | 2010-09-01 | 2011-08-31 | Pirazoles fungicidas |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US8754115B2 (https=) |
| EP (1) | EP2611297B1 (https=) |
| JP (1) | JP6066910B2 (https=) |
| KR (1) | KR20130139892A (https=) |
| CN (2) | CN105130900B (https=) |
| AR (1) | AR082869A1 (https=) |
| AU (1) | AU2011295998A1 (https=) |
| BR (2) | BR112013004835B1 (https=) |
| ES (1) | ES2546671T3 (https=) |
| MX (1) | MX2013002400A (https=) |
| PL (1) | PL2611297T3 (https=) |
| TW (1) | TW201245155A (https=) |
| UY (1) | UY33582A (https=) |
| WO (1) | WO2012030922A1 (https=) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR075713A1 (es) | 2009-03-03 | 2011-04-20 | Du Pont | Pirazoles fungicidas |
| TWI504350B (zh) | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
| TWI568721B (zh) | 2012-02-01 | 2017-02-01 | 杜邦股份有限公司 | 殺真菌之吡唑混合物 |
| US20140235689A1 (en) * | 2013-02-20 | 2014-08-21 | E I Du Pont De Nemours And Company | Fungicidal pyrazoles |
| JPWO2014157569A1 (ja) | 2013-03-28 | 2017-02-16 | 武田薬品工業株式会社 | 複素環化合物 |
| TWI652012B (zh) * | 2013-05-20 | 2019-03-01 | 杜邦股份有限公司 | 殺真菌吡唑的固態形式 |
| EP3036223A1 (en) | 2013-08-20 | 2016-06-29 | E. I. du Pont de Nemours and Company | Fungicidal pyrazoles |
| PL3078265T3 (pl) * | 2013-12-05 | 2017-10-31 | Kureha Corp | Substancja chemiczna do zastosowań rolniczych lub ogrodniczych, metoda ochrony roślin przed chorobami oraz produkt ochrony roślin przed chorobami |
| EP3078266A4 (en) | 2013-12-05 | 2016-11-23 | Kureha Corp | AGRICULTURAL OR HORTICULTURAL CHEMICAL, METHOD OF CONTROLLING PLANT DISEASES AND PLANT DISEASE CONTROL PRODUCT |
| WO2015089800A1 (en) | 2013-12-19 | 2015-06-25 | Eli Lilly And Company | Fluorophenyl pyrazol compounds |
| US20170037014A1 (en) * | 2014-05-06 | 2017-02-09 | E. I. Du Pont De Nemours And Company | Fungicidal pyrazoles |
| US10246420B2 (en) | 2014-07-24 | 2019-04-02 | Bayer Cropscience Aktiengesellschaft | Pyrazole derivatives |
| BR112017018140A2 (pt) | 2015-03-19 | 2018-04-10 | Du Pont | ?composto, composição fungicida e método de controle de doenças de plantas? |
| WO2016201662A1 (en) * | 2015-06-18 | 2016-12-22 | Eli Lilly And Company | Fluoropyridyl pyrazol compounds |
| EP3412658A1 (en) * | 2017-06-09 | 2018-12-12 | Solvay Sa | Processes for the manufacture of sulfur-substitued pyrazole derivatives |
| AU2020366425A1 (en) * | 2019-10-18 | 2022-04-21 | Fmc Corporation | Methods for the preparation of 5-Bromo-2-(3-chloro-pyridin-2-yl)-2H-pyrazole-3-carboxylic acid |
| EP3976591B1 (en) * | 2019-10-18 | 2023-04-19 | FMC Corporation | Methods for the preparation of 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylic acid |
| TW202241859A (zh) * | 2021-01-29 | 2022-11-01 | 美商富曼西公司 | 用於製備５－溴－２－（３－氯－吡啶－２－基）－２ｈ－吡唑－３－甲酸之方法 |
| CN120500474A (zh) * | 2023-01-09 | 2025-08-15 | 弗陆创新有限公司 | 制备3-卤甲基取代的1-甲基-1h-吡唑-4-碳腈及其衍生物及其中间体的新方法 |
| CN116606263B (zh) * | 2023-05-26 | 2025-06-13 | 青岛科技大学 | 一种含氟苯联噻唑双酯类化合物及其用途 |
| WO2025168620A1 (en) * | 2024-02-07 | 2025-08-14 | Bayer Aktiengesellschaft | Heteroaryl-substituted 4,5-dihydro-1h-2,4,5-oxadiazines as novel fungicides |
Family Cites Families (34)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2891855A (en) | 1954-08-16 | 1959-06-23 | Geigy Ag J R | Compositions and methods for influencing the growth of plants |
| US3235361A (en) | 1962-10-29 | 1966-02-15 | Du Pont | Method for the control of undesirable vegetation |
| US3060084A (en) | 1961-06-09 | 1962-10-23 | Du Pont | Improved homogeneous, readily dispersed, pesticidal concentrate |
| US3299566A (en) | 1964-06-01 | 1967-01-24 | Olin Mathieson | Water soluble film containing agricultural chemicals |
| US3309192A (en) | 1964-12-02 | 1967-03-14 | Du Pont | Method of controlling seedling weed grasses |
| US4144050A (en) | 1969-02-05 | 1979-03-13 | Hoechst Aktiengesellschaft | Micro granules for pesticides and process for their manufacture |
| US3920442A (en) | 1972-09-18 | 1975-11-18 | Du Pont | Water-dispersible pesticide aggregates |
| JPS5527916B2 (https=) | 1973-02-05 | 1980-07-24 | ||
| NL7512983A (nl) | 1974-11-06 | 1976-05-10 | Parke Davis & Co | Werkwijze voor het bereiden van diazepineverbin- dingen, werkwijze voor het bereiden van een far- maceutisch preparaat met toepassing daarvan als- mede een zo gevormd preparaat. |
| US4172714A (en) | 1976-12-20 | 1979-10-30 | E. I. Du Pont De Nemours And Company | Dry compactible, swellable herbicidal compositions and pellets produced therefrom |
| DE3246493A1 (de) | 1982-12-16 | 1984-06-20 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von wasserdispergierbaren granulaten |
| AU559935B2 (en) | 1983-02-04 | 1987-03-26 | Warner-Lambert Company | Imidazolyl-pyrazolyl methanone derivatives |
| JPS6253970A (ja) * | 1985-09-03 | 1987-03-09 | Nippon Nohyaku Co Ltd | ピラゾ−ル誘導体及びその製法 |
| US5180587A (en) | 1988-06-28 | 1993-01-19 | E. I. Du Pont De Nemours And Company | Tablet formulations of pesticides |
| DK0777964T3 (da) | 1989-08-30 | 2002-03-11 | Kynoch Agrochemicals Proprieta | Fremgangsmåde til fremstilling af et doseringssystem |
| JPH03141276A (ja) * | 1989-10-24 | 1991-06-17 | Nissan Chem Ind Ltd | 置換ピラゾール誘導体および農園芸用殺菌剤 |
| PL167613B1 (pl) | 1990-03-12 | 1995-09-30 | Du Pont | Granulowana kompozycja rozpuszczalna lub dyspergowalna w wodzie PL |
| US5189040A (en) * | 1990-05-28 | 1993-02-23 | Sumitomo Chemical Company, Limited | Pyrazole derivatives, method for producing the same and agricultural and/or horticultural fungicides containing the same as active ingredient |
| JPH04356480A (ja) * | 1990-05-28 | 1992-12-10 | Sumitomo Chem Co Ltd | ピラゾール誘導体、その製造法およびそれを有効成分とする農園芸用殺菌剤 |
| DE69122201T2 (de) | 1990-10-11 | 1997-02-06 | Sumitomo Chemical Co | Pestizide Zusammensetzung |
| JPH0532662A (ja) * | 1990-11-09 | 1993-02-09 | Nissan Chem Ind Ltd | 置換ピラゾール誘導体および農園芸用殺菌剤 |
| JPH0551304A (ja) | 1991-06-10 | 1993-03-02 | Nippon Bayeragrochem Kk | 除草剤組成物 |
| JPH05279339A (ja) * | 1992-01-22 | 1993-10-26 | Nissan Chem Ind Ltd | 置換ピラゾール誘導体および農園芸用殺菌剤 |
| JPH0665237A (ja) * | 1992-05-07 | 1994-03-08 | Nissan Chem Ind Ltd | 置換ピラゾール誘導体および農園芸用殺菌剤 |
| EP0822187A4 (en) * | 1995-02-07 | 1998-05-13 | Nissan Chemical Ind Ltd | PYRAZOLE DERIVATIVES AS HERBICIDES |
| JP2865599B2 (ja) | 1995-10-09 | 1999-03-08 | 株式会社横井製作所 | 埋設物の探査方法 |
| DE10136065A1 (de) | 2001-07-25 | 2003-02-13 | Bayer Cropscience Ag | Pyrazolylcarboxanilide |
| TWI283164B (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| JP2009541321A (ja) | 2006-06-21 | 2009-11-26 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 細胞増殖阻害剤としてのピラジノン |
| GB0713479D0 (en) | 2007-07-11 | 2007-08-22 | Syngenta Participations Ag | Substituted aromatic heterocyclic compounds as fungicides |
| PE20091953A1 (es) * | 2008-05-08 | 2010-01-09 | Du Pont | Azoles sustituidos como fungicidas |
| AR075713A1 (es) | 2009-03-03 | 2011-04-20 | Du Pont | Pirazoles fungicidas |
| WO2012023143A1 (en) | 2010-08-19 | 2012-02-23 | E. I. Du Pont De Nemours And Company | Fungicidal pyrazoles |
| TWI504350B (zh) | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
-
2011
- 2011-08-26 TW TW100130635A patent/TW201245155A/zh unknown
- 2011-08-31 US US13/816,847 patent/US8754115B2/en not_active Expired - Fee Related
- 2011-08-31 EP EP11757463.2A patent/EP2611297B1/en not_active Not-in-force
- 2011-08-31 JP JP2013527253A patent/JP6066910B2/ja not_active Expired - Fee Related
- 2011-08-31 PL PL11757463T patent/PL2611297T3/pl unknown
- 2011-08-31 ES ES11757463.2T patent/ES2546671T3/es active Active
- 2011-08-31 MX MX2013002400A patent/MX2013002400A/es not_active Application Discontinuation
- 2011-08-31 BR BR112013004835-2A patent/BR112013004835B1/pt not_active IP Right Cessation
- 2011-08-31 CN CN201510578968.7A patent/CN105130900B/zh not_active Expired - Fee Related
- 2011-08-31 UY UY33582A patent/UY33582A/es not_active Application Discontinuation
- 2011-08-31 BR BR122017015898-8A patent/BR122017015898B1/pt not_active IP Right Cessation
- 2011-08-31 CN CN201180042397.5A patent/CN103079406B/zh not_active Expired - Fee Related
- 2011-08-31 KR KR20137008060A patent/KR20130139892A/ko not_active Withdrawn
- 2011-08-31 WO PCT/US2011/049908 patent/WO2012030922A1/en not_active Ceased
- 2011-08-31 AU AU2011295998A patent/AU2011295998A1/en not_active Abandoned
- 2011-09-01 AR ARP110103199 patent/AR082869A1/es unknown
-
2014
- 2014-04-10 US US14/249,658 patent/US9131693B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| UY33582A (es) | 2012-03-30 |
| BR122017015898B1 (pt) | 2018-05-15 |
| CN103079406A (zh) | 2013-05-01 |
| EP2611297A1 (en) | 2013-07-10 |
| CN103079406B (zh) | 2016-03-30 |
| JP2013536856A (ja) | 2013-09-26 |
| KR20130139892A (ko) | 2013-12-23 |
| AU2011295998A1 (en) | 2013-02-21 |
| AR082869A1 (es) | 2013-01-16 |
| TW201245155A (en) | 2012-11-16 |
| CN105130900A (zh) | 2015-12-09 |
| PL2611297T3 (pl) | 2015-11-30 |
| CN105130900B (zh) | 2018-05-22 |
| BR112013004835B1 (pt) | 2018-01-09 |
| EP2611297B1 (en) | 2015-06-17 |
| US9131693B2 (en) | 2015-09-15 |
| JP6066910B2 (ja) | 2017-01-25 |
| US20140221448A1 (en) | 2014-08-07 |
| US20130143940A1 (en) | 2013-06-06 |
| US8754115B2 (en) | 2014-06-17 |
| WO2012030922A1 (en) | 2012-03-08 |
| MX2013002400A (es) | 2013-06-05 |
| BR112013004835A2 (pt) | 2016-05-31 |
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